PT75240B - Process for the preparation of substituted thiazolo <3,2-a>pyrimidines - Google Patents

Process for the preparation of substituted thiazolo <3,2-a>pyrimidines

Info

Publication number: PT75240B
Authority: PT; Portugal
Prior art keywords: pyrimidines; preparation; substituted thiazolo; thiazolo; substituted
Prior art date: 1981-07-15

Application number

PT75240A

Other languages

English (en)

Other versions

PT75240A (en

Inventor

Gianfederico Doria

Carlo Passarotti

Giuliana Arcari

Ada Buttinoni

Original Assignee

Erba Farmitalia

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1981-07-15

Filing date

1982-07-13

Publication date

1984-07-23

1982-07-13 Application filed by Erba Farmitalia filed Critical Erba Farmitalia

1982-08-01 Publication of PT75240A publication Critical patent/PT75240A/pt

1984-07-23 Publication of PT75240B publication Critical patent/PT75240B/pt

Links

150000003230 pyrimidines Chemical class 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Biochemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Molecular Biology (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pain & Pain Management (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Rheumatology (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

PT75240A 1981-07-15 1982-07-13 Process for the preparation of substituted thiazolo <3,2-a>pyrimidines PT75240B (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
GB8121979		1981-07-15
GB8201621		1982-01-20
GB8212430		1982-04-29

Publications (2)

Publication Number	Publication Date
PT75240A PT75240A (en)	1982-08-01
PT75240B true PT75240B (en)	1984-07-23

Family

ID=27261230

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT75240A PT75240B (en)	1981-07-15	1982-07-13	Process for the preparation of substituted thiazolo <3,2-a>pyrimidines

Country Status (25)

Country	Link
US (2)	US4444773A (pt)
KR (1)	KR880002301B1 (pt)
AT (1)	AT384614B (pt)
AU (1)	AU551718B2 (pt)
CA (1)	CA1208635A (pt)
CH (1)	CH653036A5 (pt)
DE (1)	DE3226516A1 (pt)
DK (1)	DK156222C (pt)
ES (2)	ES8307827A1 (pt)
FI (1)	FI71940C (pt)
FR (1)	FR2509734B1 (pt)
GB (1)	GB2103608B (pt)
GR (1)	GR76208B (pt)
HU (1)	HU186951B (pt)
IE (1)	IE53426B1 (pt)
IL (1)	IL66316A (pt)
IT (1)	IT1190914B (pt)
LU (1)	LU84262A1 (pt)
NL (1)	NL8202706A (pt)
NO (1)	NO822441L (pt)
NZ (1)	NZ201194A (pt)
PT (1)	PT75240B (pt)
SE (2)	SE453295B (pt)
SU (1)	SU1358786A3 (pt)
YU (1)	YU151582A (pt)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU551718B2 (en) *	1981-07-15	1986-05-08	Farmitalia Carlo Erba S.P.A.	Substituted thiazolo(3,2-alpha)pyrimidines
US4537962A (en) *	1982-02-04	1985-08-27	Farmitalia Carlo Erba, S.P.A.	Substituted 1,3,4-thiadiazolo[3,2-A]pyrimidines and compositions containing them
US4546101A (en) *	1982-09-10	1985-10-08	Fujisawa Pharmaceutical Co., Ltd.	New cephem compounds useful for treating infectious diseases in human being and animals and processes for preparation thereof
GB8300728D0 (en) *	1983-01-12	1983-02-16	Erba Farmitalia	Substituted carboxy-thiazolo / 3 2 - a / pyrimidine derivatives
DE10112197A1 (de) *	2001-03-14	2002-09-19	Gruenenthal Gmbh	Substituierte Pyrazolo- und Thiazolopyrimidine
MX2010005769A (es) *	2008-01-11	2010-11-12	Glenmark Pharmaceuticals Sa	Derivados de pirimidina fusionados como moduladores del trpv3.
US8119647B2 (en) *	2008-04-23	2012-02-21	Glenmark Pharmaceuticals S.A.	Fused pyrimidineone compounds as TRPV3 modulators
CA2729649A1 (en) *	2008-07-02	2010-01-07	Avexa Limited	Thiazopyrimidinones and uses thereof
CN106916168B (zh) *	2017-03-13	2019-08-27	牡丹江医学院	一种治疗重症胰腺炎的化合物及其制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3594378A (en) *	1969-10-24	1971-07-20	Ayerst Mckenna & Harrison	Thiazolopyrimidine derivatives and preparation thereof
US3888983A (en) *	1970-08-14	1975-06-10	Seperic	Derivatives of thiazolino-pyrimidin-6-ones, in inducing analgesia
GB2084568A (en) *	1980-08-16	1982-04-15	Beecham Group Ltd	Imidazothiazole derivatives
AU551718B2 (en) *	1981-07-15	1986-05-08	Farmitalia Carlo Erba S.P.A.	Substituted thiazolo(3,2-alpha)pyrimidines

