NO903513L - Fremgangsmaate for fremstilling av cykliske neurokinin a-antagonister. - Google Patents

Fremgangsmaate for fremstilling av cykliske neurokinin a-antagonister.

Info

Publication number: NO903513L
Authority: NO; Norway
Prior art keywords: cycleic; neurokinin; antagonists; procedure; preparation
Prior art date: 1989-08-10

Application number

NO90903513A

Other languages

English (en)

Other versions

NO177715B (no

NO177715C (no

NO903513D0 (no

Inventor

Scott Lee Harbeson

Stephen Hendersen Buck

Original Assignee

Merrell Dow Pharma

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1989-08-10

Filing date

1990-08-09

Publication date

1991-02-11

1990-08-09 Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma

1990-08-09 Publication of NO903513D0 publication Critical patent/NO903513D0/no

1991-02-11 Publication of NO903513L publication Critical patent/NO903513L/no

1995-07-31 Publication of NO177715B publication Critical patent/NO177715B/no

1995-11-08 Publication of NO177715C publication Critical patent/NO177715C/no

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/22—Tachykinins, e.g. Eledoisins, Substance P; Related peptides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/64—Cyclic peptides containing only normal peptide links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Immunology (AREA)
Genetics & Genomics (AREA)
Biochemistry (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Molecular Biology (AREA)
Pulmonology (AREA)
Biophysics (AREA)
Biomedical Technology (AREA)
Pain & Pain Management (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Oncology (AREA)
Rheumatology (AREA)
Transplantation (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Virology (AREA)
Communicable Diseases (AREA)
Urology & Nephrology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Dermatology (AREA)
Peptides Or Proteins (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

NO903513A 1989-08-10 1990-08-09 Analogifremgangsmåte for fremstilling av cykliske neurokinin A-antagonister NO177715C (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US39223689A	1989-08-10	1989-08-10

Publications (4)

Publication Number	Publication Date
NO903513D0 NO903513D0 (no)	1990-08-09
NO903513L true NO903513L (no)	1991-02-11
NO177715B NO177715B (no)	1995-07-31
NO177715C NO177715C (no)	1995-11-08

Family

ID=23549831

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO903513A NO177715C (no)	1989-08-10	1990-08-09	Analogifremgangsmåte for fremstilling av cykliske neurokinin A-antagonister

Country Status (22)

Country	Link
US (1)	US5731286A (no)
EP (1)	EP0412542B1 (no)
JP (1)	JP2829779B2 (no)
KR (1)	KR0169123B1 (no)
CN (1)	CN1035056C (no)
AR (1)	AR246087A1 (no)
AT (1)	ATE132503T1 (no)
AU (1)	AU638264B2 (no)
CA (1)	CA2022740C (no)
DD (1)	DD297168A5 (no)
DE (1)	DE69024555T2 (no)
DK (1)	DK0412542T3 (no)
ES (1)	ES2084627T3 (no)
FI (1)	FI95913C (no)
GR (1)	GR3018984T3 (no)
HU (1)	HU206729B (no)
IE (1)	IE69382B1 (no)
IL (1)	IL95309A (no)
NO (1)	NO177715C (no)
NZ (1)	NZ234814A (no)
PT (1)	PT94952B (no)
ZA (1)	ZA906188B (no)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ZA894533B (en) *	1988-06-20	1990-03-28	Merrell Dow Pharma	Neurokinin a antogonists
DE4034829A1 (de) *	1990-11-02	1992-05-07	Merck Patent Gmbh	Cyclopeptide
US5625060A (en) *	1991-05-03	1997-04-29	Elf Sanofi	Polycyclic amine compounds and their enantiomers, their method of preparation and pharmaceutical compositions on which they are present
FR2676055B1 (fr) *	1991-05-03	1993-09-03	Sanofi Elf	Composes polycycliques amines et leurs enantiomeres, procede pour leur preparation et compositions pharmaceutiques les contenant.
AU2387592A (en) *	1991-08-08	1993-03-02	A. Menarini Industrie Farmaceutiche Riunite S.R.L.	Cyclic hexapeptides as tachyquinin antagonists, their preparation and pharmaceutical compositions thereof
US5731285A (en) *	1992-04-15	1998-03-24	A. Menatini Industrie Farmaceutiche	Tachiquinine antagonist tricyclic compounds, preparation of same and pharmaceutical compositions containing such compounds
CN102498124B (zh) *	2009-03-16	2015-05-13	多伦多大学管理委员会	环状氨基酸分子及其制备方法
CN109071602B (zh)	2015-11-11	2022-09-13	西兰制药公司	靶向α4β7整联蛋白的环肽
ES2884107T3 (es)	2016-11-11	2021-12-10	Zealand Pharma As	Multímeros de péptidos cíclicos con diana en la integrina alfa-4 beta-7
IL270465B (en)	2017-05-10	2022-09-01	Encycle Therapeutics Inc	Cyclic peptides targeting alpha4beta7 integrin

