OA06063A - Dérivés de l'anthelmintique C-076. - Google Patents

Dérivés de l'anthelmintique C-076.

Info

Publication number
OA06063A
OA06063A OA56623A OA56623A OA06063A OA 06063 A OA06063 A OA 06063A OA 56623 A OA56623 A OA 56623A OA 56623 A OA56623 A OA 56623A OA 06063 A OA06063 A OA 06063A
Authority
OA
OAPI
Prior art keywords
anthelmintic
derivatives
Prior art date
Application number
OA56623A
Other languages
English (en)
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of OA06063A publication Critical patent/OA06063A/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P17/00Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
    • C12P17/18Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms containing at least two hetero rings condensed among themselves or condensed with a common carbocyclic ring system, e.g. rifamycin
    • C12P17/181Heterocyclic compounds containing oxygen atoms as the only ring heteroatoms in the condensed system, e.g. Salinomycin, Septamycin
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P19/00Preparation of compounds containing saccharide radicals
    • C12P19/44Preparation of O-glycosides, e.g. glucosides
    • C12P19/60Preparation of O-glycosides, e.g. glucosides having an oxygen of the saccharide radical directly bound to a non-saccharide heterocyclic ring or a condensed ring system containing a non-saccharide heterocyclic ring, e.g. coumermycin, novobiocin
    • C12P19/62Preparation of O-glycosides, e.g. glucosides having an oxygen of the saccharide radical directly bound to a non-saccharide heterocyclic ring or a condensed ring system containing a non-saccharide heterocyclic ring, e.g. coumermycin, novobiocin the hetero ring having eight or more ring members and only oxygen as ring hetero atoms, e.g. erythromycin, spiramycin, nystatin
    • C12P19/623Avermectin; Milbemycin; Ivermectin; C-076

Landscapes

  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Microbiology (AREA)
  • Veterinary Medicine (AREA)
  • General Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Agronomy & Crop Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
OA56623A 1977-10-03 1978-10-03 Dérivés de l'anthelmintique C-076. OA06063A (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US83860277A 1977-10-03 1977-10-03
US83909977A 1977-10-03 1977-10-03

Publications (1)

Publication Number Publication Date
OA06063A true OA06063A (fr) 1981-06-30

Family

ID=27126041

Family Applications (1)

Application Number Title Priority Date Filing Date
OA56623A OA06063A (fr) 1977-10-03 1978-10-03 Dérivés de l'anthelmintique C-076.

Country Status (9)

Country Link
EP (1) EP0001688B1 (fr)
JP (1) JPS5461197A (fr)
AU (1) AU519570B2 (fr)
DE (1) DE2861286D1 (fr)
DK (1) DK152049C (fr)
IE (1) IE47570B1 (fr)
IT (1) IT1157353B (fr)
NZ (1) NZ188459A (fr)
OA (1) OA06063A (fr)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4203976A (en) * 1978-08-02 1980-05-20 Merck & Co., Inc. Sugar derivatives of C-076 compounds
US4200581A (en) * 1978-08-04 1980-04-29 Merck & Co., Inc. Alkyl derivatives of C-076 compounds
US4289760A (en) * 1980-05-02 1981-09-15 Merck & Co., Inc. 23-Keto derivatives of C-076 compounds
US4285963A (en) * 1980-08-07 1981-08-25 Merck & Co., Inc. Novel derivatives of C-076 compounds
US4412991A (en) * 1981-08-28 1983-11-01 Merck & Co., Inc. 22-Hydroxy derivatives of C-076 compounds, pharmaceutical compositions and method of use
US4427663A (en) * 1982-03-16 1984-01-24 Merck & Co., Inc. 4"-Keto-and 4"-amino-4"-deoxy avermectin compounds and substituted amino derivatives thereof
US4846789A (en) * 1982-07-19 1989-07-11 L. S. Van Landingham, Jr. Combatting internal parasites in warm blooded animals
US4469682A (en) * 1983-01-28 1984-09-04 Merck & Co., Inc. Avermectin and milbemycin phosphate esters, pharmaceutical compositions, and method of use
JPS60126289A (ja) * 1983-11-14 1985-07-05 Sankyo Co Ltd ミルベマイシン類の5−カ−ボネ−ト誘導体
GB2168345B (en) * 1984-12-14 1988-05-25 Ciba Geigy Ag Pesticidal 13b-substituted milbemycin derivatives
ES8605582A1 (es) * 1985-12-11 1986-03-16 Antibioticos Sa Un procedimiento para la preparacion de avermectinas
ZA872140B (en) * 1986-03-25 1988-11-30 Sankyo Co Microlide compounds,their preparation and their use
BR8701302A (pt) * 1986-03-25 1987-12-22 Sankyo Co Compostos macrolideos,sua preparacao e seu uso
EP0240274A3 (fr) * 1986-04-03 1990-03-14 Merck & Co. Inc. Avermectine comme agents pour promotion de la croissance
JPS6333341A (ja) * 1986-07-28 1988-02-13 Seitetsu Kagaku Co Ltd 配糖体の処理方法
IN167980B (fr) * 1987-01-23 1991-01-19 Pfizer
US4895837A (en) * 1988-01-29 1990-01-23 Merck & Co., Inc. Avermectin derivatives
US5387395A (en) * 1992-07-06 1995-02-07 Beckman Instruments, Inc. Fluid distribution manifold
GB2272772A (en) * 1992-11-20 1994-05-25 British Tech Group Image reconstruction
US5380838A (en) * 1993-10-08 1995-01-10 Merck & Co. Inc. Stable solvates of avermectin compounds
AU728221B2 (en) 1996-06-05 2001-01-04 Ashmont Holdings Limited Injectable compositions
MXPA02010587A (es) 2000-04-27 2003-03-10 Sankyo Co Derivados de milbemicina 13-sustituidos, su preparacion y su uso contra insectos y otras plagas.
CR6574A (es) 2001-02-27 2004-10-28 Syngenta Participations Ag Sales de avermectinas substituidas en la posicion 4 con propiedades plaguicidas
EG23124A (en) 2001-02-27 2004-04-28 Syngenta Participations Ag Avermectins substituted in the 4-position having pesticidal properties
AR036486A1 (es) 2001-08-28 2004-09-15 Syngenta Participations Ag Derivados 4"-desoxi-4"-(s)-amino avermectina, composicion plaguicida, procedimiento para la preparacion de esa composicion, metodo para controlar plagas, y uso de estos derivados para preparar una composicion
TW200407330A (en) 2002-05-07 2004-05-16 Syngenta Participations Ag 4"-Deoxy-4"-(S)-amido avermectin derivatives
US7001889B2 (en) 2002-06-21 2006-02-21 Merial Limited Anthelmintic oral homogeneous veterinary pastes
GB0302310D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0320176D0 (en) * 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
DE102007007750A1 (de) 2006-08-17 2008-02-21 Bayer Cropscience Ag Avermectinderivate
JP2010006703A (ja) * 2006-11-07 2010-01-14 Hokko Chem Ind Co Ltd アベルメクチンモノ配糖体誘導体

