NI201500142A - Derivados de 3-acetilamino-1 (fenil-heteroaril-aminocarbonil o fenil-heteroaril-carbonilamino) benceno para el tratamiento de desordenes hiperproliferativos. - Google Patents

Derivados de 3-acetilamino-1 (fenil-heteroaril-aminocarbonil o fenil-heteroaril-carbonilamino) benceno para el tratamiento de desordenes hiperproliferativos.

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Publication number
NI201500142A
NI201500142A NI201500142A NI201500142A NI201500142A NI 201500142 A NI201500142 A NI 201500142A NI 201500142 A NI201500142 A NI 201500142A NI 201500142 A NI201500142 A NI 201500142A NI 201500142 A NI201500142 A NI 201500142A
Authority
NI
Nicaragua
Prior art keywords
phenyl
acetylamino
heteroaryl
treatment
aminocarbonil
Prior art date
Application number
NI201500142A
Other languages
English (en)
Inventor
Thede Kai
Bender Eckhard
J Scott William
Richter Anja
Zorn Ludwig
Liu Ningshu
Mönning Ursula
Siegel Franziska
Golz Stefan
Hägebarth Andrea
Lienau Philip
Puehler Florian
Basting Daniel
Schneider Dirk
Möwes Manfred
Original Assignee
Bayer Pharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Pharma AG filed Critical Bayer Pharma AG
Publication of NI201500142A publication Critical patent/NI201500142A/es

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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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Abstract

La presente invención se relaciona con N - (fenil-heteroaril) -3-acetilamino-benzamidas sustituidas y N-[3-(acetilamino) fenil]-fenil - heteroaril - carboxamidas de fórmula general (I) como se describe y se define en la presente, con métodos de preparación de dichos compuestos, con compuestos intermediarios útiles para preparar dichos compuestos, con composiciones farmacéuticas y combinaciones que comprenden dichos compuestos y con el uso de dichos compuestos para la elaboración de una composición farmacéuticas para el tratamiento o profilaxis de una enfermedad.
NI201500142A 2013-03-20 2015-09-18 Derivados de 3-acetilamino-1 (fenil-heteroaril-aminocarbonil o fenil-heteroaril-carbonilamino) benceno para el tratamiento de desordenes hiperproliferativos. NI201500142A (es)

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