PT1000952E - Novos derivados 2-halogenados de 5-o-desosaminileritronolida a, processo de preparação e sua utilização como medicamentos - Google Patents

Novos derivados 2-halogenados de 5-o-desosaminileritronolida a, processo de preparação e sua utilização como medicamentos Download PDF

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Publication number
PT1000952E
PT1000952E PT99402523T PT99402523T PT1000952E PT 1000952 E PT1000952 E PT 1000952E PT 99402523 T PT99402523 T PT 99402523T PT 99402523 T PT99402523 T PT 99402523T PT 1000952 E PT1000952 E PT 1000952E
Authority
PT
Portugal
Prior art keywords
deosaminylerythronolide
medicines
making
new
well
Prior art date
Application number
PT99402523T
Other languages
English (en)
Inventor
Alexis Denis
Constantin Agouridas
Claude Fromentin
Francois Bretin
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of PT1000952E publication Critical patent/PT1000952E/pt

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biotechnology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PT99402523T 1998-10-15 1999-10-14 Novos derivados 2-halogenados de 5-o-desosaminileritronolida a, processo de preparação e sua utilização como medicamentos PT1000952E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9812937A FR2784682B1 (fr) 1998-10-15 1998-10-15 Nouveaux derives 2-halogene de 5-0-desosaminylerythronolide a, leur procede de preparation et leur application comme medicaments

Publications (1)

Publication Number Publication Date
PT1000952E true PT1000952E (pt) 2011-06-16

Family

ID=9531602

Family Applications (1)

Application Number Title Priority Date Filing Date
PT99402523T PT1000952E (pt) 1998-10-15 1999-10-14 Novos derivados 2-halogenados de 5-o-desosaminileritronolida a, processo de preparação e sua utilização como medicamentos

Country Status (10)

Country Link
US (3) US6352983B1 (pt)
EP (1) EP1000952B1 (pt)
JP (1) JP4864184B2 (pt)
AT (1) ATE501158T1 (pt)
CY (1) CY1112050T1 (pt)
DE (1) DE69943259D1 (pt)
DK (1) DK1000952T3 (pt)
ES (1) ES2362709T3 (pt)
FR (1) FR2784682B1 (pt)
PT (1) PT1000952E (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR200401847T4 (tr) 2000-06-30 2004-09-21 Pfizer Products Inc. Makrolit antibiyotikler.
FR2812635B1 (fr) * 2000-08-01 2002-10-11 Aventis Pharma Sa Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens
US7591653B2 (en) * 2006-09-08 2009-09-22 Aees, Inc. Modular power distribution center
CN106432383A (zh) * 2016-09-14 2017-02-22 重庆两江药物研发中心有限公司 索利霉素及其中间体的制备方法
US11744859B2 (en) 2017-07-07 2023-09-05 Epicentrx, Inc. Compositions and methods for parenteral administration of therapeutic agents

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL99995A (en) * 1990-11-21 1997-11-20 Roussel Uclaf Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
US5631355A (en) 1992-04-22 1997-05-20 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide a derivatives
US6274715B1 (en) * 1995-11-08 2001-08-14 Abbott Laboratories Tricyclic erythromycin derivatives
FR2742757B1 (fr) * 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
CO4990960A1 (es) * 1997-10-29 2000-12-26 Abbott Lab Derivados de cetolidos 2-halo-6-o sustituidos
US6124269A (en) * 1997-10-29 2000-09-26 Abbott Laboratories 2-Halo-6-O-substituted ketolide derivatives

Also Published As

Publication number Publication date
JP2000128896A (ja) 2000-05-09
FR2784682B1 (fr) 2002-12-06
DE69943259D1 (de) 2011-04-21
DK1000952T3 (da) 2011-06-27
EP1000952A2 (fr) 2000-05-17
EP1000952B1 (fr) 2011-03-09
US7119180B2 (en) 2006-10-10
US20020111319A1 (en) 2002-08-15
US20050065101A1 (en) 2005-03-24
EP1000952A3 (fr) 2004-01-02
FR2784682A1 (fr) 2000-04-21
US6352983B1 (en) 2002-03-05
CY1112050T1 (el) 2015-11-04
ES2362709T3 (es) 2011-07-12
JP4864184B2 (ja) 2012-02-01
ATE501158T1 (de) 2011-03-15

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