NO20044974L - Imidazo [1,2-a]pyrazin-8-ylaminer, fremgangsmater for fremstilling og anvendelse derav - Google Patents
Imidazo [1,2-a]pyrazin-8-ylaminer, fremgangsmater for fremstilling og anvendelse deravInfo
- Publication number
- NO20044974L NO20044974L NO20044974A NO20044974A NO20044974L NO 20044974 L NO20044974 L NO 20044974L NO 20044974 A NO20044974 A NO 20044974A NO 20044974 A NO20044974 A NO 20044974A NO 20044974 L NO20044974 L NO 20044974L
- Authority
- NO
- Norway
- Prior art keywords
- preparation
- ylamines
- pyrazin
- imidazo
- methods
- Prior art date
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Hematology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Oncology (AREA)
- Physical Education & Sports Medicine (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Dermatology (AREA)
- Virology (AREA)
- Rheumatology (AREA)
- Communicable Diseases (AREA)
- Vascular Medicine (AREA)
- AIDS & HIV (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- Child & Adolescent Psychology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
Abstract
Et nytt preparat omfatter en forbindelse med formel 1, de farmasøytiske akseptable salter, hydrater, solvater, krystallformer, · diastereomerer, forløpermedikamenter eller blandinger derav. Preparatet er spesielt anvendelig i behandlingen av kinaserelaterte sykdommer.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US37421302P | 2002-04-19 | 2002-04-19 | |
PCT/US2003/012222 WO2003089434A2 (en) | 2002-04-19 | 2003-04-21 | IMIDAZO[1,2-a]PYRAZIN-8-YLAMINES METHOD OF MAKING AND METHOD OF USE THEREOF |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20044974L true NO20044974L (no) | 2004-11-16 |
Family
ID=29251159
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20044974A NO20044974L (no) | 2002-04-19 | 2004-11-16 | Imidazo [1,2-a]pyrazin-8-ylaminer, fremgangsmater for fremstilling og anvendelse derav |
Country Status (12)
Country | Link |
---|---|
US (1) | US6919340B2 (no) |
EP (1) | EP1509526A2 (no) |
JP (1) | JP2005530739A (no) |
KR (1) | KR20050008691A (no) |
CN (1) | CN100537571C (no) |
AU (1) | AU2003221731B2 (no) |
BR (1) | BR0309398A (no) |
CA (1) | CA2482991A1 (no) |
IL (1) | IL164703A0 (no) |
MX (1) | MXPA04010288A (no) |
NO (1) | NO20044974L (no) |
WO (1) | WO2003089434A2 (no) |
Families Citing this family (58)
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CA2482991A1 (en) | 2002-04-19 | 2003-10-30 | Cellular Genomics, Inc. | Imidazo[1,2-a]pyrazin-8-ylamines method of making and method of use thereof |
EP1388541A1 (en) | 2002-08-09 | 2004-02-11 | Centre National De La Recherche Scientifique (Cnrs) | Pyrrolopyrazines as kinase inhibitors |
AU2003270489A1 (en) | 2002-09-09 | 2004-03-29 | Cellular Genomics, Inc. | 6-ARYL-IMIDAZO(1,2-a)PYRAZIN-8-YLAMINES, METHOD OF MAKING, AND METHOD OF USE THEREOF |
PE20050081A1 (es) | 2002-09-23 | 2005-03-01 | Schering Corp | Nuevas imidazopirazinas como inhibidores de cinasas dependientes de ciclinas |
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DE602005013085D1 (de) * | 2004-06-09 | 2009-04-16 | Oncalis Ag | Proteinkinaseinhibitoren |
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CA2667348A1 (en) * | 2006-11-03 | 2008-05-15 | University Of Maryland, Baltimore | Methods of using saha and bortezomib for treating multiple myeloma |
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-
2003
- 2003-04-21 CA CA002482991A patent/CA2482991A1/en not_active Abandoned
- 2003-04-21 CN CNB038144670A patent/CN100537571C/zh not_active Expired - Fee Related
- 2003-04-21 IL IL16470303A patent/IL164703A0/xx unknown
- 2003-04-21 AU AU2003221731A patent/AU2003221731B2/en not_active Ceased
- 2003-04-21 MX MXPA04010288A patent/MXPA04010288A/es active IP Right Grant
- 2003-04-21 KR KR10-2004-7016841A patent/KR20050008691A/ko not_active Application Discontinuation
- 2003-04-21 WO PCT/US2003/012222 patent/WO2003089434A2/en active Application Filing
- 2003-04-21 JP JP2003586154A patent/JP2005530739A/ja active Pending
- 2003-04-21 US US10/419,682 patent/US6919340B2/en not_active Expired - Fee Related
- 2003-04-21 BR BR0309398-0A patent/BR0309398A/pt not_active Application Discontinuation
- 2003-04-21 EP EP03718470A patent/EP1509526A2/en not_active Withdrawn
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2004
- 2004-11-16 NO NO20044974A patent/NO20044974L/no not_active Application Discontinuation
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IL164703A0 (en) | 2005-12-18 |
AU2003221731B2 (en) | 2010-04-15 |
EP1509526A2 (en) | 2005-03-02 |
KR20050008691A (ko) | 2005-01-21 |
BR0309398A (pt) | 2005-02-01 |
US20030212073A1 (en) | 2003-11-13 |
US6919340B2 (en) | 2005-07-19 |
WO2003089434A2 (en) | 2003-10-30 |
WO2003089434A3 (en) | 2004-01-15 |
CN100537571C (zh) | 2009-09-09 |
JP2005530739A (ja) | 2005-10-13 |
CN1668619A (zh) | 2005-09-14 |
MXPA04010288A (es) | 2005-05-17 |
CA2482991A1 (en) | 2003-10-30 |
AU2003221731A1 (en) | 2003-11-03 |
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