NO810150L - Fremgangsmaate ved fremstilling av nye angiotensin-ii-antagoniserende octapeptidestere inneholdende en aminosyreester-gruppe i 8-stilling - Google Patents
Fremgangsmaate ved fremstilling av nye angiotensin-ii-antagoniserende octapeptidestere inneholdende en aminosyreester-gruppe i 8-stillingInfo
- Publication number
- NO810150L NO810150L NO810150A NO810150A NO810150L NO 810150 L NO810150 L NO 810150L NO 810150 A NO810150 A NO 810150A NO 810150 A NO810150 A NO 810150A NO 810150 L NO810150 L NO 810150L
- Authority
- NO
- Norway
- Prior art keywords
- group
- tyr
- arg
- moiety
- general formula
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/14—Angiotensins: Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S530/00—Chemistry: natural resins or derivatives; peptides or proteins; lignins or reaction products thereof
- Y10S530/80—Antihypertensive peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Vascular Medicine (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
HU8080101A HU181009B (en) | 1980-01-18 | 1980-01-18 | Process for preparing angiotensin-ii analogues with antagonictic activity containing in position 1 sarcosyl,hydroxyacetyl or l-alpha-aminoxy-propionyl group and in positiona 8 esteric group |
Publications (3)
Publication Number | Publication Date |
---|---|
NO810150L true NO810150L (no) | 1981-07-20 |
NO155100B NO155100B (no) | 1986-11-03 |
NO155100C NO155100C (no) | 1987-02-11 |
Family
ID=10947913
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO810150A NO155100C (no) | 1980-01-18 | 1981-01-16 | Analogifremgangsmaate ved fremstilling av nye angiotensin-ii antagoniserende octapeptidestere inneholdende en aminosyreestergruppe i 8-stilling. |
Country Status (19)
Country | Link |
---|---|
US (1) | US4388304A (no) |
EP (1) | EP0034259B1 (no) |
JP (1) | JPS56138155A (no) |
AT (1) | ATE13740T1 (no) |
AU (1) | AU541526B2 (no) |
CA (1) | CA1156222A (no) |
CS (1) | CS217987B2 (no) |
DD (1) | DD156968A5 (no) |
DE (1) | DE3170906D1 (no) |
ES (1) | ES498582A0 (no) |
FI (1) | FI72732C (no) |
HU (1) | HU181009B (no) |
IL (1) | IL61923A (no) |
IN (1) | IN153212B (no) |
NO (1) | NO155100C (no) |
PH (1) | PH16791A (no) |
PL (1) | PL126240B1 (no) |
SU (1) | SU1041030A3 (no) |
YU (1) | YU41959B (no) |
Families Citing this family (48)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
HU191961B (en) * | 1984-08-02 | 1987-04-28 | Richter Gedeon Vegyeszet | Process for producing 1,5 and 8 substituted peptides of angiotenzin-ii antagonistic activity |
US5182264A (en) * | 1986-03-07 | 1993-01-26 | Schering Corporation | Angiotensin II receptor blockers as antiglaucoma agents |
US4983402A (en) * | 1989-02-24 | 1991-01-08 | Clinical Technologies Associates, Inc. | Orally administerable ANF |
US4976968A (en) * | 1989-02-24 | 1990-12-11 | Clinical Technologies Associates, Inc. | Anhydrous delivery systems for pharmacological agents |
US5447728A (en) * | 1992-06-15 | 1995-09-05 | Emisphere Technologies, Inc. | Desferrioxamine oral delivery system |
US6221367B1 (en) | 1992-06-15 | 2001-04-24 | Emisphere Technologies, Inc. | Active agent transport systems |
US5578323A (en) * | 1992-06-15 | 1996-11-26 | Emisphere Technologies, Inc. | Proteinoid carriers and methods for preparation and use thereof |
US5541155A (en) * | 1994-04-22 | 1996-07-30 | Emisphere Technologies, Inc. | Acids and acid salts and their use in delivery systems |
US5714167A (en) | 1992-06-15 | 1998-02-03 | Emisphere Technologies, Inc. | Active agent transport systems |
US6099856A (en) * | 1992-06-15 | 2000-08-08 | Emisphere Technologies, Inc. | Active agent transport systems |
US6331318B1 (en) | 1994-09-30 | 2001-12-18 | Emisphere Technologies Inc. | Carbon-substituted diketopiperazine delivery systems |
US5629020A (en) | 1994-04-22 | 1997-05-13 | Emisphere Technologies, Inc. | Modified amino acids for drug delivery |
US5443841A (en) * | 1992-06-15 | 1995-08-22 | Emisphere Technologies, Inc. | Proteinoid microspheres and methods for preparation and use thereof |
