NO146428C - Analogifremgangsmaate ved fremstilling av terapeutisk aktive olefiniske derivater av aminosyrer - Google Patents

Analogifremgangsmaate ved fremstilling av terapeutisk aktive olefiniske derivater av aminosyrer

Info

Publication number
NO146428C
NO146428C NO760234A NO760234A NO146428C NO 146428 C NO146428 C NO 146428C NO 760234 A NO760234 A NO 760234A NO 760234 A NO760234 A NO 760234A NO 146428 C NO146428 C NO 146428C
Authority
NO
Norway
Prior art keywords
preparation
amino acids
therapeutic active
analogy procedure
active olefinic
Prior art date
Application number
NO760234A
Other languages
English (en)
Norwegian (no)
Other versions
NO760234L (fr
NO146428B (no
Inventor
Brian Walter Metcalf
Michel Jung
Original Assignee
Merrell Toraude & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Toraude & Co filed Critical Merrell Toraude & Co
Publication of NO760234L publication Critical patent/NO760234L/no
Publication of NO146428B publication Critical patent/NO146428B/no
Publication of NO146428C publication Critical patent/NO146428C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C237/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyrrole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO760234A 1975-03-18 1976-01-26 Analogifremgangsmaate ved fremstilling av terapeutisk aktive olefiniske derivater av aminosyrer NO146428C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/559,544 US3960927A (en) 1975-03-18 1975-03-18 Olefinic derivatives of amino acids

Publications (3)

Publication Number Publication Date
NO760234L NO760234L (fr) 1976-09-21
NO146428B NO146428B (no) 1982-06-21
NO146428C true NO146428C (no) 1982-09-29

Family

ID=24233995

Family Applications (1)

Application Number Title Priority Date Filing Date
NO760234A NO146428C (no) 1975-03-18 1976-01-26 Analogifremgangsmaate ved fremstilling av terapeutisk aktive olefiniske derivater av aminosyrer

Country Status (20)

Country Link
US (1) US3960927A (fr)
JP (1) JPS593988B2 (fr)
BE (1) BE839657A (fr)
CA (1) CA1077487A (fr)
CH (1) CH631696A5 (fr)
DE (1) DE2607620C2 (fr)
DK (1) DK145339C (fr)
ES (1) ES445659A1 (fr)
FR (1) FR2304329A1 (fr)
GB (1) GB1472525A (fr)
IE (1) IE42410B1 (fr)
IL (1) IL48912A (fr)
MX (1) MX4654E (fr)
NL (2) NL187161C (fr)
NO (1) NO146428C (fr)
NZ (1) NZ179834A (fr)
PH (1) PH12100A (fr)
PT (1) PT64761B (fr)
SE (1) SE442295B (fr)
ZA (1) ZA76411B (fr)

