NO20050739L - Ny fremgsmate for syntesen av (7-metoksy-1-naftyl)acetonitril og dens anvendelse i syntesen av agomelatin - Google Patents

Ny fremgsmate for syntesen av (7-metoksy-1-naftyl)acetonitril og dens anvendelse i syntesen av agomelatin

Info

Publication number
NO20050739L
NO20050739L NO20050739A NO20050739A NO20050739L NO 20050739 L NO20050739 L NO 20050739L NO 20050739 A NO20050739 A NO 20050739A NO 20050739 A NO20050739 A NO 20050739A NO 20050739 L NO20050739 L NO 20050739L
Authority
NO
Norway
Prior art keywords
synthesis
agomelatine
naphthyl
acetonitrile
methoxy
Prior art date
Application number
NO20050739A
Other languages
English (en)
Other versions
NO333493B1 (no
NO20050739D0 (no
Inventor
Jean-Claude Souvie
Blanco Isaac Gonzalez
Original Assignee
Servier Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Servier Lab filed Critical Servier Lab
Publication of NO20050739D0 publication Critical patent/NO20050739D0/no
Publication of NO20050739L publication Critical patent/NO20050739L/no
Publication of NO333493B1 publication Critical patent/NO333493B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61B—DIAGNOSIS; SURGERY; IDENTIFICATION
    • A61B17/00—Surgical instruments, devices or methods, e.g. tourniquets
    • A61B17/24—Surgical instruments, devices or methods, e.g. tourniquets for use in the oral cavity, larynx, bronchial passages or nose; Tongue scrapers
    • A61B17/244—Surgical instruments, devices or methods, e.g. tourniquets for use in the oral cavity, larynx, bronchial passages or nose; Tongue scrapers for cleaning of the tongue
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61C—DENTISTRY; APPARATUS OR METHODS FOR ORAL OR DENTAL HYGIENE
    • A61C17/00—Devices for cleaning, polishing, rinsing or drying teeth, teeth cavities or prostheses; Saliva removers; Dental appliances for receiving spittle
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
    • C07C2602/04—One of the condensed rings being a six-membered aromatic ring
    • C07C2602/10—One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Dentistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Medical Informatics (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Otolaryngology (AREA)
  • Oral & Maxillofacial Surgery (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Fremgangsmåte for den industrielle syntese av forbindelsen med formel (I). Anvendelse i syntesen av agomelatin.
NO20050739A 2004-02-13 2005-02-11 Ny fremgangsmate for syntesen av (7-metoksy-1-naftyl)acetonitril og dens anvendelse i syntesen av agomelatin NO333493B1 (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0401437A FR2866337B1 (fr) 2004-02-13 2004-02-13 Nouveau procede de synthese du (7-methoxy-1-naphtyl) acetonitrile et application a la synthese de l'aglomelatine

Publications (3)

Publication Number Publication Date
NO20050739D0 NO20050739D0 (no) 2005-02-11
NO20050739L true NO20050739L (no) 2005-08-15
NO333493B1 NO333493B1 (no) 2013-06-24

Family

ID=34685017

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20050739A NO333493B1 (no) 2004-02-13 2005-02-11 Ny fremgangsmate for syntesen av (7-metoksy-1-naftyl)acetonitril og dens anvendelse i syntesen av agomelatin

Country Status (33)

