NO931040L - INDOLES AND INDAZOL DERIVATIVES, PROCEDURE FOR PREPARING AND USING THEREOF - Google Patents

INDOLES AND INDAZOL DERIVATIVES, PROCEDURE FOR PREPARING AND USING THEREOF

Info

Publication number
NO931040L
NO931040L NO93931040A NO931040A NO931040L NO 931040 L NO931040 L NO 931040L NO 93931040 A NO93931040 A NO 93931040A NO 931040 A NO931040 A NO 931040A NO 931040 L NO931040 L NO 931040L
Authority
NO
Norway
Prior art keywords
indoles
preparing
procedure
indazol
derivatives
Prior art date
Application number
NO93931040A
Other languages
Norwegian (no)
Other versions
NO931040D0 (en
Inventor
Shunji Naruto
Yuichi Sugano
Yoshiki Matsui
Toshiyuki Tonohiro
Tsugio Kaneko
Nobuyoshi Iwata
Original Assignee
Sankyo Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co filed Critical Sankyo Co
Publication of NO931040D0 publication Critical patent/NO931040D0/en
Publication of NO931040L publication Critical patent/NO931040L/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12—Radicals substituted by oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO93931040A 1992-03-23 1993-03-23 INDOLES AND INDAZOL DERIVATIVES, PROCEDURE FOR PREPARING AND USING THEREOF NO931040L (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP6532392 1992-03-23
JP915693 1993-01-22

Publications (2)

Publication Number Publication Date
NO931040D0 NO931040D0 (en) 1993-03-23
NO931040L true NO931040L (en) 1993-09-24

Family

ID=26343823

Family Applications (1)

Application Number Title Priority Date Filing Date
NO93931040A NO931040L (en) 1992-03-23 1993-03-23 INDOLES AND INDAZOL DERIVATIVES, PROCEDURE FOR PREPARING AND USING THEREOF

Country Status (11)

Country Link
EP (1) EP0562832A1 (en)
KR (1) KR930019661A (en)
CN (1) CN1081676A (en)
AU (1) AU3537893A (en)
CA (1) CA2092112A1 (en)
CZ (1) CZ47393A3 (en)
FI (1) FI931291A (en)
HU (1) HU9300828D0 (en)
IL (1) IL105139A0 (en)
NO (1) NO931040L (en)
TW (1) TW226019B (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW263504B (en) * 1991-10-03 1995-11-21 Pfizer
IT1271352B (en) * 1993-04-08 1997-05-27 Boehringer Ingelheim Italia INDOLE DERIVATIVES USEFUL IN THE TREATMENT OF DISORDERS OF THE CENTRAL NERVOUS SYSTEM
GB9310582D0 (en) * 1993-05-22 1993-07-07 Smithkline Beecham Plc Pharmaceuticals
US5620973A (en) * 1993-11-30 1997-04-15 Takeda Chemical Industries, Ltd. Tetracyclic condensed heterocyclic compounds and their use
ES2098186B1 (en) * 1995-02-09 1998-02-01 Consejo Superior Investigacion PHARMACEUTICAL COMPOSITIONS BASED ON AMINOMETHYLINDOLS FOR THERAPEUTIC APPLICATION AS NEUROPROTECTORS IN PARKINSON AND ALZHEIMER DISEASES.
GB2308362A (en) * 1995-12-19 1997-06-25 Lilly Industries Ltd Pharmaceutical indole derivatives
AU6852898A (en) * 1997-04-17 1998-11-11 Takeda Chemical Industries Ltd. Thermogenic composition and benzazepine thermogenics
EP1891954A3 (en) 1998-09-30 2009-01-14 Takeda Pharmaceutical Company Limited Acetylcholinesterase inhibitors for improving excretory potency of urinary bladder
CN1317276C (en) * 2000-09-29 2007-05-23 中国科学院上海药物研究所 Indolylpiperidine compound and preparation process and use thereof
KR100614862B1 (en) 2001-12-28 2006-08-22 다케다 야쿠힌 고교 가부시키가이샤 Preventives/remedies for voiding disturbance
TW200621237A (en) 2004-11-01 2006-07-01 Wyeth Corp [(1-h-indazol-3-yl)methyl]phenols and (hydroxyphenyl)(1h-indazol-3-yl)methanones
EP1828182B1 (en) 2004-11-29 2010-03-10 Warner-Lambert Company LLC Therapeutic pyrazolo[3,4-b]pyridines and indazoles
MX2008009022A (en) 2006-01-13 2008-09-24 Wyeth Corp Sulfonyl substituted 1h-indoles as ligands for the 5-hydroxytryptamine receptors.
RU2012136451A (en) 2010-01-28 2014-03-10 Президент Энд Феллоуз Оф Гарвард Колледж COMPOSITIONS AND METHODS FOR IMPROVING PROTEASOMIC ACTIVITY
US8293738B2 (en) 2010-05-12 2012-10-23 Abbott Laboratories Indazole inhibitors of kinase
DK2707101T3 (en) * 2011-05-12 2019-05-13 Proteostasis Therapeutics Inc PROTEOSTASE REGULATORS
US9849135B2 (en) 2013-01-25 2017-12-26 President And Fellows Of Harvard College USP14 inhibitors for treating or preventing viral infections
WO2015073528A1 (en) 2013-11-12 2015-05-21 Proteostasis Therapeutics, Inc. Proteasome activity enhancing compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2334358A1 (en) * 1975-12-12 1977-07-08 Sogeras NEW DRUGS DERIVED FROM INDOLE
FR2477544A1 (en) * 1980-03-07 1981-09-11 Pharmindustrie NOVEL CHLORO-3 QUINOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION, AND THEIR USE AS MEDICAMENTS

Also Published As

Publication number Publication date
NO931040D0 (en) 1993-03-23
TW226019B (en) 1994-07-01
FI931291A (en) 1993-09-24
IL105139A0 (en) 1993-07-08
AU3537893A (en) 1993-09-30
CZ47393A3 (en) 1993-11-17
EP0562832A1 (en) 1993-09-29
FI931291A0 (en) 1993-03-23
CA2092112A1 (en) 1993-09-24
HU9300828D0 (en) 1993-06-28
CN1081676A (en) 1994-02-09
KR930019661A (en) 1993-10-18

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