PT2007391E - Combinação compreendendo: a) um composto de pirimidil-aminobenzamida e b) um inibidor da cinase thr315ile - Google Patents
Combinação compreendendo: a) um composto de pirimidil-aminobenzamida e b) um inibidor da cinase thr315ileInfo
- Publication number
- PT2007391E PT2007391E PT77278810T PT07727881T PT2007391E PT 2007391 E PT2007391 E PT 2007391E PT 77278810 T PT77278810 T PT 77278810T PT 07727881 T PT07727881 T PT 07727881T PT 2007391 E PT2007391 E PT 2007391E
- Authority
- PT
- Portugal
- Prior art keywords
- thr315lle
- combination
- kinase inhibitor
- pyrimidylaminobenzamide compound
- pyrimidylaminobenzamide
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Dermatology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US79043806P | 2006-04-07 | 2006-04-07 | |
US79115006P | 2006-04-11 | 2006-04-11 |
Publications (1)
Publication Number | Publication Date |
---|---|
PT2007391E true PT2007391E (pt) | 2013-03-11 |
Family
ID=38229305
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT77278810T PT2007391E (pt) | 2006-04-07 | 2007-04-05 | Combinação compreendendo: a) um composto de pirimidil-aminobenzamida e b) um inibidor da cinase thr315ile |
Country Status (13)
Country | Link |
---|---|
US (1) | US20090286803A1 (pt) |
EP (2) | EP2574340A3 (pt) |
JP (2) | JP2009532440A (pt) |
KR (1) | KR20090023561A (pt) |
AU (1) | AU2007235900A1 (pt) |
BR (1) | BRPI0710496A2 (pt) |
CA (1) | CA2647803C (pt) |
ES (1) | ES2400375T3 (pt) |
MX (1) | MX2008012971A (pt) |
PL (1) | PL2007391T3 (pt) |
PT (1) | PT2007391E (pt) |
RU (2) | RU2481840C2 (pt) |
WO (1) | WO2007116029A2 (pt) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BRPI0810028A2 (pt) * | 2007-04-17 | 2014-10-21 | Novartis Ag | Éteres de amidas de ácido naftaleno carboxílico no tratamento de câncer |
JO3265B1 (ar) | 2008-12-09 | 2018-09-16 | Novartis Ag | مثبطات بيريديلوكسى اندولات vegf-r2 واستخدامها لعلاج المرض |
JP2013509444A (ja) * | 2009-10-30 | 2013-03-14 | アリアド・ファーマシューティカルズ・インコーポレイテッド | がんの治療方法及び治療用組成物 |
CN102822141A (zh) * | 2010-01-20 | 2012-12-12 | 普罗诺瓦生物医药挪威公司 | 水杨酸脂肪酸衍生物 |
CN109730996B (zh) * | 2017-03-01 | 2021-08-24 | 浙江大学 | 喹啉结构类型雄激素受体拮抗剂及其应用 |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL156368A0 (en) | 2000-12-21 | 2004-01-04 | Vertex Pharma | Pyrazole derivatives and pharmaceutical compositions containing the same |
CA2459822C (en) * | 2001-09-05 | 2013-01-29 | Jean-Pierre Robin | Treatment of chronic myelogenous leukemia, resistant or intolerant to sti571, involving homoharringtonine alone or combined with other agents |
WO2003047523A2 (en) * | 2001-12-04 | 2003-06-12 | Onyx Pharmaceuticals, Inc. | Raf-mek-erk pathway inhibitors to treat cancer |
AR037647A1 (es) | 2002-05-29 | 2004-12-01 | Novartis Ag | Derivados de diarilurea utiles para el tratamiento de enfermedades dependientes de la cinasa de proteina |
FR2841116B1 (fr) | 2002-06-19 | 2004-11-26 | Seb Sa | Cafetiere du type expresso a reservoir d'eau amovible |
GB0215676D0 (en) * | 2002-07-05 | 2002-08-14 | Novartis Ag | Organic compounds |
