MX2015013805A - Proceso para preparar sulfiminas y su conversion in situ en n-(2-amino-benzoil)-sulfiminas. - Google Patents

Proceso para preparar sulfiminas y su conversion in situ en n-(2-amino-benzoil)-sulfiminas.

Info

Publication number
MX2015013805A
MX2015013805A MX2015013805A MX2015013805A MX2015013805A MX 2015013805 A MX2015013805 A MX 2015013805A MX 2015013805 A MX2015013805 A MX 2015013805A MX 2015013805 A MX2015013805 A MX 2015013805A MX 2015013805 A MX2015013805 A MX 2015013805A
Authority
MX
Mexico
Prior art keywords
sulfimines
compound
preparing
formula
halocycloalkyl
Prior art date
Application number
MX2015013805A
Other languages
English (en)
Inventor
Karsten Körber
Timo Frassetto
Christopher Koradin
Thomas Zierke
Harald Jockers
Original Assignee
Basf Se
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Se filed Critical Basf Se
Publication of MX2015013805A publication Critical patent/MX2015013805A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C381/00—Compounds containing carbon and sulfur and having functional groups not covered by groups C07C301/00 - C07C337/00
    • C07C381/10—Compounds containing sulfur atoms doubly-bound to nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N37/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids
    • A01N37/18—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N<, e.g. carboxylic acid amides or imides; Thio analogues thereof
    • A01N37/28—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom having three bonds to hetero atoms with at the most two bonds to halogen, e.g. carboxylic acids containing the group —CO—N<, e.g. carboxylic acid amides or imides; Thio analogues thereof containing the group; Thio analogues thereof
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/02—Systems containing only non-condensed rings with a three-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

La presente invención se refiere a un proceso para preparar un compuesto de las Fórmulas (la) o (Ib), o una mezcla de estos, (ver fórmula) en donde R1 y R2 son, independientemente entre sí, hidrógeno, C1-C10-alquilo, C1-C10-haloalquilo, C3-C10-cicloalquilo, C3-C10-halocicloalquilo, o representan juntos una cadena alifática, o similar; A- es HSO4- o 1/2 SO42-; el proceso comprende la reacción de un sulfuro de la fórmula SR1R2 con ácido hidroxilamina-O-sulfónico de la fórmula; en donde la reacción se realiza en un medio acuoso en presencia de una base. La presente invención también se refiere a un proceso para preparar un compuesto de la fórmula (IV), (ver fórmula) en donde R3 es halógeno, ciano, C1-C8-alquilo, C1-C8-haloalquilo, C3-C8-cicloalquilo, C3-C8-halocicloalquilo, C2-C8-alquenilo, C2-C8-haloalquenilo, C1C8-alcoxi, fenilo o similar; R4 es hidrógeno, C1-C10-alquilo, C1-C10-haloalquilo, C3-C8-cicloalquilo, C3-C8-halocicloalquilo, C2-C10-alquenilo, C2-C10-haloalquenilo, fenilo o similar; p es 0, 1, 2, 3 o 4; y el proceso comprende: (iii) proporcionar el compuesto de las Fórmulas (la) o (Ib), o una mezcla de éstos, (iv) hacer reaccionar un compuesto de las fórmulas (la) o (Ib), o una mezcla de estos, obtenido en la etapa (i) con un compuesto de la fórmula (V) en presencia de una base, (ver formula).
MX2015013805A 2013-03-28 2014-03-27 Proceso para preparar sulfiminas y su conversion in situ en n-(2-amino-benzoil)-sulfiminas. MX2015013805A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP13161739 2013-03-28
PCT/EP2014/056164 WO2014154807A1 (en) 2013-03-28 2014-03-27 Process for preparing sulfimines and their in-situ conversion into n-(2-amino-benzoyl)-sulfimines

Publications (1)

Publication Number Publication Date
MX2015013805A true MX2015013805A (es) 2016-06-02

Family

ID=47997254

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2015013805A MX2015013805A (es) 2013-03-28 2014-03-27 Proceso para preparar sulfiminas y su conversion in situ en n-(2-amino-benzoil)-sulfiminas.

Country Status (10)

Country Link
US (1) US20160046572A1 (es)
EP (1) EP2978315A1 (es)
JP (1) JP2016520539A (es)
KR (1) KR20150135485A (es)
CN (1) CN105050405A (es)
AU (1) AU2014242984A1 (es)
BR (1) BR112015024815A2 (es)
IL (1) IL241296A0 (es)
MX (1) MX2015013805A (es)
WO (1) WO2014154807A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9556141B2 (en) 2011-11-21 2017-01-31 Basf Se Process for preparing N-substituted 1H-pyrazole-5-carboxylate compounds and derivatives thereof
US11297837B2 (en) 2016-02-19 2022-04-12 Basf Se Pesticidally activi mixtures comprising anthranilamide compounds
US10683256B2 (en) * 2016-08-22 2020-06-16 Basf Se Process for preparing substituted biphenyls

