MX2022015629A - Uso de vibegron para tratar vejiga sobreactiva. - Google Patents

Uso de vibegron para tratar vejiga sobreactiva.

Info

Publication number
MX2022015629A
MX2022015629A MX2022015629A MX2022015629A MX2022015629A MX 2022015629 A MX2022015629 A MX 2022015629A MX 2022015629 A MX2022015629 A MX 2022015629A MX 2022015629 A MX2022015629 A MX 2022015629A MX 2022015629 A MX2022015629 A MX 2022015629A
Authority
MX
Mexico
Prior art keywords
vibegron
overactive bladder
treat overactive
directed
present disclosure
Prior art date
Application number
MX2022015629A
Other languages
English (en)
Inventor
Stephen C Piscitelli
Paul Mudd
Original Assignee
Urovant Sciences Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Urovant Sciences Gmbh filed Critical Urovant Sciences Gmbh
Publication of MX2022015629A publication Critical patent/MX2022015629A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/10Drugs for disorders of the urinary system of the bladder

Abstract

La presente divulgación se refiere a un método de tratamiento de vejiga sobreactiva que comprende administrar por vía oral a un sujeto que lo necesita una cantidad de desde aproximadamente 60 mg hasta aproximadamente 90 mg (por ejemplo, aproximadamente 75 mg) de vibegron al día. La presente divulgación también se refiere a una composición de dosificación unitaria farmacéutica que comprende desde aproximadamente 60 mg hasta aproximadamente 90 mg (por ejemplo, aproximadamente 75 mg) de vibegron para administración oral.
MX2022015629A 2017-06-06 2019-12-04 Uso de vibegron para tratar vejiga sobreactiva. MX2022015629A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762515996P 2017-06-06 2017-06-06
US201862635146P 2018-02-26 2018-02-26
US201862637961P 2018-03-02 2018-03-02

Publications (1)

Publication Number Publication Date
MX2022015629A true MX2022015629A (es) 2023-01-11

Family

ID=62815097

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2022015629A MX2022015629A (es) 2017-06-06 2019-12-04 Uso de vibegron para tratar vejiga sobreactiva.

Country Status (13)

Country Link
US (1) US20210077495A1 (es)
EP (1) EP3634420A1 (es)
JP (2) JP2020522560A (es)
KR (1) KR20200012949A (es)
CN (3) CN117695286A (es)
AU (1) AU2018282104A1 (es)
BR (1) BR112019025636A2 (es)
CA (1) CA3064989A1 (es)
CL (1) CL2019003533A1 (es)
IL (1) IL271164A (es)
MX (1) MX2022015629A (es)
PH (1) PH12019502651A1 (es)
WO (1) WO2018224989A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3730141A4 (en) * 2017-12-21 2021-10-13 Kyorin Pharmaceutical Co., Ltd. THERAPEUTIC FOR NIGHTLY POLLAKISURIA
TW202038963A (zh) * 2018-12-05 2020-11-01 瑞士商優洛凡特科學公司 維貝隆(vibegron)於治療患有良性***增生之男性中膀胱過動症症狀之用途
CN113840607A (zh) 2019-03-18 2021-12-24 尤偌万科学有限公司 维贝格龙治疗膀胱过度活动症的用途
DE102020124101A1 (de) 2020-02-04 2021-08-05 Samsung Electronics Co., Ltd. Elektronische vorrichtung mit einer speichervorrichtung und trainingsverfahren
IL303911A (en) 2020-12-22 2023-08-01 Urovant Sciences Gmbh Methods for dioxin monitoring using Vibergon to treat irritable bladder

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0015246D0 (en) * 2000-06-22 2000-08-16 Astrazeneca Ab Method for the treatment of urinary incontinence
PE20091825A1 (es) 2008-04-04 2009-12-04 Merck & Co Inc Hidroximetil pirrolidinas como agonistas del receptor adrenergico beta 3
ES2584427T3 (es) 2011-10-27 2016-09-27 Merck Sharp & Dohme Corp. Proceso para la preparación de agonistas beta 3 y productos intermedios
WO2013062881A1 (en) 2011-10-27 2013-05-02 Merck Sharp & Dohme Corp. Process for making beta 3 agonists and intermediates
UA112028C2 (uk) * 2012-12-14 2016-07-11 Пфайзер Лімітед Похідні імідазопіридазину як модулятори гамка-рецептора
DK2968269T3 (da) 2013-03-15 2019-10-07 Merck Sharp & Dohme Fremgangsmåde til fremstilling af beta-3-agonister og mellemprodukter

Also Published As

Publication number Publication date
CN117695286A (zh) 2024-03-15
BR112019025636A2 (pt) 2020-08-25
AU2018282104A1 (en) 2019-12-12
IL271164A (en) 2020-01-30
CA3064989A1 (en) 2018-12-13
KR20200012949A (ko) 2020-02-05
CN110869022A (zh) 2020-03-06
PH12019502651A1 (en) 2020-06-08
WO2018224989A1 (en) 2018-12-13
US20210077495A1 (en) 2021-03-18
JP2020522560A (ja) 2020-07-30
CL2019003533A1 (es) 2020-06-26
CN117695287A (zh) 2024-03-15
EP3634420A1 (en) 2020-04-15
JP2023071826A (ja) 2023-05-23

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