PE20000633A1 - THERAPEUTIC COMBINATIONS FOR MUSCULOSKELETAL FRAGILITY - Google Patents
THERAPEUTIC COMBINATIONS FOR MUSCULOSKELETAL FRAGILITYInfo
- Publication number
- PE20000633A1 PE20000633A1 PE1999000522A PE00052299A PE20000633A1 PE 20000633 A1 PE20000633 A1 PE 20000633A1 PE 1999000522 A PE1999000522 A PE 1999000522A PE 00052299 A PE00052299 A PE 00052299A PE 20000633 A1 PE20000633 A1 PE 20000633A1
- Authority
- PE
- Peru
- Prior art keywords
- etil
- pyridin
- oxo
- tartrate
- salt
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Abstract
SE REFIERE A UNA COMPOSICION FARMACEUTICA QUE COMPRENDE a)UN MODULADOR SELECTIVO DEL RECEPTOR DE ESTROGENOS (SERM) TAL COMO (-)-CIS-6-FENIL-5-(4-(2-PIRROLIDIN-1-IL-ETOXI)-FENIL)-5,6,7,8-TETRAHIDRONAFTALENO-2-OL O SU SAL D-TARTRATO; b)UN SECRETAGOGO DE LA HORMONA DE CRECIMIENTO TAL COMO 2-AMINO-N-(1(R)-(2,4-DIFLUORO-BENCILOXIMETIL)-2-OXO-2-(3-OXO-3a(R)-PIRIDIN-2-ILMETIL)-2-(2,2,2-TRIFLUORO-ETIL)-2,3,3a,4,6,7-HEXAHIDRO-PIRAZOLO[4,3-c]PIRIDIN-5-IL)-ETIL)-2-METIL-PROPIONAMIDA O SU SAL L-TARTRATO. LA COMPOSICION PUEDE SER UTIL PARA EL TRATAMIENTO DE LA FRAGILIDAD MUSCULOESQUELETICA, OSTEOPOROSIS, OSTEOTOMIA, PERDIDA OSEA IDIOPATICA INFANTIL, PERDIDA OSEA ASOCIADA CON PERIODONTITIS, CURACION DE HUESO DESPUES DE UNA RECONSTRUCCION FACIAL, RECONSTRUCCION MAXILAR, RECONSTRUCCION MANDIBULARREFERS TO A PHARMACEUTICAL COMPOSITION INCLUDING a) A SELECTIVE MODULATOR OF THE ESTROGEN RECEPTOR (SERM) SUCH AS (-) - CIS-6-PHENYL-5- (4- (2-PYRROLIDIN-1-IL-ETOXY) -PHENIL ) -5,6,7,8-TETRAHYDRONAPHTHALENE-2-OL OR ITS D-TARTRATE SALT; b) A SECRETAGOG OF GROWTH HORMONE SUCH AS 2-AMINO-N- (1 (R) - (2,4-DIFLUORO-BENZYLOXIMETHYL) -2-OXO-2- (3-OXO-3a (R) -PYRIDIN -2-ILMETIL) -2- (2,2,2-TRIFLUORO-ETIL) -2,3,3a, 4,6,7-HEXAHIDRO-PIRAZOLO [4,3-c] PYRIDIN-5-IL) -ETIL ) -2-METHYL-PROPIONAMIDE OR ITS SALT L-TARTRATE. THE COMPOSITION MAY BE USEFUL FOR THE TREATMENT OF MUSCULOSKELETAL FRAGILITY, OSTEOPOROSIS, OSTEOTOMY, CHILDHOOD IDIOPATIC BONE LOSS, BONE LOSS ASSOCIATED WITH PERIODONTITIS, BONE HEALING AFTER MAXIMUM RECONSTRUCTION, FACIAL RECONSTRUCTION
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US8942498P | 1998-06-16 | 1998-06-16 |
Publications (1)
Publication Number | Publication Date |
---|---|
PE20000633A1 true PE20000633A1 (en) | 2000-07-26 |
Family
ID=22217565
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PE1999000522A PE20000633A1 (en) | 1998-06-16 | 1999-06-11 | THERAPEUTIC COMBINATIONS FOR MUSCULOSKELETAL FRAGILITY |
Country Status (29)
Country | Link |
---|---|
EP (1) | EP1085867A1 (en) |
JP (1) | JP2002518328A (en) |
KR (1) | KR20010052817A (en) |
CN (1) | CN1305378A (en) |
AP (1) | AP9901581A0 (en) |