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4665157A (en) *	1985-09-30	1987-05-12	Mcneilab, Inc.	Peptide antagonists of neurokinin B
US4742156A (en) *	1985-09-30	1988-05-03	Mcneilab, Inc.	Peptide antagonists of neurokinin B and opthalmic solutions containing them
DE3711335A1 (de) *	1987-04-03	1988-10-20	Merck Patent Gmbh	Aminosaeurederivate
GB8807246D0 (en) *	1988-03-25	1988-04-27	Merck Sharp & Dohme	Therapeutic agents
ZA894533B (en) *	1988-06-20	1990-03-28	Merrell Dow Pharma	Neurokinin a antogonists
IE903957A1 (en) *	1989-11-06	1991-05-08	Sanofi Sa	Aromatic amine compounds, their method of preparation and¹pharmaceutical compositions in which they are present
IL99320A (en) *	1990-09-05	1995-07-31	Sanofi Sa	Arylalkylamines, their preparation and pharmaceutical preparations containing them
FR2677361A1 (fr) *	1991-06-04	1992-12-11	Adir	Nouveaux peptides et pseudopeptides, derives de tachykinines, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.

1990
- 1990-08-06 AU AU60222/90A patent/AU638264B2/en not_active Expired
- 1990-08-06 ZA ZA906188A patent/ZA906188B/xx unknown
- 1990-08-07 AR AR90317547A patent/AR246087A1/es active
- 1990-08-07 CA CA002022740A patent/CA2022740C/en not_active Expired - Lifetime
- 1990-08-07 IL IL9530990A patent/IL95309A/en not_active IP Right Cessation
- 1990-08-08 FI FI903922A patent/FI95913C/fi active IP Right Grant
- 1990-08-08 NZ NZ234814A patent/NZ234814A/en unknown
- 1990-08-09 NO NO903513A patent/NO177715C/no unknown
- 1990-08-09 KR KR1019900012226A patent/KR0169123B1/ko not_active IP Right Cessation
- 1990-08-09 CN CN90106972A patent/CN1035056C/zh not_active Expired - Fee Related
- 1990-08-09 ES ES90115309T patent/ES2084627T3/es not_active Expired - Lifetime
- 1990-08-09 IE IE288690A patent/IE69382B1/en not_active IP Right Cessation
- 1990-08-09 DE DE69024555T patent/DE69024555T2/de not_active Expired - Lifetime
- 1990-08-09 AT AT90115309T patent/ATE132503T1/de not_active IP Right Cessation
- 1990-08-09 DK DK90115309.8T patent/DK0412542T3/da active
- 1990-08-09 PT PT94952A patent/PT94952B/pt not_active IP Right Cessation
- 1990-08-09 JP JP2209390A patent/JP2829779B2/ja not_active Expired - Lifetime
- 1990-08-09 HU HU904952A patent/HU206729B/hu not_active IP Right Cessation
- 1990-08-09 EP EP90115309A patent/EP0412542B1/en not_active Expired - Lifetime
- 1990-08-10 DD DD90343398A patent/DD297168A5/de unknown
1996
- 1996-02-14 GR GR960400385T patent/GR3018984T3/el unknown
1997
- 1997-03-05 US US08/811,913 patent/US5731286A/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
ES2084627T3 (es)	1996-05-16
DK0412542T3 (da)	1996-01-29
JP2829779B2 (ja)	1998-12-02
IL95309A0 (en)	1991-06-30
CA2022740C (en)	2000-05-02
AU638264B2 (en)	1993-06-24
IE902886A1 (en)	1991-02-27
CN1035056C (zh)	1997-06-04
DE69024555D1 (de)	1996-02-15
CA2022740A1 (en)	1991-02-11
CN1049353A (zh)	1991-02-20
PT94952A (pt)	1991-04-18
EP0412542A3 (en)	1991-07-24
US5731286A (en)	1998-03-24
ATE132503T1 (de)	1996-01-15
IL95309A (en)	1995-07-31
NZ234814A (en)	1992-03-26
ZA906188B (en)	1991-06-26
KR0169123B1 (ko)	1999-01-15
FI95913C (fi)	1996-04-10
JPH03141295A (ja)	1991-06-17
AR246087A1 (es)	1994-03-30
NO177715B (no)	1995-07-31
DE69024555T2 (de)	1996-05-15
AU6022290A (en)	1991-05-16
HU206729B (en)	1992-12-28
EP0412542B1 (en)	1996-01-03
NO177715C (no)	1995-11-08
IE69382B1 (en)	1996-09-04
FI903922A0 (fi)	1990-08-08
FI95913B (fi)	1995-12-29
HU904952D0 (en)	1991-01-28
EP0412542A2 (en)	1991-02-13
DD297168A5 (de)	1992-01-02
PT94952B (pt)	1997-07-31
KR910004665A (ko)	1991-03-29
HUT54713A (en)	1991-03-28
NO903513D0 (no)	1990-08-09
GR3018984T3 (en)	1996-05-31

