MX338610B - Composiciones farmaceuticas que comprenden sulbactam e inhibidor de beta-lactamasa. - Google Patents

Composiciones farmaceuticas que comprenden sulbactam e inhibidor de beta-lactamasa.

Info

Publication number
MX338610B
MX338610B MX2013015002A MX2013015002A MX338610B MX 338610 B MX338610 B MX 338610B MX 2013015002 A MX2013015002 A MX 2013015002A MX 2013015002 A MX2013015002 A MX 2013015002A MX 338610 B MX338610 B MX 338610B
Authority
MX
Mexico
Prior art keywords
sulbactam
beta
pharmaceutical compositions
lactamase inhibitor
acceptable salt
Prior art date
Application number
MX2013015002A
Other languages
English (en)
Other versions
MX2013015002A (es
Inventor
Manesh Vithalbhai Patel
Sachin Bhagwat
Original Assignee
Wockhardt Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wockhardt Ltd filed Critical Wockhardt Ltd
Publication of MX2013015002A publication Critical patent/MX2013015002A/es
Publication of MX338610B publication Critical patent/MX338610B/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41881,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/424Oxazoles condensed with heterocyclic ring systems, e.g. clavulanic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • A61K31/43Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • A61K31/431Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems containing further heterocyclic rings, e.g. ticarcillin, azlocillin, oxacillin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Se describen composiciones y métodos para tratar o prevenir infecciones bacterianas. Las composiciones farmacéuticas comprenden típicamente una cantidad farmacéuticamente efectiva de: (a) sulbactam o su sal farmacéuticamente aceptable, y (b) por lo menos un inhibidor de beta-lactamasa o una sal de ella, aceptable para uso farmacéutico, a condición de que el inhibidor de beta lactamasa no sea sulbactam.
MX2013015002A 2011-07-26 2011-10-04 Composiciones farmaceuticas que comprenden sulbactam e inhibidor de beta-lactamasa. MX338610B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN2125MU2011 2011-07-26
PCT/IB2011/054349 WO2013014496A1 (en) 2011-07-26 2011-10-04 Pharmaceutical compositions comprising sulbactam and beta-lactamase inhibitor

Publications (2)

Publication Number Publication Date
MX2013015002A MX2013015002A (es) 2014-10-22
MX338610B true MX338610B (es) 2016-04-25

Family

ID=44925586

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2013015002A MX338610B (es) 2011-07-26 2011-10-04 Composiciones farmaceuticas que comprenden sulbactam e inhibidor de beta-lactamasa.

Country Status (13)

Country Link
US (1) US9744160B2 (es)
EP (1) EP2736508A1 (es)
JP (1) JP5808860B2 (es)
KR (1) KR101737167B1 (es)
CN (1) CN103687598B (es)
AU (1) AU2011373911B2 (es)
BR (1) BR112013032711A2 (es)
CA (1) CA2842777C (es)
MX (1) MX338610B (es)
NZ (1) NZ616806A (es)
RU (1) RU2560846C1 (es)
WO (1) WO2013014496A1 (es)
ZA (1) ZA201307956B (es)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9095594B2 (en) * 2011-07-26 2015-08-04 Wockhardt Ltd. Pharmaceutical compositions comprising beta-lactam antibiotic, sulbactam and beta-lactamase inhibitor
US8962843B2 (en) 2012-03-30 2015-02-24 Cubist Pharmaceuticals, Inc. 1,3,4-oxadiazole and 1,3,4-thiadiazole beta-lactamase inhibitors
US8969570B2 (en) 2012-03-30 2015-03-03 Cubist Pharmaceuticals, Inc. Beta-lactamase inhibitors
JP2015512419A (ja) 2012-03-30 2015-04-27 キュービスト ファーマシューティカルズ, インコーポレイテッド イソオキザゾールβ−ラクタマーゼ阻害剤
US8916709B2 (en) 2012-03-30 2014-12-23 Cubist Pharmaceuticals, Inc. 1,2,4-oxadiazole and 1,2,4-thiadiazole β-lactamase inhibitors
WO2014152996A1 (en) 2013-03-14 2014-09-25 Cubist Pharmaceuticals, Inc. Crystalline form of a beta-lactamase inhibitor
US9120796B2 (en) 2013-10-02 2015-09-01 Cubist Pharmaceuticals, Inc. B-lactamase inhibitor picoline salt
RU2702361C2 (ru) * 2013-10-22 2019-10-08 Вокхардт Лимитед Фармацевтические композиции, содержащие антибактериальные агенты
US20160271118A1 (en) * 2013-10-30 2016-09-22 Wockhardt Limited Pharmaceutical compositions comprising antibacterial agents
JP2017507162A (ja) * 2014-03-14 2017-03-16 ウォックハート リミテッド 抗菌薬を含む医薬組成物
US20170151221A1 (en) * 2014-03-29 2017-06-01 Wockhardt Limited Pharmaceutical compositions comprising cefepime or sulbactam
WO2016081452A1 (en) 2014-11-17 2016-05-26 Entasis Therapeutics Limited Combination therapy for treatment of resistant bacterial infections
RU2589929C1 (ru) * 2015-08-12 2016-07-10 Олег Иванович Квасенков Способ производства хлебного кваса
WO2018053215A1 (en) 2016-09-16 2018-03-22 Entasis Therapeutics Limited Beta-lactamase inhibitor compounds
SG11201909443YA (en) 2017-05-08 2019-11-28 Entasis Therapeutics Inc Compounds and methods for treating bacterial infections
US11905286B2 (en) 2018-08-09 2024-02-20 Antabio Sas Diazabicyclooctanones as inhibitors of serine beta-lactamases
CN109864970A (zh) * 2019-04-22 2019-06-11 苏州东瑞制药有限公司 一种舒巴坦钠组合物无菌粉及其制备方法
CN113559099A (zh) * 2021-08-27 2021-10-29 丹诺医药(苏州)有限公司 包含舒巴坦和阿维巴坦的药物组合物及其应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1206261B1 (en) 1999-08-16 2006-03-08 Revaax Pharmaceuticals LLC Pharmaceutical compositions comprising clavulanic acid or derivative thereof for the treatment of behavioral diseases
US20090275552A1 (en) * 2006-04-28 2009-11-05 Mahesh Vithalbhai Patel Therapy for Treating Resistant Bacterial Infections
FR2951171A1 (fr) * 2009-10-09 2011-04-15 Novexel Nouveau sel de sodium d'un compose azabicyclique sous forme enantiomere cristallisee et nouvelles formes polymorphes et pseudopolymorphes ainsi que leur preparation
CN102106857B (zh) * 2009-12-29 2012-07-18 齐鲁动物保健品有限公司 注射用复方头孢噻呋钠冻干粉针剂