US5693338A (en) * | 1994-09-29 | 1997-12-02 | Emisphere Technologies, Inc. | Diketopiperazine-based delivery systems |
US5792451A (en) * | 1994-03-02 | 1998-08-11 | Emisphere Technologies, Inc. | Oral drug delivery compositions and methods |
US5811127A (en) * | 1992-06-15 | 1998-09-22 | Emisphere Technologies, Inc. | Desferrioxamine oral delivery system |
US5401516A (en) * | 1992-12-21 | 1995-03-28 | Emisphere Technologies, Inc. | Modified hydrolyzed vegetable protein microspheres and methods for preparation and use thereof |
US5958457A (en) * | 1993-04-22 | 1999-09-28 | Emisphere Technologies, Inc. | Compositions for the delivery of antigens |
US5643957A (en) * | 1993-04-22 | 1997-07-01 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
US6610329B2 (en) * | 1993-04-22 | 2003-08-26 | Emisphere Technologies Inc. | Compositions for the delivery of antigens |
US5709861A (en) * | 1993-04-22 | 1998-01-20 | Emisphere Technologies, Inc. | Compositions for the delivery of antigens |
US5766633A (en) * | 1993-04-22 | 1998-06-16 | Emisphere Technologies, Inc. | Oral drug delivery compositions and methods |
US5965121A (en) * | 1995-03-31 | 1999-10-12 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
US5866536A (en) * | 1995-03-31 | 1999-02-02 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
US6090958A (en) * | 1995-03-31 | 2000-07-18 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
BR9604880A (pt) * | 1995-03-31 | 1998-05-19 | Emisphere Tech Inc | Composto composição forma de unidade de dosagem métodos para administração de um agente biologicamente ativo para preparar uma composição para administração de um agente ativo e para preparar um composto e composição farmacológica |
US5650386A (en) * | 1995-03-31 | 1997-07-22 | Emisphere Technologies, Inc. | Compositions for oral delivery of active agents |
US6001347A (en) | 1995-03-31 | 1999-12-14 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
US5989539A (en) * | 1995-03-31 | 1999-11-23 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
US5820881A (en) * | 1995-04-28 | 1998-10-13 | Emisphere Technologies, Inc. | Microspheres of diamide-dicarboxylic acids |
US5667806A (en) * | 1995-06-07 | 1997-09-16 | Emisphere Technologies, Inc. | Spray drying method and apparatus |
US5824345A (en) * | 1995-06-07 | 1998-10-20 | Emisphere Technologies, Inc. | Fragrances and flavorants |
US6051258A (en) * | 1995-06-07 | 2000-04-18 | Emisphere Technologies, Inc. | Proteinoid emulsions and methods for preparation and use thereof |
US5750147A (en) * | 1995-06-07 | 1998-05-12 | Emisphere Technologies, Inc. | Method of solubilizing and encapsulating itraconazole |
WO1997010197A1 (en) * | 1995-09-11 | 1997-03-20 | Emisphere Technologies, Inc. | METHOD FOR PREPARING φ-AMINOALKANOIC ACID DERIVATIVES FROM CYCLOALKANONES |
AU2595697A (en) * | 1996-03-29 | 1997-10-22 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
WO1997047288A1 (en) | 1996-06-14 | 1997-12-18 | Emisphere Technologies, Inc. | Microencapsulated fragrances and method for preparation |
US6358504B1 (en) * | 1997-02-07 | 2002-03-19 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
US5879681A (en) * | 1997-02-07 | 1999-03-09 | Emisphere Technolgies Inc. | Compounds and compositions for delivering active agents |
US6060513A (en) * | 1997-02-07 | 2000-05-09 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
US5876710A (en) * | 1997-02-07 | 1999-03-02 | Emisphere Technologies Inc. | Compounds and compositions for delivering active agents |
US5939381A (en) * | 1997-02-07 | 1999-08-17 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
US5990166A (en) * | 1997-02-07 | 1999-11-23 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
US5804688A (en) * | 1997-02-07 | 1998-09-08 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
US6313088B1 (en) | 1997-02-07 | 2001-11-06 | Emisphere Technologies, Inc. | 8-[(2-hydroxy-4-methoxy benzoyl) amino]-octanoic acid compositions for delivering active agents |
