NO20072127L - Heteroatomholdige trisykliske forbindelser - Google Patents
Heteroatomholdige trisykliske forbindelserInfo
- Publication number
- NO20072127L NO20072127L NO20072127A NO20072127A NO20072127L NO 20072127 L NO20072127 L NO 20072127L NO 20072127 A NO20072127 A NO 20072127A NO 20072127 A NO20072127 A NO 20072127A NO 20072127 L NO20072127 L NO 20072127L
- Authority
- NO
- Norway
- Prior art keywords
- heteroatomic
- tricyclic compounds
- tricyclic
- compounds
- epi
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Immunology (AREA)
- Pharmacology & Pharmacy (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Pyridine Compounds (AREA)
- Steroid Compounds (AREA)
Abstract
En fremgangsmåte for fremstilling av 33-Epi-33-klor-FR 520 i ett trinn fra FR520 der beskyttelsesgrupper unngås.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0422643A GB0422643D0 (en) | 2004-10-12 | 2004-10-12 | Organic compounds |
GB0427599A GB0427599D0 (en) | 2004-12-16 | 2004-12-16 | Organic compounds |
PCT/EP2005/010889 WO2006040111A2 (en) | 2004-10-12 | 2005-10-10 | Heteroatoms-containing tricyclic compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20072127L true NO20072127L (no) | 2007-06-08 |
NO338603B1 NO338603B1 (no) | 2016-09-12 |
Family
ID=36084355
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20072127A NO338603B1 (no) | 2004-10-12 | 2007-04-24 | Fremgangsmåte for fremstilling av en heteroatomholdig trisyklisk forbindelse |
Country Status (28)
Country | Link |
---|---|
US (1) | US7514554B2 (no) |
EP (1) | EP1802635B8 (no) |
JP (1) | JP5032326B2 (no) |
KR (1) | KR101228188B1 (no) |
CN (1) | CN101031573B (no) |
AR (1) | AR051386A1 (no) |
AU (1) | AU2005293799B2 (no) |
BR (1) | BRPI0516873A (no) |
CA (1) | CA2581046C (no) |
DK (1) | DK1802635T3 (no) |
EC (1) | ECSP077384A (no) |
ES (1) | ES2389206T3 (no) |
GT (1) | GT200500282A (no) |
HK (1) | HK1105634A1 (no) |
IL (1) | IL182307A (no) |
JO (1) | JO2727B1 (no) |
MA (1) | MA28932B1 (no) |
MX (1) | MX2007004258A (no) |
MY (1) | MY140880A (no) |
NO (1) | NO338603B1 (no) |
NZ (1) | NZ554010A (no) |
PE (1) | PE20060581A1 (no) |
PL (1) | PL1802635T3 (no) |
PT (1) | PT1802635E (no) |
RU (1) | RU2394037C2 (no) |
TN (1) | TNSN07133A1 (no) |
TW (1) | TWI361192B (no) |
WO (1) | WO2006040111A2 (no) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2006060614A1 (en) * | 2004-12-01 | 2006-06-08 | Teva Gyógyszergyár Zàrtköruen Muködo Rèszvènytàrsasàg | Methods for preparing pimecrolimus |
IT1394309B1 (it) | 2009-05-22 | 2012-06-06 | Poli Ind Chimica Spa | Nuovo approccio chimico-enzimatico alla sintesi del pimecrolimus |
CN106854228B (zh) * | 2015-12-08 | 2020-05-29 | 博瑞生物医药(苏州)股份有限公司 | 一种吡美莫司的制备方法 |
EP3178824A1 (en) | 2015-12-08 | 2017-06-14 | Medichem, S.A. | Process for preparing pimecrolimus |
US10975097B2 (en) * | 2017-05-01 | 2021-04-13 | Meda Ab | Process to convert technical ascomycin into purified pimecrolimus |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4464366A (en) * | 1979-12-19 | 1984-08-07 | Ciba Geigy Corporation | Cephem compounds having a terminal aminocarboxylic acid grouping and containing an azacyclyl(thio)ureido group |
US4894366A (en) * | 1984-12-03 | 1990-01-16 | Fujisawa Pharmaceutical Company, Ltd. | Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same |
NZ235991A (en) * | 1989-11-09 | 1993-05-26 | Sandoz Ltd | Macrolide compounds and pharmaceutical compositions thereof |
US5352671A (en) * | 1989-11-09 | 1994-10-04 | Sandoz Ltd. | Heteroatoms-containing tricyclic compounds |
EP0480623A1 (en) | 1990-10-11 | 1992-04-15 | Merck & Co. Inc. | New halomacrolides and derivatives having immunosuppressive activity |
MY110603A (en) | 1993-05-27 | 1998-08-29 | Novartis Ag | Tetrahydropyran derivatives |
US6160117A (en) * | 1997-11-06 | 2000-12-12 | Zeneca Limited | Chemical process |
GB0012383D0 (en) * | 2000-05-22 | 2000-07-12 | Novartis Ag | Organic compounds |
US6667312B2 (en) * | 2000-12-08 | 2003-12-23 | 3M Innovative Properties Company | Thioether substituted imidazoquinolines |
-
2005
- 2005-10-07 GT GT200500282A patent/GT200500282A/es unknown
- 2005-10-09 JO JO2005138A patent/JO2727B1/en active
- 2005-10-10 DK DK05793907.6T patent/DK1802635T3/da active
- 2005-10-10 JP JP2007536064A patent/JP5032326B2/ja active Active
- 2005-10-10 NZ NZ554010A patent/NZ554010A/en unknown
- 2005-10-10 CA CA2581046A patent/CA2581046C/en active Active
- 2005-10-10 US US11/575,757 patent/US7514554B2/en active Active
- 2005-10-10 WO PCT/EP2005/010889 patent/WO2006040111A2/en active Application Filing
- 2005-10-10 AU AU2005293799A patent/AU2005293799B2/en active Active
- 2005-10-10 BR BRPI0516873-2A patent/BRPI0516873A/pt not_active Application Discontinuation
- 2005-10-10 ES ES05793907T patent/ES2389206T3/es active Active
- 2005-10-10 KR KR1020077008216A patent/KR101228188B1/ko active IP Right Grant
- 2005-10-10 PT PT05793907T patent/PT1802635E/pt unknown
- 2005-10-10 MX MX2007004258A patent/MX2007004258A/es active IP Right Grant
- 2005-10-10 PL PL05793907T patent/PL1802635T3/pl unknown
- 2005-10-10 RU RU2007117497/04A patent/RU2394037C2/ru active
- 2005-10-10 CN CN2005800333070A patent/CN101031573B/zh active Active
- 2005-10-10 EP EP05793907.6A patent/EP1802635B8/en active Active
- 2005-10-11 AR ARP050104257A patent/AR051386A1/es not_active Application Discontinuation
- 2005-10-11 MY MYPI20054764A patent/MY140880A/en unknown
- 2005-10-11 PE PE2005001202A patent/PE20060581A1/es not_active Application Discontinuation
- 2005-10-11 TW TW094135403A patent/TWI361192B/zh active
-
2007
- 2007-03-29 IL IL182307A patent/IL182307A/en active IP Right Grant
- 2007-04-11 TN TNP2007000133A patent/TNSN07133A1/fr unknown
- 2007-04-11 EC EC2007007384A patent/ECSP077384A/es unknown
- 2007-04-12 MA MA29826A patent/MA28932B1/fr unknown
- 2007-04-24 NO NO20072127A patent/NO338603B1/no unknown
- 2007-10-05 HK HK07110850.1A patent/HK1105634A1/xx unknown
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