NL170135C - Werkwijze ter bereiding van nieuwe p-acylamino n-gesubstitueerde benzamiden en werkwijze ter bereiding van een farmaceutisch preparaat met anti-ulcerwerking. - Google Patents
Werkwijze ter bereiding van nieuwe p-acylamino n-gesubstitueerde benzamiden en werkwijze ter bereiding van een farmaceutisch preparaat met anti-ulcerwerking.Info
- Publication number
- NL170135C NL170135C NLAANVRAGE7705565,A NL7705565A NL170135C NL 170135 C NL170135 C NL 170135C NL 7705565 A NL7705565 A NL 7705565A NL 170135 C NL170135 C NL 170135C
- Authority
- NL
- Netherlands
- Prior art keywords
- preparing
- acylamino
- pharmaceutical preparation
- substituted benzamides
- ulcer effect
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyridine Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US05/690,300 US4044147A (en) | 1976-05-26 | 1976-05-26 | N-(acyl)-p-amino-N'-(monosubstituted)-benzamide anti-ulcer agents |
Publications (3)
Publication Number | Publication Date |
---|---|
NL7705565A NL7705565A (nl) | 1977-11-29 |
NL170135B NL170135B (nl) | 1982-05-03 |
NL170135C true NL170135C (nl) | 1982-10-01 |
Family
ID=24771930
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NLAANVRAGE7705565,A NL170135C (nl) | 1976-05-26 | 1977-05-20 | Werkwijze ter bereiding van nieuwe p-acylamino n-gesubstitueerde benzamiden en werkwijze ter bereiding van een farmaceutisch preparaat met anti-ulcerwerking. |
Country Status (10)
Country | Link |
---|---|
US (1) | US4044147A (nl) |
JP (1) | JPS52144640A (nl) |
BE (1) | BE855022A (nl) |
DE (1) | DE2723051C3 (nl) |
DK (1) | DK223177A (nl) |
FR (1) | FR2352790A1 (nl) |
GB (1) | GB1539862A (nl) |
IE (1) | IE44499B1 (nl) |
LU (1) | LU77403A1 (nl) |
NL (1) | NL170135C (nl) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2600513A1 (de) * | 1976-01-08 | 1977-07-28 | Hoechst Ag | Acylamino(alkyl)benzolderivate und verfahren zu ihrer herstellung |
US4500714A (en) * | 1981-10-15 | 1985-02-19 | Chugai Seiyaku Kabushiki Kaisha | 3-Substituted-ureido-N-pyridyl benzamides |
US4735956A (en) * | 1985-09-13 | 1988-04-05 | Merck & Co., Inc. | Certain 1,4-dihydro-2,6-di-lower hydrocarbyl-4-heterocyclic-3,5-pyridine dicarboxylates which are useful as calcium channel blockers |
US5658953A (en) * | 1995-04-03 | 1997-08-19 | Centaur Pharmaceuticals, Inc. | Pharmaceutical compositions of acetamidobenzamide compounds for neurodegenerative disorders |
US5643965A (en) * | 1995-04-03 | 1997-07-01 | Centaur Pharmaceuticals, Inc. | Aminobenzamide compounds for the treatment of neurodegenerative disorders |
US5955506A (en) * | 1996-04-03 | 1999-09-21 | Centaur Pharmaceuticals, Inc. | Benzamides for neurodegenerative disorder treatment |
EP1214293A1 (en) | 1999-09-08 | 2002-06-19 | Guilford Pharmaceuticals Inc. | Non-peptidic cyclophilin binding compounds and their use |
MXPA03006666A (es) | 2001-01-25 | 2004-05-31 | Guilford Pharm Inc | Compuestos de union de ciclofilina carbociclicos trisubstituidos y su uso. |
RU2008102236A (ru) * | 2005-06-22 | 2009-07-27 | РЕДДИ Манне САТЬЯНАРАЯНА (IN) | Улучшенный способ получения эзетимиб |
US20070049748A1 (en) * | 2005-08-26 | 2007-03-01 | Uppala Venkata Bhaskara R | Preparation of ezetimibe |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2212268C3 (de) * | 1971-03-15 | 1979-09-13 | Sumitomo Chemical Co., Ltd., Osaka (Japan) | N-Halogenacetylanilinoessigsäureester, Verfahren zu deren Herstellung und diese enthaltende herbicide Massen |
JPS50157336A (nl) * | 1974-06-11 | 1975-12-19 |
-
1976
- 1976-05-26 US US05/690,300 patent/US4044147A/en not_active Expired - Lifetime
-
1977
- 1977-03-01 IE IE441/77A patent/IE44499B1/en unknown
- 1977-05-20 NL NLAANVRAGE7705565,A patent/NL170135C/nl not_active IP Right Cessation
- 1977-05-20 DK DK223177A patent/DK223177A/da unknown
- 1977-05-21 DE DE2723051A patent/DE2723051C3/de not_active Expired
- 1977-05-23 JP JP5973877A patent/JPS52144640A/ja active Granted
- 1977-05-24 LU LU77403A patent/LU77403A1/xx unknown
- 1977-05-24 GB GB21872/77A patent/GB1539862A/en not_active Expired
- 1977-05-25 FR FR7715966A patent/FR2352790A1/fr active Granted
- 1977-05-25 BE BE177890A patent/BE855022A/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
NL7705565A (nl) | 1977-11-29 |
US4044147A (en) | 1977-08-23 |
BE855022A (fr) | 1977-11-25 |
DE2723051A1 (de) | 1977-12-01 |
DE2723051C3 (de) | 1980-07-31 |
IE44499L (en) | 1977-11-26 |
FR2352790A1 (fr) | 1977-12-23 |
DE2723051B2 (de) | 1979-11-22 |
DK223177A (da) | 1977-11-27 |
GB1539862A (en) | 1979-02-07 |
JPS574626B2 (nl) | 1982-01-27 |
NL170135B (nl) | 1982-05-03 |
JPS52144640A (en) | 1977-12-02 |
LU77403A1 (nl) | 1979-01-19 |
IE44499B1 (en) | 1981-12-16 |
FR2352790B1 (nl) | 1980-11-14 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
V1 | Lapsed because of non-payment of the annual fee |