US5863944A (en) * | 1997-04-30 | 1999-01-26 | Emisphere Technologies, Inc. | Compounds and compositions for delivering active agents |
US5962710A (en) * | 1997-05-09 | 1999-10-05 | Emisphere Technologies, Inc. | Method of preparing salicyloylamino acids |
IL140993A0 (en) * | 2000-05-15 | 2002-02-10 | Bayer Ag | Trypsin substrate and diagnostic device, and method of using same |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3907762A (en) * | 1971-12-27 | 1975-09-23 | Univ Sherbrooke | Angiotensin{hd II {B position 8 analogs |
US3923769A (en) * | 1974-05-10 | 1975-12-02 | Francis Merlin Bumpus | {8 N-Me-Ile{40 ,Ile{hu 8{b {9 -Angiotensin II as an angiotensin antagonist |
US3925345A (en) * | 1974-05-10 | 1975-12-09 | Francis Merlin Bumpus | (sar' 1',thr' 8'+9 angiotensin ii as an angiotensin antagonist |
US3923770A (en) * | 1974-05-10 | 1975-12-02 | Francis Merlin Bumpus | {8 Me{hd 2{b Gly{hu 1{b , Ile{hu 8{b {9 -Anziotensin II as an angiotensin antagonist |
US3975365A (en) * | 1975-01-27 | 1976-08-17 | G. D. Searle & Co. | Inhibitory octapeptides angiotensin II |
US3976770A (en) * | 1975-02-10 | 1976-08-24 | Francis Merlin Bumpus | Sar'-(OMe)Thr8 Angiotensin II as an angiotensin II antagonist |
US3973006A (en) * | 1975-02-21 | 1976-08-03 | E. R. Squibb & Sons, Inc. | Peptide enzyme inhibitors of angiotensin I |
HU177133B (en) * | 1977-07-18 | 1981-07-28 | Richter Gedeon Vegyeszet | Process for preparing angiotensin ii analogues containing alpha- amino-oxy-acid in position 1 with angiotensin ii antagonist activity |
HU177134B (en) * | 1977-07-18 | 1981-07-28 | Richter Gedeon Vegyeszet | Process for preparing angiotensin ii analogues containing alpha-hydroxy-acid in position 1 with angiotensin ii antagonist activity |
-
1980
- 1980-01-18 HU HU8080101A patent/HU181009B/hu not_active IP Right Cessation
-
1981
- 1981-01-08 CS CS81173A patent/CS217987B2/cs unknown
- 1981-01-13 PH PH25082A patent/PH16791A/en unknown
- 1981-01-14 US US06/225,048 patent/US4388304A/en not_active Expired - Fee Related
- 1981-01-16 IN IN47/CAL/81A patent/IN153212B/en unknown
- 1981-01-16 NO NO810150A patent/NO155100C/no unknown
- 1981-01-16 DD DD81227055A patent/DD156968A5/de unknown
- 1981-01-16 YU YU92/81A patent/YU41959B/xx unknown
- 1981-01-16 CA CA000368682A patent/CA1156222A/en not_active Expired
- 1981-01-16 AU AU66277/81A patent/AU541526B2/en not_active Ceased
- 1981-01-16 FI FI810122A patent/FI72732C/fi not_active IP Right Cessation
- 1981-01-16 ES ES498582A patent/ES498582A0/es active Granted
- 1981-01-16 IL IL61923A patent/IL61923A/xx unknown
- 1981-01-16 PL PL1981229244A patent/PL126240B1/pl unknown
- 1981-01-16 SU SU813226301A patent/SU1041030A3/ru active
- 1981-01-17 JP JP463281A patent/JPS56138155A/ja active Pending
- 1981-01-19 DE DE8181100356T patent/DE3170906D1/de not_active Expired
- 1981-01-19 AT AT81100356T patent/ATE13740T1/de not_active IP Right Cessation
- 1981-01-19 EP EP81100356A patent/EP0034259B1/de not_active Expired
Also Published As
Publication number | Publication date |
---|---|
FI810122L (fi) | 1981-07-19 |
DE3170906D1 (en) | 1985-07-18 |
ATE13740T1 (de) | 1985-06-15 |
PL126240B1 (en) | 1983-07-30 |
CS217987B2 (en) | 1983-02-25 |
FI72732C (fi) | 1987-07-10 |
JPS56138155A (en) | 1981-10-28 |
EP0034259A1 (de) | 1981-08-26 |
NO155100C (no) | 1987-02-11 |
YU41959B (en) | 1988-04-30 |
CA1156222A (en) | 1983-11-01 |
EP0034259B1 (de) | 1985-06-12 |
NO155100B (no) | 1986-11-03 |
PL229244A1 (no) | 1981-10-30 |
HU181009B (en) | 1983-05-30 |
DD156968A5 (de) | 1982-10-06 |
ES8205754A1 (es) | 1982-07-01 |
AU541526B2 (en) | 1985-01-10 |
IL61923A0 (en) | 1981-02-27 |
YU9281A (en) | 1983-09-30 |
US4388304A (en) | 1983-06-14 |
SU1041030A3 (ru) | 1983-09-07 |
IL61923A (en) | 1984-01-31 |
IN153212B (no) | 1984-06-16 |
FI72732B (fi) | 1987-03-31 |
AU6627781A (en) | 1981-07-23 |
PH16791A (en) | 1984-02-28 |
ES498582A0 (es) | 1982-07-01 |
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