WO2004026234A2 (en) * | 2002-09-19 | 2004-04-01 | University Of South Florida | Method of treating leukemia with a combination of suberoylanilide hydromaxic acid and imatinib mesylate |
DE10330916A1 (de) | 2003-07-04 | 2005-02-03 | Pilz Gmbh & Co. Kg | Vorrichtung und Verfahren zum automatisierten Steuern eines Betriebsablaufs bei einer technischen Anlage |
US7338957B2 (en) | 2003-08-28 | 2008-03-04 | Irm Llc | Compounds and compositions as protein kinase inhibitors |
EP1758892B1 (en) | 2004-06-10 | 2012-10-17 | Irm Llc | Compounds and compositions as protein kinase inhibitors |
KR20070050918A (ko) * | 2004-07-02 | 2007-05-16 | 뉴텍 파마 피엘씨 | 암의 치료 |
PE20060664A1 (es) | 2004-09-15 | 2006-08-04 | Novartis Ag | Amidas biciclicas como inhibidores de cinasa |
GB0421525D0 (en) * | 2004-09-28 | 2004-10-27 | Novartis Ag | Inhibitors of protein kineses |
US20070161645A1 (en) * | 2005-11-02 | 2007-07-12 | Targegen, Inc. | Thiazole inhibitors targeting resistant kinase mutations |
-
2007
- 2007-04-05 JP JP2009503595A patent/JP2009532440A/ja active Pending
- 2007-04-05 PL PL07727881T patent/PL2007391T3/pl unknown
- 2007-04-05 BR BRPI0710496-0A patent/BRPI0710496A2/pt not_active IP Right Cessation
- 2007-04-05 EP EP12197654.2A patent/EP2574340A3/en not_active Withdrawn
- 2007-04-05 KR KR1020087027200A patent/KR20090023561A/ko not_active Application Discontinuation
- 2007-04-05 MX MX2008012971A patent/MX2008012971A/es active IP Right Grant
- 2007-04-05 WO PCT/EP2007/053413 patent/WO2007116029A2/en active Application Filing
- 2007-04-05 ES ES07727881T patent/ES2400375T3/es active Active
- 2007-04-05 RU RU2008143704/15A patent/RU2481840C2/ru not_active IP Right Cessation
- 2007-04-05 PT PT77278810T patent/PT2007391E/pt unknown
- 2007-04-05 EP EP07727881.0A patent/EP2007391B8/en not_active Not-in-force
- 2007-04-05 AU AU2007235900A patent/AU2007235900A1/en not_active Abandoned
- 2007-04-05 US US12/295,812 patent/US20090286803A1/en not_active Abandoned
- 2007-04-05 CA CA2647803A patent/CA2647803C/en not_active Expired - Fee Related
-
2013
- 2013-01-29 RU RU2013103746/15A patent/RU2013103746A/ru unknown
- 2013-06-05 JP JP2013119191A patent/JP2013224304A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
RU2013103746A (ru) | 2014-08-10 |
ES2400375T8 (es) | 2013-09-10 |
PL2007391T3 (pl) | 2013-05-31 |
ES2400375T3 (es) | 2013-04-09 |
JP2009532440A (ja) | 2009-09-10 |
EP2007391B8 (en) | 2013-05-29 |
KR20090023561A (ko) | 2009-03-05 |
MX2008012971A (es) | 2008-10-15 |
WO2007116029A2 (en) | 2007-10-18 |
CA2647803A1 (en) | 2007-10-18 |
EP2574340A3 (en) | 2013-04-17 |
CA2647803C (en) | 2014-05-27 |
EP2007391A2 (en) | 2008-12-31 |
US20090286803A1 (en) | 2009-11-19 |
JP2013224304A (ja) | 2013-10-31 |
RU2008143704A (ru) | 2010-05-20 |
WO2007116029A3 (en) | 2008-12-11 |
EP2007391B1 (en) | 2012-12-19 |
RU2481840C2 (ru) | 2013-05-20 |
EP2574340A2 (en) | 2013-04-03 |
AU2007235900A1 (en) | 2007-10-18 |
BRPI0710496A2 (pt) | 2011-08-16 |
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