1982
- 1982-07-06 AU AU85648/82A patent/AU551718B2/en not_active Ceased
- 1982-07-06 NL NL8202706A patent/NL8202706A/nl not_active Application Discontinuation
- 1982-07-07 LU LU84262A patent/LU84262A1/xx unknown
- 1982-07-07 NZ NZ201194A patent/NZ201194A/en unknown
- 1982-07-08 AT AT0266182A patent/AT384614B/de not_active IP Right Cessation
- 1982-07-08 ES ES513808A patent/ES8307827A1/es not_active Expired
- 1982-07-12 FI FI822468A patent/FI71940C/fi not_active IP Right Cessation
- 1982-07-12 SE SE8204292A patent/SE453295B/sv not_active IP Right Cessation
- 1982-07-12 IT IT22353/82A patent/IT1190914B/it active
- 1982-07-12 YU YU01515/82A patent/YU151582A/xx unknown
- 1982-07-12 SE SE8204292D patent/SE8204292L/xx not_active Application Discontinuation
- 1982-07-13 CH CH4272/82A patent/CH653036A5/de not_active IP Right Cessation
- 1982-07-13 SU SU823466583A patent/SU1358786A3/ru active
- 1982-07-13 PT PT75240A patent/PT75240B/pt unknown
- 1982-07-14 DK DK314682A patent/DK156222C/da not_active IP Right Cessation
- 1982-07-14 HU HU822289A patent/HU186951B/hu not_active IP Right Cessation
- 1982-07-14 GR GR68755A patent/GR76208B/el unknown
- 1982-07-14 US US06/398,302 patent/US4444773A/en not_active Expired - Fee Related
- 1982-07-14 CA CA000407223A patent/CA1208635A/en not_active Expired
- 1982-07-14 NO NO822441A patent/NO822441L/no unknown
- 1982-07-14 GB GB08220385A patent/GB2103608B/en not_active Expired
- 1982-07-14 IE IE1692/82A patent/IE53426B1/en unknown
- 1982-07-14 IL IL66316A patent/IL66316A/xx unknown
- 1982-07-15 FR FR8212391A patent/FR2509734B1/fr not_active Expired
- 1982-07-15 KR KR8203145A patent/KR880002301B1/ko active
- 1982-07-15 DE DE19823226516 patent/DE3226516A1/de not_active Ceased
1983
- 1983-03-16 ES ES520642A patent/ES520642A0/es active Granted
1984
- 1984-05-30 US US06/615,346 patent/US4551457A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
SU1358786A3 (ru)	1987-12-07
SE8204292D0 (sv)	1982-07-12
IE53426B1 (en)	1988-11-09
IT8222353A0 (it)	1982-07-12
IT1190914B (it)	1988-02-24
KR840000569A (ko)	1984-02-25
IT8222353A1 (it)	1984-01-12
AU551718B2 (en)	1986-05-08
FR2509734A1 (fr)	1983-01-21
KR880002301B1 (ko)	1988-10-22
DK156222C (da)	1989-12-04
LU84262A1 (fr)	1983-02-07
IL66316A0 (en)	1982-11-30
IE821692L (en)	1983-01-15
DK314682A (da)	1983-01-16
NO822441L (no)	1983-01-17
FI822468A0 (fi)	1982-07-12
US4444773A (en)	1984-04-24
FI822468L (fi)	1983-01-16
FI71940C (fi)	1987-03-09
IL66316A (en)	1986-04-29
AU8564882A (en)	1983-01-20
NL8202706A (nl)	1983-02-01
PT75240A (en)	1982-08-01
AT384614B (de)	1987-12-10
ATA266182A (de)	1987-05-15
GB2103608B (en)	1985-01-30
DK156222B (da)	1989-07-10
SE453295B (sv)	1988-01-25
GB2103608A (en)	1983-02-23
ES8404363A1 (es)	1984-05-01
US4551457A (en)	1985-11-05
ES520642A0 (es)	1984-05-01
ES513808A0 (es)	1983-08-01
FR2509734B1 (fr)	1985-07-19
SE8204292L (sv)	1983-03-14
YU151582A (en)	1985-04-30
ES8307827A1 (es)	1983-08-01
FI71940B (fi)	1986-11-28
DE3226516A1 (de)	1983-02-03
CH653036A5 (de)	1985-12-13
NZ201194A (en)	1985-02-28
CA1208635A (en)	1986-07-29
HU186951B (en)	1985-10-28
GR76208B (pt)	1984-08-03

