NO924617D0 - Fremgangsmaate for fremstilling av 10beta-h-steroider - Google Patents

Fremgangsmaate for fremstilling av 10beta-h-steroider

Info

Publication number
NO924617D0
NO924617D0 NO1992924617A NO924617A NO924617D0 NO 924617 D0 NO924617 D0 NO 924617D0 NO 1992924617 A NO1992924617 A NO 1992924617A NO 924617 A NO924617 A NO 924617A NO 924617 D0 NO924617 D0 NO 924617D0
Authority
NO
Norway
Prior art keywords
pct
steroids
10beta
preparing
procedure
Prior art date
Application number
NO1992924617A
Other languages
English (en)
Other versions
NO924617L (no
NO304115B1 (no
Inventor
Eckhard Ottow
Guenter Neef
Arwed Cleve
Rudolf Wiechert
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of NO924617D0 publication Critical patent/NO924617D0/no
Publication of NO924617L publication Critical patent/NO924617L/no
Publication of NO304115B1 publication Critical patent/NO304115B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0059—Estrane derivatives substituted in position 17 by a keto group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005—Ketals
    • C07J21/006—Ketals at position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J21/005—Ketals
    • C07J21/008—Ketals at position 17
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
    • C07J41/0083—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
NO924617A 1990-06-01 1992-11-30 FremgangsmÕte for fremstilling av 10<beta>-H-steroider NO304115B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4018167A DE4018167A1 (de) 1990-06-01 1990-06-01 Verfahren zur herstellung von 10(beta)-h-steroiden
PCT/EP1991/001018 WO1991018918A1 (de) 1990-06-01 1991-06-03 VERFAHREN ZUR HERSTELLUNG VON 10β-H-STEROIDEN

Publications (3)

Publication Number Publication Date
NO924617D0 true NO924617D0 (no) 1992-11-30
NO924617L NO924617L (no) 1992-11-30
NO304115B1 NO304115B1 (no) 1998-10-26

Family

ID=6407912

Family Applications (1)

Application Number Title Priority Date Filing Date
NO924617A NO304115B1 (no) 1990-06-01 1992-11-30 FremgangsmÕte for fremstilling av 10<beta>-H-steroider

Country Status (12)

Country Link
US (1) US5405979A (no)
EP (1) EP0532562B1 (no)
JP (1) JP2999258B2 (no)
AT (1) ATE114317T1 (no)
CA (1) CA2084313C (no)
DE (2) DE4018167A1 (no)
DK (1) DK0532562T3 (no)
ES (1) ES2065039T3 (no)
FI (1) FI111642B (no)
HU (1) HU218484B (no)
NO (1) NO304115B1 (no)
WO (1) WO1991018918A1 (no)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4042007A1 (de) * 1990-12-22 1992-06-25 Schering Ag 6,7-modifizierte-11(beta)-aryl-4-estrene
DE19610667C2 (de) * 1996-03-08 1998-04-09 Schering Ag (Z)-11ß-[4-(Dimethylamino)phenyl]17ß-hydroxy-17alpha-(3-hydroxy-1-propenyl)estr-4-en-3-on als kristallines Ansolvat
DE102011004899A1 (de) 2011-03-01 2012-09-06 Bayer Pharma Aktiengesellschaft 17-Hydroxy-17-pentafluorethyl-estra-4,9(10)-dien-11-aryl-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung zur Behandlung von Krankheiten
JP6906525B2 (ja) 2015-12-23 2021-07-21 オリック ファーマシューティカルズ，インク． グルココルチコイド受容体の阻害剤
WO2017112904A1 (en) 2015-12-23 2017-06-29 Oric Pharmaceuticals, Inc. Inhibitors of glucocorticoid receptor
CA3009525A1 (en) * 2015-12-23 2017-06-29 Oric Pharmaceuticals, Inc. Inhibitors of glucocorticoid receptor
MX2019004030A (es) 2016-10-07 2019-09-16 Oric Pharmaceuticals Inc Inhibidores del receptor de glucocorticoides.
CA3095042A1 (en) * 2018-04-11 2019-10-17 Oric Pharmaceuticals, Inc. Solid forms and formulations comprising a glucocorticoid receptor antagonist and uses thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3014120A1 (de) * 1980-04-12 1981-10-29 Hoechst Ag, 6000 Frankfurt Verfahren zur synthese von oestron bzw. oestronderivaten
AU572589B2 (en) * 1983-12-14 1988-05-12 Upjohn Company, The 11(alpha)-difluoromethyl and (e)-and (z)-11-fluoromethylene steroids
IE60780B1 (en) * 1987-01-23 1994-08-10 Akzo Nv New 11-aryl steroid derivatives

Also Published As

Publication number Publication date
FI925445A0 (fi) 1992-11-30
EP0532562A1 (de) 1993-03-24
CA2084313C (en) 2002-12-10
DE59103592D1 (de) 1995-01-12
JP2999258B2 (ja) 2000-01-17
NO924617L (no) 1992-11-30
EP0532562B1 (de) 1994-11-23
ATE114317T1 (de) 1994-12-15
NO304115B1 (no) 1998-10-26
WO1991018918A1 (de) 1991-12-12
HUT62596A (en) 1993-05-28
HU9203775D0 (en) 1993-03-29
ES2065039T3 (es) 1995-02-01
US5405979A (en) 1995-04-11
HU218484B (hu) 2000-09-28
CA2084313A1 (en) 1991-12-02
FI111642B (fi) 2003-08-29
FI925445A (fi) 1992-11-30
DE4018167A1 (de) 1991-12-05
DK0532562T3 (da) 1995-05-15
JPH05507271A (ja) 1993-10-21

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Legal Events

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