MX2020013004A - Compuestos inhibidores del transportador de monoamina 2 (vmat2), composiciones, y metodos relacionados con los mismos. - Google Patents

Compuestos inhibidores del transportador de monoamina 2 (vmat2), composiciones, y metodos relacionados con los mismos.

Info

Publication number
MX2020013004A
MX2020013004A MX2020013004A MX2020013004A MX2020013004A MX 2020013004 A MX2020013004 A MX 2020013004A MX 2020013004 A MX2020013004 A MX 2020013004A MX 2020013004 A MX2020013004 A MX 2020013004A MX 2020013004 A MX2020013004 A MX 2020013004A
Authority
MX
Mexico
Prior art keywords
vmat2 inhibitor
compositions
inhibitor compounds
methods relating
methods
Prior art date
Application number
MX2020013004A
Other languages
English (en)
Inventor
Nicole Harriott
Christopher F O'brien
Original Assignee
Neurocrine Biosciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurocrine Biosciences Inc filed Critical Neurocrine Biosciences Inc
Publication of MX2020013004A publication Critical patent/MX2020013004A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Organic Chemistry (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)

Abstract

En la presente se proporcionan métodos para tratar trastornos psiquiátricos relacionados con el síndrome de supresión 22q11.2 y para seleccionar sujetos para tratamiento con un inhibidor de VMAT2. Los métodos proporcionados en la presente comprenden administrar un inhibidor de VMAT2 a un sujeto en necesidad del mismo.
MX2020013004A 2018-06-14 2019-06-13 Compuestos inhibidores del transportador de monoamina 2 (vmat2), composiciones, y metodos relacionados con los mismos. MX2020013004A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862684935P 2018-06-14 2018-06-14
PCT/US2019/037046 WO2019241555A1 (en) 2018-06-14 2019-06-13 Vmat2 inhibitor compounds, compositions, and methods relating thereto

Publications (1)

Publication Number Publication Date
MX2020013004A true MX2020013004A (es) 2021-02-17

Family

ID=67263041

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2020013004A MX2020013004A (es) 2018-06-14 2019-06-13 Compuestos inhibidores del transportador de monoamina 2 (vmat2), composiciones, y metodos relacionados con los mismos.

Country Status (16)

Country Link
EP (1) EP3806856A1 (es)
JP (1) JP2021528386A (es)
KR (1) KR20210021006A (es)
CN (1) CN112638387A (es)
AU (1) AU2019287524A1 (es)
BR (1) BR112020024018A2 (es)
CA (1) CA3100694A1 (es)
EA (1) EA202092750A1 (es)
IL (1) IL278758A (es)
JO (1) JOP20200298A1 (es)
MA (1) MA52896A (es)
MX (1) MX2020013004A (es)
PH (1) PH12020552088A1 (es)
SG (1) SG11202011544UA (es)
TW (1) TW202011963A (es)
WO (1) WO2019241555A1 (es)

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CA3051832A1 (en) 2017-01-27 2018-08-02 Neurocrine Bioscienes, Inc. Methods for the administration of certain vmat2 inhibitors
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EA202090932A1 (ru) 2017-10-10 2021-05-20 Нейрокрин Байосайенсиз, Инк Способы введения некоторых vmat2-ингибиторов
US10993941B2 (en) 2017-10-10 2021-05-04 Neurocrine Biosciences, Inc. Methods for the administration of certain VMAT2 inhibitors
JOP20200336A1 (ar) 2018-08-15 2020-12-22 Neurocrine Biosciences Inc طرق إعطاء مثبطات vmat2 معينة
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Also Published As

Publication number Publication date
AU2019287524A1 (en) 2020-12-24
PH12020552088A1 (en) 2021-08-02
EP3806856A1 (en) 2021-04-21
IL278758A (en) 2021-01-31
WO2019241555A1 (en) 2019-12-19
KR20210021006A (ko) 2021-02-24
TW202011963A (zh) 2020-04-01
JOP20200298A1 (ar) 2020-11-22
CA3100694A1 (en) 2019-12-19
MA52896A (fr) 2021-04-21
JP2021528386A (ja) 2021-10-21
EA202092750A1 (ru) 2021-05-13
CN112638387A (zh) 2021-04-09
SG11202011544UA (en) 2020-12-30
BR112020024018A2 (pt) 2021-02-23

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