PA8579401A1 - Derivados de 2,3-dihidro-isoindol-1-ona como inhibidores de mao-b - Google Patents
Derivados de 2,3-dihidro-isoindol-1-ona como inhibidores de mao-bInfo
- Publication number
- PA8579401A1 PA8579401A1 PA20038579401A PA8579401A PA8579401A1 PA 8579401 A1 PA8579401 A1 PA 8579401A1 PA 20038579401 A PA20038579401 A PA 20038579401A PA 8579401 A PA8579401 A PA 8579401A PA 8579401 A1 PA8579401 A1 PA 8579401A1
- Authority
- PA
- Panama
- Prior art keywords
- dihidro
- isoindol
- ona
- inhibitors
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/46—Iso-indoles; Hydrogenated iso-indoles with an oxygen atom in position 1
Abstract
DERIVADOS DE 2,3-DIHIDRO-ISOINDOL-1-ONA, PROCESOS PARA SU PRODUCCION, SU USO COMO COMPOSICIONES FARMACEUTICAS Y MEDICAMENTOS QUE LAS COMPRENDEN, PARA LA PREVENCION Y TRATAMIENTO DE ENFERMEDADES QUE SON MEDIADAS POR INHIBIDORES DE LA MONOAMINOXIDASA B.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP02017676 | 2002-08-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
PA8579401A1 true PA8579401A1 (es) | 2004-02-16 |
Family
ID=31502695
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PA20038579401A PA8579401A1 (es) | 2002-08-07 | 2003-08-04 | Derivados de 2,3-dihidro-isoindol-1-ona como inhibidores de mao-b |
Country Status (16)
Country | Link |
---|---|
US (1) | US6846832B2 (es) |
EP (1) | EP1539694A1 (es) |
JP (1) | JP4322805B2 (es) |
KR (1) | KR20050059062A (es) |
CN (1) | CN1305848C (es) |
AR (1) | AR040788A1 (es) |
BR (1) | BR0313543A (es) |
CA (1) | CA2493143A1 (es) |
GT (1) | GT200300165A (es) |
MX (1) | MXPA05001327A (es) |
PA (1) | PA8579401A1 (es) |
PE (1) | PE20040753A1 (es) |
PL (1) | PL375417A1 (es) |
RU (1) | RU2322437C2 (es) |
TW (1) | TW200413315A (es) |
WO (1) | WO2004014856A1 (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BRPI0410746A (pt) * | 2003-05-19 | 2006-06-27 | Irm Llc | compostos e composições imunossupressoras |
MY150088A (en) | 2003-05-19 | 2013-11-29 | Irm Llc | Immunosuppressant compounds and compositions |
EP2281556A1 (en) | 2005-02-25 | 2011-02-09 | F. Hoffmann-La Roche AG | Tablets with improved drugs substance dispersibility |
CN102190616B (zh) * | 2010-03-18 | 2015-07-29 | 苏州泽璟生物制药有限公司 | 一种氘代的ω-二苯基脲的合成及生产的方法和工艺 |
ES2753194T3 (es) * | 2012-03-02 | 2020-04-07 | Tms Co Ltd | Derivado de cromano |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3834861A1 (de) | 1988-10-13 | 1990-04-19 | Basf Ag | Arylalkoxycumarine, verfahren zu ihrer herstellung und diese enthaltende therapeutische mittel |
TW219935B (es) * | 1991-12-25 | 1994-02-01 | Mitsubishi Chemicals Co Ltd | |
US5326760A (en) * | 1992-06-29 | 1994-07-05 | Glaxo, Inc. | Aminobutanoic acid compounds having metalloprotease inhibiting properties |
ES2098186B1 (es) | 1995-02-09 | 1998-02-01 | Consejo Superior Investigacion | Composiciones farmaceuticas a base de aminometilindoles para su aplicacion terapeutica como neuroprotectores en las enfermedades de parkinson y alzheimer. |
US5679715A (en) | 1995-06-07 | 1997-10-21 | Harris; Richard Y. | Method for treating multiple sclerosis |
JP3258027B2 (ja) | 1996-03-15 | 2002-02-18 | サマーセット・ファーマシューティカルズ・インコーポレイテッド | セレジリン投与による末梢ニューロパシーの予防および治療方法 |
WO2001034172A2 (en) | 1999-11-05 | 2001-05-17 | Vela Pharmaceuticals Inc. | Methods and compositions for treating reward deficiency syndrome |
US6660736B2 (en) * | 2002-03-27 | 2003-12-09 | Hoffmann-La Roche Inc. | Phthalimido derivatives and a process for their preparation |
-
2003
- 2003-07-22 US US10/625,116 patent/US6846832B2/en not_active Expired - Fee Related
- 2003-07-31 CN CNB038189747A patent/CN1305848C/zh not_active Expired - Fee Related
- 2003-07-31 JP JP2004526827A patent/JP4322805B2/ja not_active Expired - Fee Related
- 2003-07-31 PL PL03375417A patent/PL375417A1/xx not_active Application Discontinuation
- 2003-07-31 RU RU2005106200/04A patent/RU2322437C2/ru not_active IP Right Cessation
- 2003-07-31 KR KR1020057002233A patent/KR20050059062A/ko not_active Application Discontinuation
- 2003-07-31 BR BR0313543-8A patent/BR0313543A/pt not_active IP Right Cessation