Publication	Publication Date	Title
DE3260183D1 (en)	1984-07-05	Process for the preparation of alpha-alkyl acroleines
PT75247A (en)	1982-08-01	Novel bicyclic pyrimidin-5-one derivatives
HRP930089B1 (en)	1996-12-31	PROCESS FOR THE PREPARATION OF SPS-aze
AU8752482A (en)	1983-03-03	Imidazo (1,2-a)quinazolin-2-ones
PT75240A (en)	1982-08-01	Process for the preparation of substituted thiazolo <3,2-a>pyrimidines
AU8187482A (en)	1982-09-30	Imidazo(1,2-a)pyrimidine derivatives
PT71197A (en)	1980-06-01	Process for the preparation of substituted pyrido/1,2-a/pyrimidines
RO83114B (ro)	1984-02-28	Procedeu pentru prepararea ditiazolil-(2, 2')-disulfurilor
PT77258B (en)	1986-03-21	Process for preparing new imidazo/1,2-a/pyrimidines
DE3261387D1 (en)	1985-01-10	Process for the preparation of 3-alkyl-3-acyloxy-4-hydroxybutenes
GB2114129B (en)	1985-05-15	Substituted 1,3,4-thiadiazolo(3,2-a) pyrimidines and process for their preparation
DE3266652D1 (en)	1985-11-07	Process for the preparation of 2-alkoxy-(1,3)-dioxolanes
PT74339B (en)	1983-07-04	Process for the preparation of alpha-haloalkylamides
YU135182A (en)	1986-04-30	Process for preparing new imidazo(1,2-a)pyrimidines
DE3265814D1 (en)	1985-10-03	Process for the preparation of halogeno-2-mercaptobenzoxazoles
GB2111471B (en)	1985-09-25	Process for the preparation of acicular -feooh
ZA824619B (en)	1983-04-27	Process for the preparation of 5,6,7,7a-tetrahydro-4h-thieno(3,2-c)pyridin-2-ones
ZA824797B (en)	1983-04-27	Substituted thiazolo(3,2-a)pyrimidines and process for their preparation
DE3263745D1 (en)	1985-06-27	Process for the preparation of 4-aminobutyramide
DE3260205D1 (en)	1984-07-12	Process for the preparation of 2-chloro-4-nitrotoluene
DE3262828D1 (en)	1985-05-02	Process for the preparation of 1,2-benzisothiazolin-3-ones
DE3263730D1 (en)	1985-06-27	Process for the preparation of dihydroxypropyltheophylline
ZA825018B (en)	1984-02-29	Novel bicyclic pyrimidin-5-one derivatives
IL66819A0 (en)	1982-12-31	Process for the preparation of macrophages-activating-factor
DE3260366D1 (en)	1984-08-16	Process for the preparation of 4,7-dichloro-3-hydroxy-thionaphthene