Country Link
US (2) US7470806B2 (no)
EP (1) EP1564205B1 (no)
JP (1) JP4157529B2 (no)
KR (1) KR100682698B1 (no)
CN (1) CN1300100C (no)
AR (1) AR047740A1 (no)
AT (1) ATE395326T1 (no)
AU (1) AU2005200615B8 (no)
BR (1) BRPI0502037B8 (no)
CA (1) CA2495975A1 (no)
CY (1) CY1111081T1 (no)
DE (1) DE602005006634D1 (no)
DK (1) DK1564205T3 (no)
EA (1) EA007787B1 (no)
ES (1) ES2308409T3 (no)
FR (1) FR2866337B1 (no)
GE (1) GEP20063929B (no)
HK (1) HK1078564A1 (no)
HR (1) HRP20080315T3 (no)
MA (1) MA27516A1 (no)
ME (1) ME01403B (no)
MX (1) MXPA05001636A (no)
MY (1) MY140089A (no)
NO (1) NO333493B1 (no)
NZ (1) NZ538193A (no)
PL (1) PL1564205T3 (no)
PT (1) PT1564205E (no)
RS (1) RS50594B (no)
SG (1) SG114705A1 (no)
SI (1) SI1564205T1 (no)
UA (1) UA79623C2 (no)
WO (1) WO2005077889A1 (no)
ZA (1) ZA200501255B (no)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2580183B1 (en) 2010-06-10 2014-07-23 Gador S.A. New process for the preparation of n-[2-(7-methoxy-1-naphthyl)-ethyl]acetamide
WO2013054273A2 (en) 2011-10-11 2013-04-18 Ranbaxy Laboratories Limited Process for the preparation of agomelatine
US20140336380A1 (en) 2011-12-01 2014-11-13 Ranbaxy Laboratories Limited Process for the preparation of agomelatine
ITMI20121444A1 (it) 2012-08-27 2014-02-28 Procos Spa Processo per la produzione di agomelatine
FR3014434B1 (fr) * 2013-12-05 2015-12-25 Servier Lab Nouveau procede de synthese du 7-methoxy-naphtalene-1-carbaldehyde et application a la synthese de l'agomelatine
CN112574066A (zh) * 2019-09-27 2021-03-30 江苏豪森药业集团有限公司 一种阿戈美拉汀中间体的制备方法
CN111377829A (zh) * 2020-04-10 2020-07-07 苏州敬业医药化工有限公司 一种7-甲氧基-1-萘乙腈的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4327022A (en) * 1973-08-16 1982-04-27 Sterling Drug Inc. Heterocyclic alkyl naphthols
US4169108A (en) * 1973-08-16 1979-09-25 Sterling Drug Inc. 5(OR 6)-[(Substituted-amino)alkyl]-2,3-naphthalenediols
US3931188A (en) * 1974-05-06 1976-01-06 Bristol-Myers Company 3-Hydroxy-5,6-benzomorphinan derivatives
US3992403A (en) * 1975-05-30 1976-11-16 Schering Corporation 2-Imidazolines and their use as hypoglycemic agents
FR2658818B1 (fr) * 1990-02-27 1993-12-31 Adir Cie Nouveaux derives a structure naphtalenique, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.

Also Published As

Publication number Publication date
CA2495975A1 (fr) 2005-08-13
SI1564205T1 (sl) 2008-08-31
PL1564205T3 (pl) 2008-09-30
DE602005006634D1 (de) 2008-06-26
ATE395326T1 (de) 2008-05-15
AU2005200615B2 (en) 2011-05-12
ME01403B (me) 2010-05-07
FR2866337B1 (fr) 2006-05-26
SG114705A1 (en) 2005-09-28
CN1300100C (zh) 2007-02-14
KR100682698B1 (ko) 2007-02-15
UA79623C2 (en) 2007-07-10
EA007787B1 (ru) 2007-02-27
ES2308409T3 (es) 2008-12-01
GEP20063929B (en) 2006-09-25
ZA200501255B (en) 2005-11-30
HK1078564A1 (en) 2006-03-17
AU2005200615B8 (en) 2011-05-26
CN1680297A (zh) 2005-10-12
FR2866337A1 (fr) 2005-08-19
AU2005200615A1 (en) 2005-09-01
CY1111081T1 (el) 2015-06-11
JP4157529B2 (ja) 2008-10-01
NO333493B1 (no) 2013-06-24
PT1564205E (pt) 2008-06-19
DK1564205T3 (da) 2008-09-29
US20090118544A1 (en) 2009-05-07
NZ538193A (en) 2005-12-23
MY140089A (en) 2009-11-30
MXPA05001636A (es) 2005-08-19
US20050182270A1 (en) 2005-08-18
EP1564205A1 (fr) 2005-08-17
US7994359B2 (en) 2011-08-09
HRP20080315T3 (en) 2008-07-31
EA200500204A1 (ru) 2005-08-25
BRPI0502037A (pt) 2005-11-16
KR20060041903A (ko) 2006-05-12
WO2005077889A1 (fr) 2005-08-25
RS50594B (sr) 2010-05-07
AR047740A1 (es) 2006-02-15
NO20050739D0 (no) 2005-02-11
MA27516A1 (fr) 2005-09-01
US7470806B2 (en) 2008-12-30
EP1564205B1 (fr) 2008-05-14
BRPI0502037B1 (pt) 2018-07-10
JP2005239717A (ja) 2005-09-08
BRPI0502037B8 (pt) 2021-05-25

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