- 2003-07-31 CA CA002493143A patent/CA2493143A1/en not_active Abandoned
- 2003-07-31 MX MXPA05001327A patent/MXPA05001327A/es active IP Right Grant
- 2003-07-31 WO PCT/EP2003/008456 patent/WO2004014856A1/en active Application Filing
- 2003-07-31 EP EP03784117A patent/EP1539694A1/en not_active Withdrawn
- 2003-08-04 PA PA20038579401A patent/PA8579401A1/es unknown
- 2003-08-04 TW TW092121280A patent/TW200413315A/zh unknown
- 2003-08-04 PE PE2003000766A patent/PE20040753A1/es not_active Application Discontinuation
- 2003-08-05 AR AR20030102801A patent/AR040788A1/es not_active Application Discontinuation
- 2003-08-05 GT GT200300165A patent/GT200300165A/es unknown
Also Published As
Publication number | Publication date |
---|---|
PL375417A1 (en) | 2005-11-28 |
CN1675181A (zh) | 2005-09-28 |
MXPA05001327A (es) | 2005-04-28 |
US6846832B2 (en) | 2005-01-25 |
CA2493143A1 (en) | 2004-02-19 |
WO2004014856A1 (en) | 2004-02-19 |
AR040788A1 (es) | 2005-04-20 |
RU2005106200A (ru) | 2005-10-20 |
JP2005539015A (ja) | 2005-12-22 |
GT200300165A (es) | 2004-03-16 |
TW200413315A (en) | 2004-08-01 |
US20040082603A1 (en) | 2004-04-29 |
CN1305848C (zh) | 2007-03-21 |
KR20050059062A (ko) | 2005-06-17 |
PE20040753A1 (es) | 2004-11-20 |
AU2003255334A1 (en) | 2004-02-25 |
BR0313543A (pt) | 2005-06-21 |
EP1539694A1 (en) | 2005-06-15 |
JP4322805B2 (ja) | 2009-09-02 |
RU2322437C2 (ru) | 2008-04-20 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DOP2009000155A (es) | Derivados de hetero-pentaciclo-fenilo fusionados, composicion farmaceutica que los comprende y usos para preparar un medicamento util para el tratamiento de una condicion mediada por p38 | |
CR8778A (es) | Revestimientos de azucar y metodos para estos | |
BRPI0418251C1 (pt) | fosfonatos, monofosfonamidatos, bisfosfonamidatos, e, composição farmacêutica os compreendendo | |
UY30710A1 (es) | Nuevos derivados de 1,4-benzotiepina-1,1-dioxido sustituidos con radicales ciclohexilo, método para su preparacion, productos farmacéuticos que comprenden estos compuestos y su uso. | |
PA8583601A1 (es) | Derivados de pirrolidona como inhibidores de maob | |
DOP2009000165A (es) | Derivados de oxindol sustituido, medicamentos que los comprenden y uso de los mismos | |
DE502005008790D1 (de) | Substituierte phenylaminopyrimidine | |
UY27455A1 (es) | Derivados n-(1,4,5,6-tetrahidro-ciclopentapirazol -3-il)- sustituidos. su obtención y uso como fármacos. | |
ECSP088541A (es) | [(1h-indol-5-il)-heteroariloxi]-(1-aza-biciclo[3.3.1]nonanos como ligandos colinérgicos del n-achr para el tratamiento de trastornos psicóticos y neurodegenerativos | |
CY1108932T1 (el) | Ενωσεις 4-(ετεροκυκλυλ)-βενζολοσουλφοξιμινης για την θεραπευτικη αγωγη φλεγμονωδων ασθενειων | |
EA200801580A1 (ru) | Новые производные пирониндола и способ их получения | |
UY28098A1 (es) | Derivados de anilinopirazol útiles en el tratamiento de la diabetes | |
HN2003000162A (es) | Derivados de isoindolona, proceso de preparacion y compuestos intermedios de este proceso, su uso como medicamentos, y composiciones farmaceuticas que los contienen. | |
UY28313A1 (es) | Nonadepsipeptidos acilados | |
DOP2006000024A (es) | Tiazolidinonas, su preparación y su uso como medicamento | |
BR112023018237A2 (pt) | Fenalquilaminas e métodos para fabricação e uso das mesmas | |
PA8597501A1 (es) | Derivados azabiciclicos de piridiloximetilo y bencisoxazol | |
DOP2003000621A (es) | Inhibidores triariloxiariloxipirimidin-2,4,6-triona de metaloproteinasa | |
ECSP003707A (es) | Diazepanes | |
UY28115A1 (es) | Derivados del acido isoftalico | |
GT200800066A (es) | Derivados de 9-cloro-15-deoxiprostaglandina, procedimiento para su preparacion y su uso como medicamento. | |
PA8579401A1 (es) | Derivados de 2,3-dihidro-isoindol-1-ona como inhibidores de mao-b | |
UY27733A1 (es) | Derivados de ciclopenteno. | |
ECSP055917A (es) | Derivados de diazepanes útiles como inhibidores de lfa | |
UY26179A1 (es) | Amidas sustituidas del ácido fenilciclohexanocarboxilico y su uso como inhibidores de la incorporación de adenosina. |