PL2407466T3 - Związek piperazynowy zdolny do inhibitowania syntazy prostaglandyny d - Google Patents

Związek piperazynowy zdolny do inhibitowania syntazy prostaglandyny d

Info

Publication number
PL2407466T3
PL2407466T3 PL10750777T PL10750777T PL2407466T3 PL 2407466 T3 PL2407466 T3 PL 2407466T3 PL 10750777 T PL10750777 T PL 10750777T PL 10750777 T PL10750777 T PL 10750777T PL 2407466 T3 PL2407466 T3 PL 2407466T3
Authority
PL
Poland
Prior art keywords
synthase
compound capable
piperazine compound
inhibiting prostaglandin
prostaglandin
Prior art date
Application number
PL10750777T
Other languages
English (en)
Inventor
Yoshihiro Urade
Makoto Kitade
Kazuhiko Shigeno
Keiko Yamane
Katsunao Tanaka
Original Assignee
Taiho Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Taiho Pharmaceutical Co Ltd filed Critical Taiho Pharmaceutical Co Ltd
Publication of PL2407466T3 publication Critical patent/PL2407466T3/pl

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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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PL10750777T 2009-03-09 2010-03-08 Związek piperazynowy zdolny do inhibitowania syntazy prostaglandyny d PL2407466T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2009055721 2009-03-09
EP10750777.4A EP2407466B1 (en) 2009-03-09 2010-03-08 Piperazine compound capable of inhibiting prostaglandin d synthase
PCT/JP2010/053760 WO2010104024A1 (ja) 2009-03-09 2010-03-08 プロスタグランジンd合成酵素を阻害するピペラジン化合物

Publications (1)

Publication Number Publication Date
PL2407466T3 true PL2407466T3 (pl) 2016-06-30

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Application Number Title Priority Date Filing Date
PL10750777T PL2407466T3 (pl) 2009-03-09 2010-03-08 Związek piperazynowy zdolny do inhibitowania syntazy prostaglandyny d

Country Status (19)

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US (2) US8865714B2 (pl)
EP (1) EP2407466B1 (pl)
JP (1) JP5111657B2 (pl)
KR (1) KR101421785B1 (pl)
CN (1) CN102341385B (pl)
AU (1) AU2010222122B2 (pl)
BR (1) BRPI1009212B8 (pl)
CA (1) CA2754613C (pl)
DK (1) DK2407466T3 (pl)
ES (1) ES2564454T3 (pl)
HK (1) HK1165419A1 (pl)
HU (1) HUE027702T2 (pl)
MX (1) MX2011009423A (pl)
MY (1) MY159870A (pl)
PL (1) PL2407466T3 (pl)
RU (1) RU2496778C2 (pl)
SG (1) SG173865A1 (pl)
TW (1) TWI450893B (pl)
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RU2011140869A (ru) 2013-04-20
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EP2407466A1 (en) 2012-01-18
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US20140128394A1 (en) 2014-05-08
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AU2010222122B2 (en) 2013-06-27
EP2407466B1 (en) 2016-01-13
CA2754613C (en) 2016-07-12
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KR101421785B1 (ko) 2014-07-22
BRPI1009212B1 (pt) 2024-02-20
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TWI450893B (zh) 2014-09-01
CA2754613A1 (en) 2010-09-16
MX2011009423A (es) 2011-09-28
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