NO20015274D0 - ACE-2 inhiberende forbindelser og fremgangsmåter for anvendelse derav - Google Patents
ACE-2 inhiberende forbindelser og fremgangsmåter for anvendelse deravInfo
- Publication number
- NO20015274D0 NO20015274D0 NO20015274A NO20015274A NO20015274D0 NO 20015274 D0 NO20015274 D0 NO 20015274D0 NO 20015274 A NO20015274 A NO 20015274A NO 20015274 A NO20015274 A NO 20015274A NO 20015274 D0 NO20015274 D0 NO 20015274D0
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- Prior art keywords
- ace
- methods
- inhibitory compounds
- inhibitory
- compounds
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- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/07—Optical isomers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/14—The ring being saturated
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pulmonology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Neurology (AREA)
- Physical Education & Sports Medicine (AREA)
- Urology & Nephrology (AREA)
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- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Hospice & Palliative Care (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Dermatology (AREA)
- Endocrinology (AREA)
- Epidemiology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Furan Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US13203499P | 1999-04-30 | 1999-04-30 | |
US17105299P | 1999-12-16 | 1999-12-16 | |
PCT/US2000/011550 WO2000066104A2 (en) | 1999-04-30 | 2000-04-28 | Ace-2 inhibiting compounds and methods of use thereof |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20015274D0 true NO20015274D0 (no) | 2001-10-29 |
NO20015274L NO20015274L (no) | 2001-12-28 |
Family
ID=26830036
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20015274A NO20015274L (no) | 1999-04-30 | 2001-10-29 | ACE-2 inhiberende forbindelser og fremgangsmåter for anvendelse derav |
Country Status (13)
Country | Link |
---|---|
US (1) | US6632830B1 (no) |
EP (1) | EP1183019A2 (no) |
JP (1) | JP2002543120A (no) |
KR (1) | KR20020008168A (no) |
CN (1) | CN1377259A (no) |
AU (1) | AU4500200A (no) |
BR (1) | BR0010166A (no) |
CA (1) | CA2372387A1 (no) |
IL (1) | IL146000A0 (no) |
MX (1) | MXPA01010993A (no) |
NO (1) | NO20015274L (no) |
TR (1) | TR200103094T2 (no) |
WO (1) | WO2000066104A2 (no) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7045532B2 (en) * | 1999-04-30 | 2006-05-16 | Millennium Pharmaceuticals, Inc. | ACE-2 modulating compounds and methods of use thereof |
EP1401864A1 (en) | 2001-06-04 | 2004-03-31 | Human Genome Sciences | Methods and compositions for modulating ace-2 activity |
WO2002098448A1 (en) | 2001-06-04 | 2002-12-12 | Human Genome Sciences, Inc. | Methods and compositions for modulating ace-2 activity |
RU2358699C2 (ru) | 2001-06-18 | 2009-06-20 | Ноувен Фамэсьютикэлз, Инк. | Композиция для чрескожной доставки лекарственного средства (варианты), способ ее получения и использование |
US6805878B2 (en) | 2001-09-13 | 2004-10-19 | Noven Pharmaceuticals, Inc. | Transdermal administration of ACE inhibitors |
SI2332582T1 (sl) | 2002-06-19 | 2014-03-31 | Apeiron Biologics Ag | Aktivacija ACE2 za zdravljenje srčne, pljučne in ledvične bolezni in hipertenzije |