AR (1) | AR018868A1 (en) |
AU (1) | AU3342099A (en) |
BG (1) | BG105128A (en) |
BR (1) | BR9911357A (en) |
CA (1) | CA2335112A1 (en) |
CO (1) | CO5070586A1 (en) |
EA (1) | EA200001189A1 (en) |
GT (1) | GT199900083A (en) |
HR (1) | HRP20000857A2 (en) |
HU (1) | HUP0102395A2 (en) |
ID (1) | ID26726A (en) |
IL (1) | IL139587A0 (en) |
IS (1) | IS5727A (en) |
MA (1) | MA26648A1 (en) |
NO (1) | NO20006381L (en) |
OA (1) | OA11569A (en) |
PA (1) | PA8472101A1 (en) |
PE (1) | PE20000633A1 (en) |
PL (1) | PL345064A1 (en) |
SK (1) | SK18902000A3 (en) |
TN (1) | TNSN99118A1 (en) |
UY (1) | UY25557A1 (en) |
WO (1) | WO1999065488A1 (en) |
ZA (1) | ZA993973B (en) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1004306A3 (en) * | 1998-08-06 | 2000-06-07 | Pfizer Products Inc. | Estrogen agonists/antagonists |
JP2004507502A (en) | 2000-08-30 | 2004-03-11 | ファイザー・プロダクツ・インク | Sustained release formulation for growth hormone secretagogue |
IL145106A0 (en) * | 2000-08-30 | 2002-06-30 | Pfizer Prod Inc | Intermittent administration of a geowth hormone secretagogue |
US7524866B2 (en) | 2001-11-29 | 2009-04-28 | Gtx, Inc. | Prevention and treatment of androgen—deprivation induced osteoporosis |
EP1666033B1 (en) * | 2001-11-29 | 2008-12-31 | GTX, Inc. | Prevention and treatment of androgen-deprivation induced osteoporosis |
US7476653B2 (en) | 2003-06-18 | 2009-01-13 | Tranzyme Pharma, Inc. | Macrocyclic modulators of the ghrelin receptor |
CU23558A1 (en) | 2006-02-28 | 2010-07-20 | Ct Ingenieria Genetica Biotech | COMPOUNDS ANALOG TO THE PEPTIDIC SECRETAGOGS OF THE GROWTH HORMONE |
JP2010518090A (en) | 2007-02-09 | 2010-05-27 | トランザイム・ファーマ,インコーポレイテッド | Macrocyclic ghrelin receptor modulators and methods of use thereof |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
UA51676C2 (en) * | 1995-11-02 | 2002-12-16 | Пфайзер Інк. | (-)cis-6(S)-phenyl-5(R)-[4-(2-pyrrolidin-I-ylethoxy)phenyl]-5,6,7,8-tetrahydronaphthalen-2-ol D-tartrate, a method of its preparation, method of THE treatment OF diseases medicated by agonists of estrogen and a pharmaceutical composition |
TW432073B (en) * | 1995-12-28 | 2001-05-01 | Pfizer | Pyrazolopyridine compounds |
HN1996000101A (en) * | 1996-02-28 | 1997-06-26 | Inc Pfizer | COMBINED THERAPY FOR OSTEOPOROSIS |
-
1999
- 1999-05-03 JP JP2000554368A patent/JP2002518328A/en active Pending
- 1999-05-03 CA CA002335112A patent/CA2335112A1/en not_active Abandoned
- 1999-05-03 PL PL99345064A patent/PL345064A1/en unknown
- 1999-05-03 WO PCT/IB1999/000796 patent/WO1999065488A1/en not_active Application Discontinuation
- 1999-05-03 KR KR1020007014140A patent/KR20010052817A/en not_active Application Discontinuation
