PT65164B - PROCESS FOR THE PREPARATION OF NEW SUBSTITUTED BENZAMIDES AND THEIR DERIVATIVES - Google Patents

PROCESS FOR THE PREPARATION OF NEW SUBSTITUTED BENZAMIDES AND THEIR DERIVATIVES

Info

Publication number
PT65164B
PT65164B PT65164A PT6516476A PT65164B PT 65164 B PT65164 B PT 65164B PT 65164 A PT65164 A PT 65164A PT 6516476 A PT6516476 A PT 6516476A PT 65164 B PT65164 B PT 65164B
Authority
PT
Portugal
Prior art keywords
derivatives
preparation
new substituted
substituted benzamides
benzamides
Prior art date
Application number
PT65164A
Other languages
French (fr)
Portuguese (pt)
Other versions
PT65164A (en
Original Assignee
Ile De France
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ile De France filed Critical Ile De France
Publication of PT65164A publication Critical patent/PT65164A/en
Publication of PT65164B publication Critical patent/PT65164B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D207/00Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C07D207/09Radicals substituted by nitrogen atoms, not forming part of a nitro radical

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Otolaryngology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrrole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
PT65164A 1975-06-10 1976-06-01 PROCESS FOR THE PREPARATION OF NEW SUBSTITUTED BENZAMIDES AND THEIR DERIVATIVES PT65164B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7518001A FR2313935A1 (en) 1975-06-10 1975-06-10 NEW BENZAMIDES SUBSTITUTES, THEIR DERIVATIVES AND THEIR PREPARATION PROCESS

Publications (2)

Publication Number Publication Date
PT65164A PT65164A (en) 1976-07-01
PT65164B true PT65164B (en) 1977-11-17

Family

ID=9156239

Family Applications (1)

Application Number Title Priority Date Filing Date
PT65164A PT65164B (en) 1975-06-10 1976-06-01 PROCESS FOR THE PREPARATION OF NEW SUBSTITUTED BENZAMIDES AND THEIR DERIVATIVES

Country Status (37)

Country Link
JP (1) JPS6055503B2 (en)
AR (1) AR210888A1 (en)
AT (1) AT358571B (en)
AU (1) AU506001B2 (en)
BE (1) BE842059A (en)
BG (1) BG27360A3 (en)
CA (1) CA1064930A (en)
CH (1) CH596175A5 (en)
CS (1) CS189007B2 (en)
DD (1) DD124380A5 (en)
DE (1) DE2623075A1 (en)
DK (1) DK255276A (en)
EG (1) EG12285A (en)
ES (1) ES448643A1 (en)
FI (1) FI761669A (en)
FR (1) FR2313935A1 (en)
GB (1) GB1500105A (en)
HK (1) HK46979A (en)
HU (1) HU172195B (en)
IE (1) IE43375B1 (en)
IN (1) IN142899B (en)
LU (1) LU75104A1 (en)
MW (1) MW1676A1 (en)
MX (1) MX3580E (en)
NL (1) NL186382C (en)
NO (1) NO146058C (en)
NZ (1) NZ181072A (en)
OA (1) OA05350A (en)
PH (1) PH13912A (en)
PL (2) PL103075B1 (en)
PT (1) PT65164B (en)
RO (1) RO70265A (en)
SE (1) SE415971B (en)
SU (2) SU607551A3 (en)
YU (1) YU39352B (en)
ZA (1) ZA763042B (en)
ZM (1) ZM6576A1 (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ186175A (en) * 1977-01-27 1980-03-05 Shionogi & Co Meta-sulphonamidobenzamide derivatives
FR2415099A1 (en) * 1978-01-20 1979-08-17 Ile De France NEW DERIVATIVES OF 4-AMINO-5-ALKYLSULFONYL ORTHO-ANISAMIDES, THEIR METHODS OF PREPARATION AND THEIR APPLICATION AS PSYCHOTROPES
FR2438650A1 (en) * 1978-10-11 1980-05-09 Ile De France N- (1-METHYL 2-PYRROLIDINYL METHYL) 2,3-DIMETHOXY 5-METHYLSULFAMOYL BENZAMIDE AND DERIVATIVES THEREOF, THEIR PREPARATION METHODS AND THEIR APPLICATION IN THE TREATMENT OF LOWER URINARY DISORDERS
JPS597160A (en) * 1982-06-28 1984-01-14 ラボラトリーオス・デラグランヘ・エセ・ア N-(1-propyl-2-pyrrolidinylmethyl)-2-methoxy-5- sulfamoylbenzamide, manufacture and antidepressive
US4808624A (en) * 1984-06-28 1989-02-28 Bristol-Myers Company Pharmacologically active substituted benzamides
US4820715A (en) * 1984-06-28 1989-04-11 Bristol-Myers Company Anti-emetic quinuclidinyl benzamides
US5011992A (en) * 1984-06-28 1991-04-30 Bristol-Myers Squibb Company Pharmacologically active substituted benzamides
JP3026845B2 (en) * 1991-02-20 2000-03-27 日清製粉株式会社 Piperidine derivative
EP2895457B1 (en) 2012-09-17 2020-05-20 Nektar Therapeutics Oligomer-containing benzamide-based compounds

Also Published As

Publication number Publication date
AT358571B (en) 1980-09-25
GB1500105A (en) 1978-02-08
HU172195B (en) 1978-06-28
SU607551A3 (en) 1978-05-15
CS189007B2 (en) 1979-03-30
DE2623075A1 (en) 1976-12-30
BG27360A3 (en) 1979-10-12
IN142899B (en) 1977-09-03
ES448643A1 (en) 1977-07-01
LU75104A1 (en) 1977-03-09
PT65164A (en) 1976-07-01
HK46979A (en) 1979-07-20
NZ181072A (en) 1978-07-28
DD124380A5 (en) 1977-02-16
PL102929B1 (en) 1979-05-31
SE7606424L (en) 1976-12-11
RO70265A (en) 1981-06-30
OA05350A (en) 1981-02-28
FR2313935A1 (en) 1977-01-07
AR210888A1 (en) 1977-09-30
CH596175A5 (en) 1978-02-28
PH13912A (en) 1980-11-04
FR2313935B1 (en) 1979-04-27
NL186382C (en) 1990-11-16
SE415971B (en) 1980-11-17
PL103075B1 (en) 1979-05-31
PL190247A1 (en) 1978-03-13
DK255276A (en) 1976-12-11
NL7606284A (en) 1976-12-14
ZA763042B (en) 1977-04-27
ZM6576A1 (en) 1977-06-21
BE842059A (en) 1976-11-22
IE43375B1 (en) 1981-02-11
SU645557A3 (en) 1979-01-30
AU506001B2 (en) 1979-12-13
NO146058B (en) 1982-04-13
EG12285A (en) 1978-09-30
MX3580E (en) 1981-03-19
NL186382B (en) 1990-06-18
CA1064930A (en) 1979-10-23
YU131876A (en) 1982-06-30
IE43375L (en) 1976-12-10
NO146058C (en) 1982-07-28
NO761977L (en) 1976-12-13
JPS6055503B2 (en) 1985-12-05
ATA400176A (en) 1980-02-15
FI761669A (en) 1976-12-11
AU1436076A (en) 1977-12-01
YU39352B (en) 1984-10-31
JPS5231041A (en) 1977-03-09
MW1676A1 (en) 1977-10-12

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