Families Citing this family (58)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4039549A (en) * 1975-03-18 1977-08-02 Merrell Toraude Et Compagnie Olefinic derivatives of amino acids
US4041041A (en) * 1975-03-18 1977-08-09 Merrell Toraude Et Compagnie Acetylene derivatives of amino acids
CA1121375A (fr) * 1977-07-01 1982-04-06 Brian W. Metcalf Derives d'amines et d'acides amines
US4139563A (en) * 1977-07-01 1979-02-13 Merrell Toraude Et Compagnie α-ACETYLENIC DERIVATIVES OF AMINES
CA1157030A (fr) * 1977-07-01 1983-11-15 Brian W. Metcalf ACIDES AMINES .alpha.-VINYLIQUES
US4147873A (en) * 1977-07-01 1979-04-03 Merrell Toraude Et Compagnie α-Vinyl derivatives of α-amino acids
US4326071A (en) * 1977-09-28 1982-04-20 Merrell Toraude Et Compagnie Halomethyl derivatives of gamma-aminobutyric acid and related compounds
US4187316A (en) * 1978-01-12 1980-02-05 Merrell Toraude Et Compagnie Substituted 1,5-cyclohexadiene carboxylic acid derivatives
US4254284A (en) * 1978-01-30 1981-03-03 Merrell Toraude Et Compagnie Process for preparing 4-aminohex-5-ynoic acid
US4178463A (en) * 1978-01-30 1979-12-11 Merrell Toraude Et Compagnie Process for making 4-aminohex-5-enoic acid
US4880793A (en) * 1978-07-24 1989-11-14 Merck & Co., Inc. Combination of thienamycin-type antibiotics with dipeptidase inhibitors
US5147868A (en) * 1978-07-24 1992-09-15 Merck & Co., Inc. Thienamycin renal peptidase inhibitors
US4323704A (en) * 1979-06-25 1982-04-06 Merrell Toraude Et Compagnie αAcetylene and α-vinyl derivatives of amino acids
US4539208A (en) * 1980-09-17 1985-09-03 Merck & Co., Inc. Combination of thienamycin-type antibiotics with dipeptidase inhibitors
US4372974A (en) * 1980-06-25 1983-02-08 New York University Anticonvulsive compositions and method of treating convulsive disorders
GB2120244B (en) * 1982-05-17 1985-05-01 Merrell Toraude & Co Aminoalkadiene derivative
GB2133002B (en) * 1982-12-30 1986-01-29 Merrell Toraude & Co Process for preparing 4-amino-5-hexenoic acid
GB8311804D0 (en) * 1983-04-29 1983-06-02 Merrell Toraude & Co Treatment of seizure disorders and pharmaceutical compositions
US4668703A (en) * 1983-07-07 1987-05-26 Syntex (U.S.A.) Inc. γ-allenyl-γ-aminobutyric acids
ATE31407T1 (de) * 1983-07-07 1988-01-15 Syntex Inc Gamma-allenyl-gamma-aminobuttersaeuren.
US4661510A (en) * 1983-08-17 1987-04-28 Syntex (U.S.A.) Inc. α-allenic-α-amino acids as enzyme inhibitors
US4588825A (en) * 1983-10-11 1986-05-13 Merrell Dow Pharmaceuticals Inc. Intermediates for the synthesis of 4-amino-4,5-dihydro-2-furancarboxylic acid
US4632994A (en) * 1983-11-04 1986-12-30 Gruppo Lepetit S.P.A. Process for decomposing N-oxide derivatives producing 5-vinyl-2-pyrrolidones
JPS6137389U (ja) * 1984-08-09 1986-03-08 永大産業株式会社 家具用の戸
DE3536146A1 (de) * 1985-10-10 1987-04-16 Degussa Verfahren zur enantioselektiven herstellung von (alpha)-vinyl-(alpha)-aminocarbonsaeuren
US4806680A (en) * 1986-03-17 1989-02-21 Merck & Co., Inc. 3-halovinylglycine antibacterial agents
US4727062A (en) * 1986-03-17 1988-02-23 Merck & Co., Inc. 3-Halovinylglycine antibacterial agents
AU629419B2 (en) 1989-11-07 1992-10-01 Aventis Inc. Process for the production of vinyl-gaba
US5208345A (en) * 1990-12-17 1993-05-04 Merrell Dow Pharmaceuticals Inc. Process for the production of (S)-vinyl and allenyl gaba
AU644919B2 (en) * 1990-12-17 1993-12-23 Aventisub Ii Inc. Process for the production of (S)-vinyl and allenyl gaba
EP0546230A1 (fr) * 1991-12-10 1993-06-16 Merrell Dow Pharmaceuticals Inc. Nouveau procédé pour la préparation de l'acide 4-amino 5-hexénoique
US5705660A (en) * 1994-08-22 1998-01-06 Board Of Regents, University Of Nebraska-Lincoln Method for the synthesis of α-oxiranyl amino acids
US7098206B2 (en) * 1998-01-21 2006-08-29 Smithkline Beecham Corporation Pharmaceutically active morpholinol
US6998400B2 (en) * 1998-01-22 2006-02-14 Smithkline Beecham Corporation Pharmaceutically active morpholinol
AU2349999A (en) 1998-01-29 1999-08-16 Sepracor, Inc. Pharmacological uses of pure (+) -bupropion
JP2002501892A (ja) * 1998-01-29 2002-01-22 セプラコア インコーポレーテッド 光学的に純粋な(−)−ビュープロピオンの薬学的使用
US6541520B1 (en) 1998-08-05 2003-04-01 Brookhaven Science Associates Treatment of addiction and addiction-related behavior
US6855820B2 (en) 1999-01-20 2005-02-15 Smithkline Beecham Corporation Pharmaceutically active morpholinol
US6734213B2 (en) 1999-01-20 2004-05-11 Smithkline Beecham Corporation Pharmaceutically active morpholinol
US6342496B1 (en) * 1999-03-01 2002-01-29 Sepracor Inc. Bupropion metabolites and methods of use
US6337328B1 (en) * 1999-03-01 2002-01-08 Sepracor, Inc. Bupropion metabolites and methods of use
EE200300249A (et) 2000-11-30 2003-10-15 Pfizer Products Inc. GABA agonistide ja aldoosreduktaasi inhibiitoritekombinatsioon
PT1337271E (pt) 2000-11-30 2005-01-31 Pfizer Prod Inc Combinacao de agonistas de gaba e inibidores de sorbitol desidrogenase
WO2004100992A2 (fr) * 2003-05-16 2004-11-25 Pfizer Products Inc. Combinaisons therapeutiques d'antipsychotiques atypiques avec des modulateurs de l'acide 4-aminobutanoique et/ou des medicaments anticonvulsivants
ES2515092T3 (es) 2003-12-11 2014-10-29 Sunovion Pharmaceuticals Inc. Combinación de un sedante y un modulador neurotransmisor y métodos de mejorar la calidad del sueño y de tratar la depresión
JP2007537151A (ja) * 2004-01-29 2007-12-20 ファイザー・プロダクツ・インク γ−アミノ酪酸モジュレータと5−HT1B受容体アンタゴニストとの組合せ
JP2009506069A (ja) 2005-08-26 2009-02-12 ブレインセルス,インコーポレイティド ムスカリン性受容体調節による神経発生
EP2258359A3 (fr) 2005-08-26 2011-04-06 Braincells, Inc. Neurogenèse par modulation des récepteurs muscariniques avec sabcomeline
JP2009512711A (ja) 2005-10-21 2009-03-26 ブレインセルス,インコーポレイティド Pde阻害による神経新生の調節
EP1942879A1 (fr) 2005-10-31 2008-07-16 Braincells, Inc. Modulation de la neurogenese dont la mediation est assuree par recepteur gaba
US20100216734A1 (en) 2006-03-08 2010-08-26 Braincells, Inc. Modulation of neurogenesis by nootropic agents
EP2021000A2 (fr) 2006-05-09 2009-02-11 Braincells, Inc. Neurogenèse par modulation de l'angiotensine
AU2007249435A1 (en) 2006-05-09 2007-11-22 Braincells, Inc. 5 HT receptor mediated neurogenesis
AU2007292848A1 (en) 2006-09-08 2008-03-13 Braincells, Inc. Combinations containing a 4-acylaminopyridine derivative
US20100184806A1 (en) 2006-09-19 2010-07-22 Braincells, Inc. Modulation of neurogenesis by ppar agents
CA2679741A1 (fr) * 2007-03-15 2008-09-18 Sun Pharma Advanced Research Company Ltd. Nouveaux promedicaments
WO2010099217A1 (fr) 2009-02-25 2010-09-02 Braincells, Inc. Modulation de neurogenèse à l'aide de combinaisons de d-cyclosérine
EP2537827B1 (fr) 2011-06-24 2014-06-11 Targeon SAS Procédé pour la préparation d'acide 4-amino-5-hexénoïque du succinimide