Also Published As

Publication number Publication date
BR112013032711A2 (pt) 2017-01-17
JP5808860B2 (ja) 2015-11-10
CA2842777A1 (en) 2013-01-31
NZ616806A (en) 2015-03-27
KR101737167B1 (ko) 2017-05-17
AU2011373911B2 (en) 2016-09-22
US20140094447A1 (en) 2014-04-03
US9744160B2 (en) 2017-08-29
JP2014521631A (ja) 2014-08-28
WO2013014496A1 (en) 2013-01-31
KR20140053900A (ko) 2014-05-08
RU2560846C1 (ru) 2015-08-20
MX2013015002A (es) 2014-10-22
ZA201307956B (en) 2015-01-28
AU2011373911A1 (en) 2013-11-07
CN103687598A (zh) 2014-03-26
EP2736508A1 (en) 2014-06-04
CA2842777C (en) 2015-12-29
CN103687598B (zh) 2016-03-16

Similar Documents

Publication Publication Date Title
MX338610B (es) Composiciones farmaceuticas que comprenden sulbactam e inhibidor de beta-lactamasa.
NZ617104A (en) Pharmaceutical compositions comprising beta-lactam antibiotic, sulbactam and beta-lactamase inhibitor
EP4349820A3 (en) Compounds and compositions for treating conditions associated with nlrp activity
PH12016501750A1 (en) Human plasma kallikrein inhibitors
NZ730809A (en) Methods for treating filoviridae virus infections
WO2013122888A3 (en) Methods of treating bacterial infections
PH12017500852A1 (en) Combination therapy for treatment of resistant bacterial infections
MX2019010602A (es) Inhibidores de cdk.
IN2014DN10670A (es)
PH12015501588B1 (en) Compounds and methods for treating bacterial infections
TN2012000458A1 (en) Uses of dgat1 inhibitors
EA032271B9 (ru) Вещества, фармацевтическая композиция и методы применения при лечении воспалительных заболеваний
MX2021010297A (es) Inhibidores de calicreina plasmatica humana.
NZ706734A (en) Pharmaceutical compositions useful for the treatment or control of bacterial infections
MX2015013151A (es) Métodos de tratamiento de disquinesia y trastornos relacionados.
AU2012225365A8 (en) Peptide deformylase inhibitors
MX2016005869A (es) Inhibidor de beta-lactamasa cristalina.
UA88315U (en) Antibacterial composition
JOP20120346B1 (ar) مركبات لعلاج ومنع الإلتصاق، وتركيبات صيدلية متعلقة بالمركب وطرق لمنع وعلاج الإلتصاقات
UA110834C2 (uk) Сполука-інгібітор сигнального шляху notch
MY182136A (en) Pharmaceutical compositions

Legal Events

Date Code Title Description
FG Grant or registration