NL170135C - Werkwijze ter bereiding van nieuwe p-acylamino n-gesubstitueerde benzamiden en werkwijze ter bereiding van een farmaceutisch preparaat met anti-ulcerwerking. - Google Patents

Werkwijze ter bereiding van nieuwe p-acylamino n-gesubstitueerde benzamiden en werkwijze ter bereiding van een farmaceutisch preparaat met anti-ulcerwerking.

Info

Publication number
NL170135C
NL170135C NLAANVRAGE7705565,A NL7705565A NL170135C NL 170135 C NL170135 C NL 170135C NL 7705565 A NL7705565 A NL 7705565A NL 170135 C NL170135 C NL 170135C
Authority
NL
Netherlands
Prior art keywords
preparing
acylamino
pharmaceutical preparation
substituted benzamides
ulcer effect
Prior art date
Application number
NLAANVRAGE7705565,A
Other languages
English (en)
Other versions
NL7705565A (nl
NL170135B (nl
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NL7705565A publication Critical patent/NL7705565A/nl
Publication of NL170135B publication Critical patent/NL170135B/nl
Application granted granted Critical
Publication of NL170135C publication Critical patent/NL170135C/nl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81Amides; Imides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81Amides; Imides
    • C07D213/82Amides; Imides in position 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
NLAANVRAGE7705565,A 1976-05-26 1977-05-20 Werkwijze ter bereiding van nieuwe p-acylamino n-gesubstitueerde benzamiden en werkwijze ter bereiding van een farmaceutisch preparaat met anti-ulcerwerking. NL170135C (nl)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/690,300 US4044147A (en) 1976-05-26 1976-05-26 N-(acyl)-p-amino-N'-(monosubstituted)-benzamide anti-ulcer agents

Publications (3)

Publication Number Publication Date
NL7705565A NL7705565A (nl) 1977-11-29
NL170135B NL170135B (nl) 1982-05-03
NL170135C true NL170135C (nl) 1982-10-01

Family

ID=24771930

Family Applications (1)

Application Number Title Priority Date Filing Date
NLAANVRAGE7705565,A NL170135C (nl) 1976-05-26 1977-05-20 Werkwijze ter bereiding van nieuwe p-acylamino n-gesubstitueerde benzamiden en werkwijze ter bereiding van een farmaceutisch preparaat met anti-ulcerwerking.

Country Status (10)

Country Link
US (1) US4044147A (nl)
JP (1) JPS52144640A (nl)
BE (1) BE855022A (nl)
DE (1) DE2723051C3 (nl)
DK (1) DK223177A (nl)
FR (1) FR2352790A1 (nl)
GB (1) GB1539862A (nl)
IE (1) IE44499B1 (nl)
LU (1) LU77403A1 (nl)
NL (1) NL170135C (nl)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2600513A1 (de) * 1976-01-08 1977-07-28 Hoechst Ag Acylamino(alkyl)benzolderivate und verfahren zu ihrer herstellung
US4500714A (en) * 1981-10-15 1985-02-19 Chugai Seiyaku Kabushiki Kaisha 3-Substituted-ureido-N-pyridyl benzamides
US4735956A (en) * 1985-09-13 1988-04-05 Merck & Co., Inc. Certain 1,4-dihydro-2,6-di-lower hydrocarbyl-4-heterocyclic-3,5-pyridine dicarboxylates which are useful as calcium channel blockers
US5658953A (en) * 1995-04-03 1997-08-19 Centaur Pharmaceuticals, Inc. Pharmaceutical compositions of acetamidobenzamide compounds for neurodegenerative disorders
US5643965A (en) * 1995-04-03 1997-07-01 Centaur Pharmaceuticals, Inc. Aminobenzamide compounds for the treatment of neurodegenerative disorders
US5955506A (en) * 1996-04-03 1999-09-21 Centaur Pharmaceuticals, Inc. Benzamides for neurodegenerative disorder treatment
EP1214293A1 (en) 1999-09-08 2002-06-19 Guilford Pharmaceuticals Inc. Non-peptidic cyclophilin binding compounds and their use
MXPA03006666A (es) 2001-01-25 2004-05-31 Guilford Pharm Inc Compuestos de union de ciclofilina carbociclicos trisubstituidos y su uso.
RU2008102236A (ru) * 2005-06-22 2009-07-27 РЕДДИ Манне САТЬЯНАРАЯНА (IN) Улучшенный способ получения эзетимиб
US20070049748A1 (en) * 2005-08-26 2007-03-01 Uppala Venkata Bhaskara R Preparation of ezetimibe

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2212268C3 (de) * 1971-03-15 1979-09-13 Sumitomo Chemical Co., Ltd., Osaka (Japan) N-Halogenacetylanilinoessigsäureester, Verfahren zu deren Herstellung und diese enthaltende herbicide Massen
JPS50157336A (nl) * 1974-06-11 1975-12-19

Also Published As

Publication number Publication date
NL7705565A (nl) 1977-11-29
US4044147A (en) 1977-08-23
BE855022A (fr) 1977-11-25
DE2723051A1 (de) 1977-12-01
DE2723051C3 (de) 1980-07-31
IE44499L (en) 1977-11-26
FR2352790A1 (fr) 1977-12-23
DE2723051B2 (de) 1979-11-22
DK223177A (da) 1977-11-27
GB1539862A (en) 1979-02-07
JPS574626B2 (nl) 1982-01-27
NL170135B (nl) 1982-05-03
JPS52144640A (en) 1977-12-02
LU77403A1 (nl) 1979-01-19
IE44499B1 (en) 1981-12-16
FR2352790B1 (nl) 1980-11-14

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Legal Events

Date Code Title Description
V1 Lapsed because of non-payment of the annual fee