MX2018002538A - Derivados de espinosina. - Google Patents
Derivados de espinosina.Info
- Publication number
- MX2018002538A MX2018002538A MX2018002538A MX2018002538A MX2018002538A MX 2018002538 A MX2018002538 A MX 2018002538A MX 2018002538 A MX2018002538 A MX 2018002538A MX 2018002538 A MX2018002538 A MX 2018002538A MX 2018002538 A MX2018002538 A MX 2018002538A
- Authority
- MX
- Mexico
- Prior art keywords
- derivatives
- spinosyn
- insecticides
- spinosyn derivatives
- spinosyns
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
- A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
- A01N43/22—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom rings with more than six members
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N45/00—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds having three or more carbocyclic rings condensed among themselves, at least one ring not being a six-membered ring
- A01N45/02—Biocides, pest repellants or attractants, or plant growth regulators, containing compounds having three or more carbocyclic rings condensed among themselves, at least one ring not being a six-membered ring having three carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D313/00—Heterocyclic compounds containing rings of more than six members having one oxygen atom as the only ring hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N2300/00—Combinations or mixtures of active ingredients covered by classes A01N27/00 - A01N65/48 with other active or formulation relevant ingredients, e.g. specific carrier materials or surfactants, covered by classes A01N25/00 - A01N65/48
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Environmental Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Zoology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Dermatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Saccharide Compounds (AREA)
- Compositions Of Macromolecular Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Medicinal Preparation (AREA)
Abstract
Se proveen composiciones que incluyen derivados de espinosinas y métodos de producción de derivados de espinosinas. Los derivados de espinosina descriptos en la presente incluyen derivados de espinosina funcionalizados en el doble enlace C5-C6 de la espinosina A para proveer un sistema de anillo adicional. El método produce derivados de espinosina que exhiben actividad hacia insectos, arácnidos, y/o nemátodos y que resultan de utilidad en los mercados agrícola y de la salud animal.
Applications Claiming Priority (6)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562214083P | 2015-09-03 | 2015-09-03 | |
| US201662290676P | 2016-02-03 | 2016-02-03 | |
| US201662303078P | 2016-03-03 | 2016-03-03 | |
| US201662303015P | 2016-03-03 | 2016-03-03 | |
| US201662380664P | 2016-08-29 | 2016-08-29 | |
| PCT/US2016/049870 WO2017040763A1 (en) | 2015-09-03 | 2016-09-01 | Spinosyn derivatives as insecticides |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2018002538A true MX2018002538A (es) | 2018-08-14 |
Family
ID=56940400
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2018002540A MX2018002540A (es) | 2015-09-03 | 2016-09-01 | Derivados de espinosina y metodos de preparacion. |
| MX2018002538A MX2018002538A (es) | 2015-09-03 | 2016-09-01 | Derivados de espinosina. |
| MX2018002539A MX2018002539A (es) | 2015-09-03 | 2016-09-02 | Derivados de espinosina y metodos de preparacion. |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2018002540A MX2018002540A (es) | 2015-09-03 | 2016-09-01 | Derivados de espinosina y metodos de preparacion. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2018002539A MX2018002539A (es) | 2015-09-03 | 2016-09-02 | Derivados de espinosina y metodos de preparacion. |