US20040143009A1 (en) * | 2002-11-05 | 2004-07-22 | L'oreal | Amines, uses thereof |
US20050203168A1 (en) * | 2004-03-11 | 2005-09-15 | The Regents Of The University Of Michigan | Angiotensin converting enzyme inhibitor use for treatment and prevention of gastrointestinal disorders |
US8569277B2 (en) * | 2004-08-11 | 2013-10-29 | Palo Alto Investors | Methods of treating a subject for a condition |
TWI360539B (en) | 2004-10-28 | 2012-03-21 | Shionogi & Co | 3-carbamoyl-2-pyridone derivatives |
US7261742B2 (en) | 2005-10-13 | 2007-08-28 | S.C. Johnson & Son, Inc. | Method of deodorizing a textile |
US7407922B2 (en) * | 2005-10-13 | 2008-08-05 | S.C. Johnson & Son, Inc. | Deodorizing compositions |
EP2059234B1 (en) * | 2006-09-08 | 2011-11-02 | Ore Pharmaceuticals Inc. | Method for reducing or alleviating inflammation in the digestive tract |
US7842709B2 (en) * | 2006-09-08 | 2010-11-30 | Ore Pharmaceuticals Inc. | Method for treating inflammatory diseases of the digestive tract |
AU2006350707A1 (en) | 2006-11-08 | 2008-05-15 | Chongxi Yu | Transdermal delivery systems of peptides and related compounds |
US20090186014A1 (en) * | 2007-10-10 | 2009-07-23 | Ore Pharmaceuticals Inc. | Method for treatment of pancreatitis |
EP2077119A1 (de) * | 2007-12-21 | 2009-07-08 | Apeiron Biologics Forschungs- und Entwicklungsgesellschaft M.B.H. | Behandlung von Fibrosen und Lebererkrankungen |
WO2009114516A1 (en) * | 2008-03-10 | 2009-09-17 | Ore Pharmaceuticals Inc. | Therapy for disorders of the proximal digestive tract |
WO2010093804A1 (en) | 2009-02-12 | 2010-08-19 | Ore Pharmaceuticals, Inc. | Ace2 inhibitors for reducing gastrointestinal adverse effects of cytotoxic agents |
CA2761489C (en) | 2009-05-08 | 2021-07-20 | Lina Xu | High penetration prodrug compositions of peptides and peptide-related compounds |
CN102532260A (zh) * | 2011-11-29 | 2012-07-04 | 浙江省农业科学院 | 蚕蛹蛋白源二肽da及其用途 |
EP3039009B1 (en) | 2013-08-30 | 2019-05-01 | The University of British Columbia | Mao-b selective inhibitor compounds, pharmaceutical compositions thereof and uses thereof |
WO2018145268A1 (zh) * | 2017-02-08 | 2018-08-16 | 上海市第六人民医院 | 降压药在预防和治疗骨坏死中的应用 |
CN107577908B (zh) * | 2017-07-21 | 2020-07-03 | 浙江农林大学 | 一种新型功能配合物的分子设计方法 |
US11337909B2 (en) | 2017-11-29 | 2022-05-24 | Max-Delbrück-Centrum Für Molekulare Medizin In Der Helmholtz-Gemeinschaft | Methods for modulating pigmentation by angiotensin-converting enzyme 2 modulation |
JP6651493B2 (ja) * | 2017-12-05 | 2020-02-19 | チョンシー ユー | ペプチド及び関連化合物の経皮送達システム |
CN108191969B (zh) * | 2018-01-19 | 2021-01-01 | 渤海大学 | 两种来源于大西洋鳟鱼胶原蛋白的ace抑制肽 |
WO2021202399A1 (en) * | 2020-03-29 | 2021-10-07 | Kumuda, Inc. | Methods of treating coronavirus infections using angiotensin-converting enzyme 2 inhibitors |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
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US4344949A (en) * | 1980-10-03 | 1982-08-17 | Warner-Lambert Company | Substituted acyl derivatives of 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acids |
US4591648A (en) * | 1981-04-01 | 1986-05-27 | National Research Development Corp. | Histidine protection |
DE3219113A1 (de) * | 1982-05-21 | 1983-11-24 | Bayer Ag, 5090 Leverkusen | Verwendung von n-substituierten 2,3-diaminocarbonsaeuren in arzneimitteln und ihre herstellung |