Publication	Publication Date	Title
NO900831D0 (no)	1990-02-21	Fremgangsmaate for fremstilling av piperidinforbindelser.
NO890269D0 (no)	1989-01-20	Fremgangsmaate for fremstilling av 1,4-disubstituerte-piperidinyl-forbindelser.
NO902003D0 (no)	1990-05-07	Fremgangsmaate for fremstilling av n-heteroaryl-4-quinolinaminer.
NO900774D0 (no)	1990-02-19	Fremgangsmaate for fremstilling av polyamider.
NO901554D0 (no)	1990-04-05	Fremgangsmaate for fremstilling av dinatrium-cefodizim.
NO904059D0 (no)	1990-09-18	Fremgangsmaate for fremstilling av nye substituerte isokinoliner.
NO904285L (no)	1991-04-04	Fremgangsmaate for fremstilling av substituerte karboksytetrahydroisokinoliner.
NO903513L (no)	1991-02-11	Fremgangsmaate for fremstilling av cykliske neurokinin a-antagonister.
NO892542L (no)	1989-12-21	Fremgangsmaate for fremstilling av neurokinin a antagonister.
NO901391L (no)	1990-10-01	Fremgangsmaate for fremstilling av et 1,8-naftyridin-derivat.
NO904069D0 (no)	1990-09-18	Fremgangsmaate for fremstilling av nye alkanofenoner.
NO901067L (no)	1990-09-10	Fremgangsmaate for fremstilling av tiofener.
NO903666L (no)	1991-02-25	Fremgangsmaate for fremstilling av pyrrolokinolinforbindelser.
NO904061L (no)	1991-03-20	Fremgangsmaate for fremstilling av nmda-antagonister.
NO904060D0 (no)	1990-09-18	Fremgangsmaate for fremstilling av substituerte dibenzofuraner.
NO900969L (no)	1990-09-04	Fremgangsmaate for fremstilling av n-allymetatrifluormetylanilin.
NO904535D0 (no)	1990-10-19	Fremgangsmaate for fremstilling av fenoxy-heterocykliske forbindelser.
NO880409D0 (no)	1988-01-29	Fremgangsmaate for fremstilling av 14,15-substituerte lanosteroler.
NO904070D0 (no)	1990-09-18	Fremgangsmaate for fremstilling av alkanfenoner.
NO901401D0 (no)	1990-03-27	Fremgangsmaate for fremstilling av nye 1-difenylmethylpiperidinderivater.
NO890538L (no)	1990-08-09	Fremgangsmaate for fremstilling av oxadiazolyl-azabicyclo-heptaner.
NO890539D0 (no)	1989-02-08	Fremgangsmaate for fremstilling av lipofile oxadiazoler.
NO920207D0 (no)	1992-01-16	Fremgangsmaate for fremstilling av 6-methyl-oestra-4,6-diener
ATE91413T1 (de)	1993-07-15	Hypotensiver wirkstoff.
FI894896A0 (fi)	1989-10-16	Anordning foer separering av aemnen fraon vatten.