Country Status (12)
| Country | Link |
|---|---|
| US (3) | US10717756B2 (es) |
| EP (3) | EP3344612B1 (es) |
| JP (3) | JP2018532708A (es) |
| KR (3) | KR20180048871A (es) |
| CN (3) | CN108137529A (es) |
| AU (3) | AU2016317854A1 (es) |
| BR (2) | BR112018004313A2 (es) |
| CA (3) | CA2997540A1 (es) |
| CL (2) | CL2018000525A1 (es) |
| IL (2) | IL257760A (es) |
| MX (3) | MX2018002540A (es) |
| WO (4) | WO2017040763A1 (es) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2018532708A (ja) | 2015-09-03 | 2018-11-08 | アグリメティス，エルエルシー | 殺虫剤としてのスピノシン誘導体 |
| CN110191888A (zh) * | 2017-01-13 | 2019-08-30 | 阿格里麦蒂斯有限责任公司 | 氮丙啶多杀菌素衍生物和制备方法 |
| KR20200111177A (ko) * | 2017-12-15 | 2020-09-28 | 타르서스 파마수티칼스, 아이엔씨. | 안검염을 치료하기 위한 이속사졸린 구충제 제제 및 방법 |
| AR116524A1 (es) * | 2018-10-04 | 2021-05-19 | Elanco Tiergesundheit Ag | Potenciación de tratamiento de helmintos |
| EP4079744A1 (en) | 2021-04-23 | 2022-10-26 | Acies Bio d.o.o. | Novel spinosyn prodrugs |
| CA3216243A1 (en) | 2021-04-23 | 2022-10-27 | Acies Bio D.O.O. | Novel spinosyn prodrugs |
| EP4101858A1 (en) | 2021-06-08 | 2022-12-14 | Acies Bio d.o.o. | Novel spinosyn compounds |
Family Cites Families (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1049845B (de) | 1957-01-04 | 1959-02-05 | Consortium Elektrochem Ind | Verfahren zur Herstellung von Carbonylverbindungen |
| US5362634A (en) | 1989-10-30 | 1994-11-08 | Dowelanco | Process for producing A83543 compounds |
| US5876980A (en) | 1995-04-11 | 1999-03-02 | Cytel Corporation | Enzymatic synthesis of oligosaccharides |
| US5922577A (en) | 1995-04-11 | 1999-07-13 | Cytel Corporation | Enzymatic synthesis of glycosidic linkages |
| US5728554A (en) | 1995-04-11 | 1998-03-17 | Cytel Corporation | Enzymatic synthesis of glycosidic linkages |
| US6030815A (en) | 1995-04-11 | 2000-02-29 | Neose Technologies, Inc. | Enzymatic synthesis of oligosaccharides |
| EP0837870B1 (en) * | 1995-06-14 | 2002-07-24 | Dow AgroSciences LLC | Synthetic modification to spinosyn compounds |
| US6001981A (en) * | 1996-06-13 | 1999-12-14 | Dow Agrosciences Llc | Synthetic modification of Spinosyn compounds |
| US6143526A (en) | 1998-03-09 | 2000-11-07 | Baltz; Richard H. | Biosynthetic genes for spinosyn insecticide production |
| TR200003818T2 (tr) | 1998-07-02 | 2001-06-21 | Eli Lilly And Company | İnsanda bit kontrolü için formülasyonlar. |
| US6927210B1 (en) | 1999-08-12 | 2005-08-09 | Eli Lilly And Company | Ectoparasiticidal aqueous suspension formulations of spinosyns |
| AU770879B2 (en) | 1999-08-12 | 2004-03-04 | Eli Lilly And Company | Ectoparasiticidal aqueous suspension formulations of spinosyns |
| TWI275592B (en) | 2001-03-21 | 2007-03-11 | Dow Agrosciences Llc | Synthetic derivatives of 21-butenyl and related spinosyns |
| US6919464B1 (en) | 2001-03-21 | 2005-07-19 | Dow Agrosciences Llc | Synthetic derivatives of 21-butenyl and related spinosyns |
| DK1492404T3 (da) | 2002-02-19 | 2012-04-23 | Dow Agrosciences Llc | Nye spinosyndannende polyketidsyntaser |
| JP4674702B2 (ja) | 2003-04-09 | 2011-04-20 | バイオジェネリクス エージー | グリコペギレ−ション法およびその方法により生成されたタンパク質／ペプチド |
| AU2004319804B2 (en) | 2004-04-29 | 2010-08-05 | Elanco Us Inc. | Use Of Spinosyns For Wound Healing |
| CA2737875C (en) | 2008-09-22 | 2015-11-24 | Christine Kritikou | Spinosyn antifouling compositions, methods of use thereof and articles protected from attachment of biofouling organisms |
| WO2010150100A1 (en) | 2009-06-24 | 2010-12-29 | Entarco Sa | The use of spinosyns and spinosyn compositions against diseases caused by protozoans, viral infections and cancer |
| KR20150080647A (ko) | 2010-01-25 | 2015-07-09 | 일라이 릴리 앤드 캄파니 | 말과 말파리 유충을 내부적으로 억제 또는 처리하기 위한 방법 |