US4542234A (en) * | 1983-10-06 | 1985-09-17 | Usv Pharmaceutical Corp. | Process for the separation of (S,S) diastereoisomers |
US4925969A (en) * | 1985-02-04 | 1990-05-15 | Kanegafuchi Kagaku Kogyo Kabushiki Kaisha | Process for preparing ethyl-alpha-amino-gamma-oxo-gamma-phenybutyrate derivatives |
US5665371A (en) * | 1985-05-20 | 1997-09-09 | Hoerrmann; Wilhelm | Medicines which contain derivatives of proline or hydroxyproline |
JPS6447754A (en) * | 1987-08-18 | 1989-02-22 | Kanegafuchi Chemical Ind | Novel process for producing alpha-(1-carboxyethyl)amino-gamma-phenylbutyric acid ethyl esters |
US5110799A (en) * | 1989-07-28 | 1992-05-05 | Merck & Co., Inc. | Antiherpetic agents |
US5827820A (en) * | 1992-04-06 | 1998-10-27 | Baxter International Inc. | Aqueous peritoneal dialysis solution |
JP2886748B2 (ja) * | 1992-09-17 | 1999-04-26 | 富士写真フイルム株式会社 | 写真用処理組成物及び処理方法 |
ES2113574T3 (es) * | 1993-06-01 | 1998-05-01 | Ono Pharmaceutical Co | Derivados del acido pentanoico. |
US5481018A (en) * | 1995-03-31 | 1996-01-02 | The Dow Chemical Company | Amino nitrile intermediate for the preparation of alanine diacetic acid |
WO1998000398A1 (en) * | 1996-06-28 | 1998-01-08 | University Of Southern California | Method for the synthesis of amines and amino acids with organoboron derivatives |
US6194556B1 (en) * | 1997-12-11 | 2001-02-27 | Millennium Pharmaceuticals, Inc. | Angiotensin converting enzyme homolog and therapeutic and diagnostic uses therfor |
US6989363B1 (en) * | 1997-12-11 | 2006-01-24 | Millennium Pharmaceuticals, Inc. | Angiotensin converting enzyme homolog and therapeutic and diagnostic uses therefor |
-
2000
- 2000-04-28 JP JP2000614989A patent/JP2002543120A/ja not_active Withdrawn
- 2000-04-28 TR TR2001/03094T patent/TR200103094T2/xx unknown
- 2000-04-28 KR KR1020017013877A patent/KR20020008168A/ko not_active Application Discontinuation
- 2000-04-28 WO PCT/US2000/011550 patent/WO2000066104A2/en not_active Application Discontinuation
- 2000-04-28 MX MXPA01010993A patent/MXPA01010993A/es unknown
- 2000-04-28 BR BR0010166-4A patent/BR0010166A/pt not_active IP Right Cessation
- 2000-04-28 AU AU45002/00A patent/AU4500200A/en not_active Abandoned
- 2000-04-28 CA CA002372387A patent/CA2372387A1/en not_active Abandoned
- 2000-04-28 CN CN00809781A patent/CN1377259A/zh active Pending
- 2000-04-28 EP EP00926478A patent/EP1183019A2/en not_active Withdrawn
- 2000-04-28 US US09/561,759 patent/US6632830B1/en not_active Expired - Fee Related
- 2000-04-28 IL IL14600000A patent/IL146000A0/xx unknown
-
2001
- 2001-10-29 NO NO20015274A patent/NO20015274L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
TR200103094T2 (tr) | 2002-03-21 |
EP1183019A2 (en) | 2002-03-06 |
NO20015274L (no) | 2001-12-28 |
AU4500200A (en) | 2000-11-17 |
WO2000066104A9 (en) | 2002-08-29 |
IL146000A0 (en) | 2002-07-25 |
CA2372387A1 (en) | 2000-11-09 |
CN1377259A (zh) | 2002-10-30 |
US6632830B1 (en) | 2003-10-14 |
BR0010166A (pt) | 2002-06-04 |
JP2002543120A (ja) | 2002-12-17 |
MXPA01010993A (es) | 2002-07-22 |
WO2000066104A3 (en) | 2001-06-28 |
KR20020008168A (ko) | 2002-01-29 |
WO2000066104A2 (en) | 2000-11-09 |
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