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS4914624A (fr) * 1972-06-08 1974-02-08
JPS5645890B2 (fr) * 1973-05-29 1981-10-29
SE434277B (sv) * 1976-04-19 1984-07-16 Merck & Co Inc Sett att framstella nya antihelmintiskt verkande foreningar genom odling av streptomyces avermitilis

Also Published As

Publication number Publication date
DK152049C (da) 1988-06-20
JPS6254113B2 (fr) 1987-11-13
DE2861286D1 (en) 1982-01-14
IE47570B1 (en) 1984-05-02
IT7851320A0 (it) 1978-09-29
IE781964L (en) 1979-04-03
EP0001688A1 (fr) 1979-05-02
IT1157353B (it) 1987-02-11
DK152049B (da) 1988-01-25
DK434478A (da) 1979-04-04
JPS5461197A (en) 1979-05-17
EP0001688B1 (fr) 1981-11-04
AU519570B2 (en) 1981-12-10
NZ188459A (en) 1982-09-07
AU4008978A (en) 1980-03-27

Similar Documents

Publication Publication Date Title
OA06063A (fr) Dérivés de l'anthelmintique C-076.
AR219560A1 (es) Procedimiento para la preparacion de derivados de 5,5-dimetil-hidantoina
OA06105A (fr) Dérivés antithéilériaux de naphthoquinone.
IT7848582A0 (it) Immidazo(1,2-a)-piridine eterociclo -sostituite nuove
MX5529E (es) Procedimiento para la preparacion de indolo-(2,3-a)-quinolizidinas
NL7806658A (nl) Werkwijze voor de bereiding van 7,8-dihydro- 14-hydro- xynormorfine.
MX5256E (es) Procedimiento para la preparacion de derivados de 20,21-dinoreburnamenina
RO77485A (fr) Procede pour la preparation des 1,2,3-thiadiazole-3-in-5-ilidenurees
RO76721A (fr) Procede pour preparer 3.12.-hydroxy-4-phenyle-cycloalcanone
AR218498A1 (es) Procedimiento de preparacion de derivados de 1,3-difenoxipropan-2-ona
MC1357A1 (fr) Derives de 2,3-indoledione
SE7804878L (sv) Forfarande for framstellning av 1,2-dikloretan
AR224501A1 (es) Procedimiento de preparacion de derivados de la tieno-(3,2-c)-piridina
NL7800191A (nl) Anthelmintisch preparaat.
NL7801259A (nl) Half-synthetische 4"-amino-oleandomycine derivaten.
FI782517A (fi) Foerfarande foer framstaellning av 2,3-polymetylen-4-oxo-4h-pyrido(1,2-a)-pyrimidiner
IT7824666A0 (it) Composti di alfa-aloacetammidi conproprieta' erbicide.
IT7822883A0 (it) Procedimento per la preparazione di 3,5 di alogeno-aniline.
IT7829237A0 (it) Procedimento di preparazione distilbeni 4,4'-diossi-sostituiti.
AR230835A1 (es) Procedimiento para la obtencion de derivados de 2,1,3-tiadiazin-4-ona-2,2-dioxido
BE865569A (fr) Derives de l'imidazole.
DK573678A (da) 3,4-methano-pyrrolidinderivater
IT7826344A0 (it) Procedimento per la preparazione di coloranti basici.
MC1279A1 (fr) Dérivés de la benzodiazépine
NL7812127A (nl) N'-fenyl-n-methylureumderivaten.