MX2022015629A - Uso de vibegron para tratar vejiga sobreactiva. - Google Patents
Uso de vibegron para tratar vejiga sobreactiva.Info
- Publication number
- MX2022015629A MX2022015629A MX2022015629A MX2022015629A MX2022015629A MX 2022015629 A MX2022015629 A MX 2022015629A MX 2022015629 A MX2022015629 A MX 2022015629A MX 2022015629 A MX2022015629 A MX 2022015629A MX 2022015629 A MX2022015629 A MX 2022015629A
- Authority
- MX
- Mexico
- Prior art keywords
- vibegron
- overactive bladder
- treat overactive
- directed
- present disclosure
- Prior art date
Links
- DJXRIQMCROIRCZ-XOEOCAAJSA-N vibegron Chemical compound C1([C@H]([C@@H]2N[C@H](CC=3C=CC(NC(=O)[C@H]4N5C(=O)C=CN=C5CC4)=CC=3)CC2)O)=CC=CC=C1 DJXRIQMCROIRCZ-XOEOCAAJSA-N 0.000 title abstract 3
- 229950007643 vibegron Drugs 0.000 title abstract 3
- 206010020853 Hypertonic bladder Diseases 0.000 title abstract 2
- 208000009722 Overactive Urinary Bladder Diseases 0.000 title abstract 2
- 208000020629 overactive bladder Diseases 0.000 title abstract 2
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
Abstract
La presente divulgación se refiere a un método de tratamiento de vejiga sobreactiva que comprende administrar por vía oral a un sujeto que lo necesita una cantidad de desde aproximadamente 60 mg hasta aproximadamente 90 mg (por ejemplo, aproximadamente 75 mg) de vibegron al día. La presente divulgación también se refiere a una composición de dosificación unitaria farmacéutica que comprende desde aproximadamente 60 mg hasta aproximadamente 90 mg (por ejemplo, aproximadamente 75 mg) de vibegron para administración oral.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201762515996P | 2017-06-06 | 2017-06-06 | |
US201862635146P | 2018-02-26 | 2018-02-26 | |
US201862637961P | 2018-03-02 | 2018-03-02 |
Publications (1)
Publication Number | Publication Date |
---|---|
MX2022015629A true MX2022015629A (es) | 2023-01-11 |
Family
ID=62815097
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
MX2022015629A MX2022015629A (es) | 2017-06-06 | 2019-12-04 | Uso de vibegron para tratar vejiga sobreactiva. |
Country Status (13)
Country | Link |
---|---|
US (1) | US20210077495A1 (es) |
EP (1) | EP3634420A1 (es) |
JP (2) | JP2020522560A (es) |
KR (1) | KR20200012949A (es) |
CN (3) | CN117695286A (es) |
AU (1) | AU2018282104A1 (es) |
BR (1) | BR112019025636A2 (es) |
CA (1) | CA3064989A1 (es) |
CL (1) | CL2019003533A1 (es) |
IL (1) | IL271164A (es) |
MX (1) | MX2022015629A (es) |
PH (1) | PH12019502651A1 (es) |
WO (1) | WO2018224989A1 (es) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP3730141A4 (en) * | 2017-12-21 | 2021-10-13 | Kyorin Pharmaceutical Co., Ltd. | THERAPEUTIC FOR NIGHTLY POLLAKISURIA |
TW202038963A (zh) * | 2018-12-05 | 2020-11-01 | 瑞士商優洛凡特科學公司 | 維貝隆(vibegron)於治療患有良性***增生之男性中膀胱過動症症狀之用途 |
CN113840607A (zh) | 2019-03-18 | 2021-12-24 | 尤偌万科学有限公司 | 维贝格龙治疗膀胱过度活动症的用途 |
DE102020124101A1 (de) | 2020-02-04 | 2021-08-05 | Samsung Electronics Co., Ltd. | Elektronische vorrichtung mit einer speichervorrichtung und trainingsverfahren |
IL303911A (en) | 2020-12-22 | 2023-08-01 | Urovant Sciences Gmbh | Methods for dioxin monitoring using Vibergon to treat irritable bladder |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0015246D0 (en) * | 2000-06-22 | 2000-08-16 | Astrazeneca Ab | Method for the treatment of urinary incontinence |
PE20091825A1 (es) | 2008-04-04 | 2009-12-04 | Merck & Co Inc | Hidroximetil pirrolidinas como agonistas del receptor adrenergico beta 3 |
ES2584427T3 (es) | 2011-10-27 | 2016-09-27 | Merck Sharp & Dohme Corp. | Proceso para la preparación de agonistas beta 3 y productos intermedios |
WO2013062881A1 (en) | 2011-10-27 | 2013-05-02 | Merck Sharp & Dohme Corp. | Process for making beta 3 agonists and intermediates |
UA112028C2 (uk) * | 2012-12-14 | 2016-07-11 | Пфайзер Лімітед | Похідні імідазопіридазину як модулятори гамка-рецептора |
DK2968269T3 (da) | 2013-03-15 | 2019-10-07 | Merck Sharp & Dohme | Fremgangsmåde til fremstilling af beta-3-agonister og mellemprodukter |
-
2018
- 2018-06-06 EP EP18737031.7A patent/EP3634420A1/en active Pending
- 2018-06-06 AU AU2018282104A patent/AU2018282104A1/en active Pending
- 2018-06-06 KR KR1020197038625A patent/KR20200012949A/ko not_active Application Discontinuation
- 2018-06-06 WO PCT/IB2018/054069 patent/WO2018224989A1/en unknown
- 2018-06-06 JP JP2019567995A patent/JP2020522560A/ja active Pending
- 2018-06-06 CA CA3064989A patent/CA3064989A1/en active Pending
- 2018-06-06 CN CN202311666042.4A patent/CN117695286A/zh active Pending
- 2018-06-06 CN CN202311666478.3A patent/CN117695287A/zh active Pending
- 2018-06-06 BR BR112019025636-9A patent/BR112019025636A2/pt unknown
- 2018-06-06 CN CN201880045540.8A patent/CN110869022A/zh active Pending
- 2018-06-06 US US16/620,179 patent/US20210077495A1/en active Pending
-
2019
- 2019-11-25 PH PH12019502651A patent/PH12019502651A1/en unknown
- 2019-12-04 MX MX2022015629A patent/MX2022015629A/es unknown
- 2019-12-04 CL CL2019003533A patent/CL2019003533A1/es unknown
- 2019-12-04 IL IL271164A patent/IL271164A/en unknown
-
2023
- 2023-03-01 JP JP2023030625A patent/JP2023071826A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
CN117695286A (zh) | 2024-03-15 |
BR112019025636A2 (pt) | 2020-08-25 |
AU2018282104A1 (en) | 2019-12-12 |
IL271164A (en) | 2020-01-30 |
CA3064989A1 (en) | 2018-12-13 |
KR20200012949A (ko) | 2020-02-05 |
CN110869022A (zh) | 2020-03-06 |
PH12019502651A1 (en) | 2020-06-08 |
WO2018224989A1 (en) | 2018-12-13 |
US20210077495A1 (en) | 2021-03-18 |
JP2020522560A (ja) | 2020-07-30 |
CL2019003533A1 (es) | 2020-06-26 |
CN117695287A (zh) | 2024-03-15 |
EP3634420A1 (en) | 2020-04-15 |
JP2023071826A (ja) | 2023-05-23 |
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