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2460708A (en) * 1946-03-22 1949-02-01 Merck & Co Inc Process for making acetamido dimethylacrylic acid
US2531595A (en) * 1949-06-09 1950-11-28 Sterling Drug Inc Preparation of alpha-acylamino-alpha-substituted-acetic acids
US2588969A (en) * 1949-11-26 1952-03-11 Eastman Kodak Co Certain acylamino-acrylates and-crotonates as insecticides
US3223729A (en) * 1962-06-06 1965-12-14 Sterling Drug Inc 3-allylhydantoic acid

Also Published As

Publication number Publication date
IE42410B1 (en) 1980-07-30
DE2607620A1 (de) 1976-09-30
DK145339C (da) 1983-03-21
ES445659A1 (es) 1977-06-01
IL48912A0 (en) 1976-03-31
ZA76411B (en) 1977-01-26
DK145339B (da) 1982-11-01
PT64761B (en) 1977-06-06
NO760234L (fr) 1976-09-21
US3960927A (en) 1976-06-01
JPS51125320A (en) 1976-11-01
CA1077487A (fr) 1980-05-13
DE2607620C2 (de) 1984-09-13
PT64761A (en) 1976-03-01
BE839657A (fr) 1976-07-16
NL7601116A (nl) 1976-09-21
SE442295B (sv) 1985-12-16
FR2304329A1 (fr) 1976-10-15
CH631696A5 (de) 1982-08-31
NL930125I2 (nl) 1997-08-01
IE42410L (en) 1976-09-18
JPS593988B2 (ja) 1984-01-27
NL187161C (nl) 1991-06-17
FR2304329B1 (fr) 1980-07-18
NO146428B (no) 1982-06-21
GB1472525A (en) 1977-05-04
NZ179834A (en) 1978-06-20
NL930125I1 (nl) 1993-11-01
SE7601205L (sv) 1976-09-19
MX4654E (es) 1982-07-19
PH12100A (en) 1978-11-02
NL187161B (nl) 1991-01-16
AU1071676A (en) 1977-08-11
DK31476A (da) 1976-09-19
IL48912A (en) 1980-09-16

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