NO931679D0 - NEW Heterocyclic Compounds as Antagonists for Excitatory Amino Acid Receptors, Procedures for their Preparation and Their Use - Google Patents

NEW Heterocyclic Compounds as Antagonists for Excitatory Amino Acid Receptors, Procedures for their Preparation and Their Use

Info

Publication number: NO931679D0
Authority: NO; Norway
Prior art keywords: antagonists; procedures; preparation; amino acid; heterocyclic compounds
Prior art date: 1990-11-15

Application number

NO931679A

Other languages

Norwegian (no)

Other versions

NO931679L (en

Inventor

Alf Claesson

Britt-Marie Swahn

Original Assignee

Astra Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-11-15

Filing date

1993-05-07

Publication date

1993-05-07

1993-05-07 Application filed by Astra Ab filed Critical Astra Ab

1993-05-07 Publication of NO931679L publication Critical patent/NO931679L/en

1993-05-07 Publication of NO931679D0 publication Critical patent/NO931679D0/en

Links

102000018899 Glutamate Receptors Human genes 0.000 title 1
108010027915 Glutamate Receptors Proteins 0.000 title 1
239000005557 antagonist Substances 0.000 title 1
150000002391 heterocyclic compounds Chemical class 0.000 title 1
238000000034 method Methods 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
- C07F9/6509—Six-membered rings
- C07F9/650952—Six-membered rings having the nitrogen atoms in the positions 1 and 4
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/576—Six-membered rings
- C07F9/59—Hydrogenated pyridine rings

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Pain & Pain Management (AREA)
Anesthesiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

NO931679A 1990-11-15 1993-05-07 NEW Heterocyclic Compounds as Antagonists for Excitatory Amino Acid Receptors, Procedures for their Preparation and Their Use NO931679D0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
SE9003652A SE9003652D0 (en)	1990-11-15	1990-11-15	NEW HETEROCYCLIC COMPOUNDS
PCT/SE1991/000753 WO1992008724A1 (en)	1990-11-15	1991-11-07	New heterocyclic compounds as antagonists of excitatory amino acid receptors, processes for their preparation and their use

Publications (2)

Publication Number	Publication Date
NO931679L NO931679L (en)	1993-05-07
NO931679D0 true NO931679D0 (en)	1993-05-07

Family

ID=20380925

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO931679A NO931679D0 (en)	1990-11-15	1993-05-07	NEW Heterocyclic Compounds as Antagonists for Excitatory Amino Acid Receptors, Procedures for their Preparation and Their Use

Country Status (17)

Country	Link
EP (1)	EP0557375A1 (en)
JP (1)	JPH06502421A (en)
CN (1)	CN1061595A (en)
AU (1)	AU652399B2 (en)
CA (1)	CA2095224A1 (en)
CZ (1)	CZ80993A3 (en)
FI (1)	FI932206A (en)
HU (1)	HU9301417D0 (en)
IE (1)	IE913922A1 (en)
IS (1)	IS3782A7 (en)
LT (1)	LTIP1718A (en)
MX (1)	MX9101979A (en)
NO (1)	NO931679D0 (en)
PT (1)	PT99515A (en)
SE (1)	SE9003652D0 (en)
SK (1)	SK46993A3 (en)
WO (1)	WO1992008724A1 (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5194430A (en) *	1990-05-17	1993-03-16	Merrell Dow Pharmaceuticals Inc.	Heterocyclic-nmda antagonists
TW281670B (en) *	1993-09-02	1996-07-21	Hoffmann La Roche
US5491241A (en) *	1993-10-18	1996-02-13	Eli Lilly And Company	Bicyclic intermediates for excitatory amino acid receptor antagonists
ES2907373T3 (en)	2016-02-04	2022-04-25	Takeda Pharmaceuticals Co	Substituted piperidine compound and use thereof

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1248531A (en) *	1984-04-17	1989-01-10	Jeffrey C. Watkins	4-substituted piperazine-2-carboxylic acids
JPS612519A (en) *	1984-04-24	1986-01-08	Aron Kasei Co Ltd	Method of injection molding
US4906621A (en) *	1985-05-24	1990-03-06	Ciba-Geigy Corporation	Certain 2-carboxypiperidyl-alkylene phosphonic acids and esters thereof useful for the treatment of disorders responsive to N-methyl-D-aspartate receptor blockade
US4740346A (en) *	1986-02-26	1988-04-26	The Budd Company	Perimeter resin feeding of composite structures
JPS63112129A (en) *	1986-10-30	1988-05-17	Toyoda Gosei Co Ltd	Multi-color resin molding die
EP0275820B1 (en) *	1986-11-21	1991-02-06	Ciba-Geigy Ag	Unsaturated phosphonic acids and derivatives

1990
- 1990-11-15 SE SE9003652A patent/SE9003652D0/en unknown
1991
- 1991-11-05 CN CN91110925A patent/CN1061595A/en active Pending
- 1991-11-07 JP JP4500566A patent/JPH06502421A/en active Pending
- 1991-11-07 EP EP91920264A patent/EP0557375A1/en not_active Withdrawn
- 1991-11-07 HU HU931417A patent/HU9301417D0/en unknown
- 1991-11-07 WO PCT/SE1991/000753 patent/WO1992008724A1/en not_active Application Discontinuation
- 1991-11-07 CZ CS93809A patent/CZ80993A3/en unknown
- 1991-11-07 CA CA002095224A patent/CA2095224A1/en not_active Abandoned
- 1991-11-07 AU AU89391/91A patent/AU652399B2/en not_active Ceased
- 1991-11-07 SK SK46993A patent/SK46993A3/en unknown
- 1991-11-08 MX MX9101979A patent/MX9101979A/en unknown
- 1991-11-12 IE IE392291A patent/IE913922A1/en unknown
- 1991-11-14 IS IS3782A patent/IS3782A7/en unknown
- 1991-11-14 PT PT99515A patent/PT99515A/en not_active Application Discontinuation
1993
- 1993-05-07 NO NO931679A patent/NO931679D0/en unknown
- 1993-05-14 FI FI932206A patent/FI932206A/en not_active Application Discontinuation
- 1993-12-30 LT LTIP1718A patent/LTIP1718A/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
FI932206A0 (en)	1993-05-14
CZ80993A3 (en)	1994-02-16
AU8939191A (en)	1992-06-11
SE9003652D0 (en)	1990-11-15
AU652399B2 (en)	1994-08-25
PT99515A (en)	1992-09-30
WO1992008724A1 (en)	1992-05-29
NO931679L (en)	1993-05-07
LTIP1718A (en)	1995-07-25
FI932206A (en)	1993-05-14
CN1061595A (en)	1992-06-03
MX9101979A (en)	1992-07-08
SK46993A3 (en)	1993-10-06
EP0557375A1 (en)	1993-09-01
IS3782A7 (en)	1992-05-16
CA2095224A1 (en)	1992-05-16
JPH06502421A (en)	1994-03-17
IE913922A1 (en)	1992-05-20
HU9301417D0 (en)	1993-09-28

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