- 1999-05-03 OA OA1200000346A patent/OA11569A/en unknown
- 1999-05-03 SK SK1890-2000A patent/SK18902000A3/en unknown
- 1999-05-03 BR BR9911357-0A patent/BR9911357A/en not_active Application Discontinuation
- 1999-05-03 AU AU33420/99A patent/AU3342099A/en not_active Abandoned
- 1999-05-03 IL IL13958799A patent/IL139587A0/en unknown
- 1999-05-03 EP EP99914723A patent/EP1085867A1/en not_active Withdrawn
- 1999-05-03 CN CN99807381A patent/CN1305378A/en active Pending
- 1999-05-03 ID IDW20002604A patent/ID26726A/en unknown
- 1999-05-03 HU HU0102395A patent/HUP0102395A2/en unknown
- 1999-05-03 EA EA200001189A patent/EA200001189A1/en unknown
- 1999-05-07 PA PA19998472101A patent/PA8472101A1/en unknown
- 1999-06-10 AP APAP/P/1999/001581A patent/AP9901581A0/en unknown
- 1999-06-11 PE PE1999000522A patent/PE20000633A1/en not_active Application Discontinuation
- 1999-06-11 UY UY25557A patent/UY25557A1/en not_active Application Discontinuation
- 1999-06-14 GT GT199900083A patent/GT199900083A/en unknown
- 1999-06-15 AR ARP990102847A patent/AR018868A1/en not_active Application Discontinuation
- 1999-06-15 ZA ZA9903973A patent/ZA993973B/en unknown
- 1999-06-15 TN TNTNSN99118A patent/TNSN99118A1/en unknown
- 1999-06-15 MA MA25622A patent/MA26648A1/en unknown
- 1999-06-16 CO CO99037624A patent/CO5070586A1/en unknown
-
2000
- 2000-11-24 IS IS5727A patent/IS5727A/en unknown
- 2000-12-14 NO NO20006381A patent/NO20006381L/en not_active Application Discontinuation
- 2000-12-14 HR HR20000857A patent/HRP20000857A2/en not_active Application Discontinuation
-
2001
- 2001-01-08 BG BG105128A patent/BG105128A/en unknown
Also Published As
Publication number | Publication date |
---|---|
ID26726A (en) | 2001-02-01 |
PL345064A1 (en) | 2001-11-19 |
EP1085867A1 (en) | 2001-03-28 |
TNSN99118A1 (en) | 2005-11-10 |
IL139587A0 (en) | 2002-02-10 |
NO20006381D0 (en) | 2000-12-14 |
GT199900083A (en) | 2000-12-05 |
AU3342099A (en) | 2000-01-05 |
WO1999065488A1 (en) | 1999-12-23 |
SK18902000A3 (en) | 2001-12-03 |
CA2335112A1 (en) | 1999-12-23 |
BG105128A (en) | 2001-11-30 |
HUP0102395A2 (en) | 2001-11-28 |
EA200001189A1 (en) | 2001-06-25 |
MA26648A1 (en) | 2004-12-20 |
JP2002518328A (en) | 2002-06-25 |
AR018868A1 (en) | 2001-12-12 |
KR20010052817A (en) | 2001-06-25 |
ZA993973B (en) | 2000-12-15 |
CO5070586A1 (en) | 2001-08-28 |
OA11569A (en) | 2004-07-01 |
CN1305378A (en) | 2001-07-25 |
BR9911357A (en) | 2001-03-13 |
HRP20000857A2 (en) | 2001-10-31 |
AP9901581A0 (en) | 1999-06-30 |
IS5727A (en) | 2000-11-24 |
UY25557A1 (en) | 2001-01-31 |
PA8472101A1 (en) | 2000-09-29 |
NO20006381L (en) | 2000-12-14 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD | Application declared void or lapsed |