PT1532105E - Derivados de antracilo possuindo uma actividade anticolecistoquinina (anti-cck-1), um processo para a sua preparação e sua utilização farmacêutica - Google Patents

Derivados de antracilo possuindo uma actividade anticolecistoquinina (anti-cck-1), um processo para a sua preparação e sua utilização farmacêutica Download PDF

Info

Publication number
PT1532105E
PT1532105E PT03766505T PT03766505T PT1532105E PT 1532105 E PT1532105 E PT 1532105E PT 03766505 T PT03766505 T PT 03766505T PT 03766505 T PT03766505 T PT 03766505T PT 1532105 E PT1532105 E PT 1532105E
Authority
PT
Portugal
Prior art keywords
sub
chosen
group
cck
activity
Prior art date
Application number
PT03766505T
Other languages
English (en)
Inventor
Lucio Claudio Rovati
Francesco Makovec
Antonio Varnavas
Lucia Lassiani
Original Assignee
Rottapharm Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rottapharm Spa filed Critical Rottapharm Spa
Publication of PT1532105E publication Critical patent/PT1532105E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/68Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D209/00Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/30Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C07D209/42Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/82Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/84Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
PT03766505T 2002-07-26 2003-07-23 Derivados de antracilo possuindo uma actividade anticolecistoquinina (anti-cck-1), um processo para a sua preparação e sua utilização farmacêutica PT1532105E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT2002TO000674A ITTO20020674A1 (it) 2002-07-26 2002-07-26 Derivati antranilici ad attivita' anticolecistochininica (anti-cck-1), procedimento per la loro preparazione e loro uso farmaceutico

Publications (1)

Publication Number Publication Date
PT1532105E true PT1532105E (pt) 2009-06-29

Family

ID=11459544

Family Applications (1)

Application Number Title Priority Date Filing Date
PT03766505T PT1532105E (pt) 2002-07-26 2003-07-23 Derivados de antracilo possuindo uma actividade anticolecistoquinina (anti-cck-1), um processo para a sua preparação e sua utilização farmacêutica

Country Status (11)

Country Link
US (1) US7294648B2 (pt)
EP (1) EP1532105B1 (pt)
JP (1) JP4530853B2 (pt)
AT (1) ATE433439T1 (pt)
AU (1) AU2003253114B8 (pt)
CA (1) CA2493789C (pt)
DE (1) DE60327932D1 (pt)
ES (1) ES2325496T3 (pt)
IT (1) ITTO20020674A1 (pt)
PT (1) PT1532105E (pt)
WO (1) WO2004013087A1 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ542491A (en) 2003-03-28 2009-04-30 Janssen Pharmaceutica Nv Benzo[1,2,5]thiadiazole compounds as CCK2 modulators
PT1651621E (pt) * 2003-08-08 2008-09-30 Janssen Pharmaceutica Nv Compostos de 2-(quinoxalin-5-ilsulfonilamino)-benzamida como moduladores de cck2
BRPI0516027A (pt) 2004-09-24 2008-08-19 Janssen Pharmaceutica Nv compostos de sulfonamida

Also Published As

Publication number Publication date
ATE433439T1 (de) 2009-06-15
ES2325496T3 (es) 2009-09-07
DE60327932D1 (de) 2009-07-23
WO2004013087A1 (en) 2004-02-12
EP1532105B1 (en) 2009-06-10
AU2003253114B2 (en) 2009-07-16
US7294648B2 (en) 2007-11-13
CA2493789C (en) 2012-05-01
JP2005533866A (ja) 2005-11-10
ITTO20020674A0 (it) 2002-07-26
JP4530853B2 (ja) 2010-08-25
AU2003253114A1 (en) 2004-02-23
EP1532105A1 (en) 2005-05-25
AU2003253114B8 (en) 2009-08-13
US20060111304A1 (en) 2006-05-25
ITTO20020674A1 (it) 2004-01-26
CA2493789A1 (en) 2004-02-12

Similar Documents

Publication Publication Date Title
BRPI0413232B8 (pt) composto tendo atividade inibitória contra transportador dependente de sódio, composição farmacêutica compreendendo o composto, uso do composto na preparação de um medicamento e processo para a preparação do composto
MY140528A (en) Spiroketal derivatives and their use as therapeutic agents for diabetes
IL160304A0 (en) ACTIVATOR FOR PEROXISOME PROLIFERATOR-RESPONSIVE RECEPTOR delta
MXPA04001240A (es) Analogos antitumorales.
ES2093332T3 (es) Nuevos derivados arilglicinamidicos, su procedimiento de preparacion y su uso para el tratamiento de la disuria.
DK1204662T3 (da) Azaindoler med serotoninreceptoraffinitet
PT1468692E (pt) Utilizacao de 2,6-dialquil-4-sililfenois para o tratamento do xantoma
DE68926981D1 (de) Cephemverbindungen und Verfahren zu ihrer Herstellung
BRPI0210746B8 (pt) derivados de 6-'2-(fosfonometóxi)alcóxi-pirimidina e seu método de preparação
PT1532105E (pt) Derivados de antracilo possuindo uma actividade anticolecistoquinina (anti-cck-1), um processo para a sua preparação e sua utilização farmacêutica
TW200505446A (en) Inhibitor of cox
CA2014521A1 (en) 2-Substituted N,N'-Ditrimethoxybenzoyl Piperazines, a Preparation Process of the Same and Therapeutic Compositions Containing Them
MX9206930A (es) Nuevos compuestos
AU703092B2 (en) Benzene derivatives
CA2027542A1 (en) Uv-absorbing cyclic enaminoketones
DE69702955T2 (de) Bis-Imide Derivate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zubereitung
DE60026161D1 (de) Amidin-derivate, ihre herstellung und verwendung als medikamenten
DE60238847D1 (de) Pyrimidinderivate enthaltendes medikament
EP1241166A4 (en) 3-MEHTYL CHROMAN AND THIOCHROME DERIVATIVES
MY111111A (en) Novel (1-phenyl-1-heterocyclyl) methanol and (1-phenyl -1-heterocyclyl) methylamine drrivatives
TH37483B (th) อนุพันธ์ 5-เมโรคิลแนพธาลีน
WO2004026548A3 (fr) Procede de traitement chimique d'un substrat en un materiau comprenant du bois
TH32102A (th) สารประกอบแนพธิล สารอินเทอมิเดียท สารผสม และวิธีใช้
HUP0303691A2 (hu) Uretánszármazékok, eljárás az előállításukra és alkalmazásuk gyógyszerkészítmények előállítására
TH14992EX (th) อนุพันธ์แอลกอฮอล์หรือแอลดิไฮด์ และการใช้สารเหล่านั้น