| EP2635122A1 (en) | 2010-11-05 | 2013-09-11 | Eli Lilly and Company | Methods for inhibiting insect infestations |
| WO2012085683A1 (en) | 2010-12-22 | 2012-06-28 | Entarco Sa | The use of spinosyns and spinosyn compositions as local anesthetics and as antiarrhythmic agents |
| CN103402357B (zh) | 2010-12-29 | 2016-12-07 | 陶氏益农公司 | 防治昆虫的方法 |
| US9631195B2 (en) | 2011-12-28 | 2017-04-25 | Dow Agrosciences Llc | Identification and characterization of the spinactin biosysnthesis gene cluster from spinosyn producing saccharopolyspora spinosa |
| US9895388B1 (en) * | 2012-07-27 | 2018-02-20 | ParaPRO | Methods and compositions useful for controlling cutaneous mites |
| CN102977166B (zh) | 2012-12-05 | 2015-07-29 | 湖南化工研究院 | 13-硫醚取代多杀菌素衍生物及其制备方法 |
| WO2014115072A1 (en) * | 2013-01-22 | 2014-07-31 | Actelion Pharmaceuticals Ltd | Heterocyclic amide derivatives as p2x7 receptor antagonists |
| US9808008B2 (en) | 2013-10-22 | 2017-11-07 | Dow Agrosciences Llc | Synergistic pesticidal compositions and related methods |
| US9873639B1 (en) | 2015-07-17 | 2018-01-23 | Joe Doccola | Agricultural biomass as a matrix for release of plant active compounds |
| JP2018532708A (ja) | 2015-09-03 | 2018-11-08 | アグリメティス，エルエルシー | 殺虫剤としてのスピノシン誘導体 |
-
2016
- 2016-09-01 JP JP2018512331A patent/JP2018532708A/ja not_active Withdrawn
- 2016-09-01 AU AU2016317854A patent/AU2016317854A1/en not_active Abandoned
- 2016-09-01 MX MX2018002540A patent/MX2018002540A/es unknown
- 2016-09-01 US US15/757,317 patent/US10717756B2/en active Active
- 2016-09-01 KR KR1020187008942A patent/KR20180048871A/ko unknown
- 2016-09-01 JP JP2018512332A patent/JP2018531912A/ja not_active Withdrawn
- 2016-09-01 EP EP16767424.1A patent/EP3344612B1/en active Active
- 2016-09-01 BR BR112018004313A patent/BR112018004313A2/pt not_active Application Discontinuation
- 2016-09-01 MX MX2018002538A patent/MX2018002538A/es unknown
- 2016-09-01 AU AU2016317848A patent/AU2016317848A1/en not_active Abandoned
- 2016-09-01 CA CA2997540A patent/CA2997540A1/en not_active Abandoned
- 2016-09-01 WO PCT/US2016/049870 patent/WO2017040763A1/en active Application Filing
- 2016-09-01 WO PCT/US2016/049879 patent/WO2017040769A1/en active Application Filing
- 2016-09-01 US US15/757,204 patent/US10570166B2/en active Active
- 2016-09-01 BR BR112018004310A patent/BR112018004310A2/pt not_active Application Discontinuation
- 2016-09-01 CN CN201680061132.2A patent/CN108137529A/zh active Pending
- 2016-09-01 CN CN201680056085.2A patent/CN108026063A/zh active Pending
- 2016-09-01 KR KR1020187008943A patent/KR20180050340A/ko unknown
- 2016-09-01 EP EP16767084.3A patent/EP3344611B1/en active Active
- 2016-09-01 CA CA2997499A patent/CA2997499A1/en not_active Abandoned
- 2016-09-02 WO PCT/US2016/050028 patent/WO2017040878A1/en active Application Filing
- 2016-09-02 AU AU2016315860A patent/AU2016315860A1/en not_active Abandoned
- 2016-09-02 CN CN201680057361.7A patent/CN108137528A/zh active Pending
- 2016-09-02 WO PCT/US2016/050034 patent/WO2017040882A1/en active Application Filing
- 2016-09-02 JP JP2018512326A patent/JP2018532707A/ja not_active Withdrawn
- 2016-09-02 MX MX2018002539A patent/MX2018002539A/es unknown
- 2016-09-02 US US15/757,307 patent/US10711026B2/en active Active
- 2016-09-02 EP EP16766747.6A patent/EP3344610B1/en active Active
- 2016-09-02 KR KR1020187008941A patent/KR20180041755A/ko unknown
- 2016-09-02 CA CA2997639A patent/CA2997639A1/en not_active Abandoned
-
2018
- 2018-02-27 CL CL2018000525A patent/CL2018000525A1/es unknown
- 2018-02-27 CL CL2018000527A patent/CL2018000527A1/es unknown
- 2018-02-27 IL IL257760A patent/IL257760A/en unknown
- 2018-02-27 IL IL257759A patent/IL257759A/en unknown
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