Family Cites Families (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3125920A1 (de) * 1981-07-01 1983-01-20 Basf Ag, 6700 Ludwigshafen "verfahren zur herstellung von sulfiden"
US4442111A (en) * 1981-07-25 1984-04-10 Dr. Karl Thomae Gesellschaft Mit Beschrankter Haftung Antithrombotic sulfimino and sulfoximino indolinones-2
IL118481A (en) * 1995-06-05 2000-08-31 Rhone Poulenc Agrochimie Sulfur compounds pesticidal compositions containing them and method of their application
AR036872A1 (es) 2001-08-13 2004-10-13 Du Pont Compuesto de antranilamida, composicion que lo comprende y metodo para controlar una plaga de invertebrados
TWI363756B (en) 2004-12-07 2012-05-11 Du Pont Method for preparing n-phenylpyrazole-1-carboxamides
AP2344A (en) 2005-07-07 2011-12-28 Basf Ag N-Thio-anthranilamid compounds and their use as pesticides.
HUP0600573A2 (en) 2006-07-12 2008-06-30 Laszlo Pirity Multifunction safety foil, especially fire-prevention foil
CN101142879A (zh) * 2007-12-07 2008-03-19 刘宝兴 种植孔和利用种植孔绿化破损山体的方法
TWI431000B (zh) 2008-03-05 2014-03-21 Du Pont 製備２－胺基－５－氰基苯甲酸衍生物之方法
BR112014003111A2 (pt) * 2011-08-12 2017-02-21 Basf Se “processo para preparar um composto de 1h-pirazol-5- carbonilcloreto n-substituído e processo para preparar um composto de sulfimina”
EP2742021A1 (en) * 2011-08-12 2014-06-18 Basf Se Aniline type compounds
JP2014522876A (ja) * 2011-08-12 2014-09-08 ビーエーエスエフ ソシエタス・ヨーロピア Ｎ−チオ−アントラニルアミド化合物、及び殺有害生物剤としてのそれらの使用
EP2742037B1 (en) * 2011-08-12 2015-10-14 Basf Se N-thio-anthranilamide compounds and their use as pesticides
IN2014CN01024A (es) * 2011-08-12 2015-04-10 Basf Se
US9556141B2 (en) * 2011-11-21 2017-01-31 Basf Se Process for preparing N-substituted 1H-pyrazole-5-carboxylate compounds and derivatives thereof
CN104023724A (zh) * 2011-12-21 2014-09-03 巴斯夫欧洲公司 N-硫代邻氨基苯甲酰胺化合物及其作为农药的用途
EP2794601B1 (en) * 2011-12-23 2019-02-20 Basf Se Isothiazoline compounds for combating invertebrate pests
CN104487439B (zh) * 2012-05-24 2017-06-09 巴斯夫欧洲公司 N‑硫代邻氨基苯甲酰胺化合物及其作为杀害虫剂的用途
CN104768377A (zh) * 2012-10-01 2015-07-08 巴斯夫欧洲公司 包含邻氨基苯甲酰胺类化合物的农药活性混合物
AR094139A1 (es) * 2012-10-01 2015-07-15 Basf Se Mezclas activas como plaguicidas, que comprenden compuestos de antranilamida
WO2014053406A1 (en) * 2012-10-01 2014-04-10 Basf Se Method of controlling ryanodine-modulator insecticide resistant insects
JP2015532274A (ja) * 2012-10-01 2015-11-09 ビーエーエスエフ ソシエタス・ヨーロピアＢａｓｆ Ｓｅ 栽培植物へのｎ−チオ−アントラニルアミド化合物の使用
BR112015005843A2 (pt) * 2012-10-01 2017-07-04 Basf Se utilização de pelo menos um composto ativo pesticida de antranilamida, métodos para proteger os vegetais do ataque ou infestação, para o controle ou combate dos insetos, para a proteção do material de propagação de vegetais e semente

Also Published As

Publication number Publication date
JP2016520539A (ja) 2016-07-14
US20160046572A1 (en) 2016-02-18
CN105050405A (zh) 2015-11-11
WO2014154807A1 (en) 2014-10-02
AU2014242984A1 (en) 2015-10-22
IL241296A0 (en) 2015-11-30
BR112015024815A2 (pt) 2017-07-18
EP2978315A1 (en) 2016-02-03
KR20150135485A (ko) 2015-12-02

Similar Documents

Publication Publication Date Title
MX2014001038A (es) Compuestos tipo anilina.
RS50512B (sr) Postupak za izradu (1s)-4,5-dimetoksi-1-(metilaminometil)- benzociklobutana i njegovih aditivnih soli kiselina kao i njegova primena za sintezu ivabradina i njegovih farmaceutski prihvatljivih aditivnih soli kiselina
MX2015002616A (es) Sintesis de bis(fluorosulfonil)imida.
RU2012138259A (ru) Способ получения ривароксабана
MX352470B (es) Disales de acido malonico y metodo para preparar dihaluros de malonilo.
MX2020006306A (es) Método novedoso para producir 4,5-dihidroisoxazol 5,5-disustituido.
MX355542B (es) Procedimiento de descarboxilacion de derivados de acido 3,5-bis(haloalquil)-pirazol-4-carboxilico.
MX2015013805A (es) Proceso para preparar sulfiminas y su conversion in situ en n-(2-amino-benzoil)-sulfiminas.
NZ598891A (en) Synthesis of a neurostimulative piperazine
IN2015DN00665A (es)
TW200738650A (en) Process for synthesis of aryloxy diaminopyrimidines
TR201007005A2 (tr) İmatinib baz üretim yöntemi
RU2009100738A (ru) Способ получения 2-пропил-3-этилхинолина
MD4392B1 (ro) Procedeu de sinteză a (2E)-3-(3,4-dimetoxifenil)prop-2-ennitrilului şi aplicarea acestuia în sinteza ivabradinei şi a sărurilor sale de adiţie cu un acid acceptabil farmaceutic
RU2013110311A (ru) Синтез соединений тиазолидиндиона
MX2012001067A (es) Procesos para la alquilacion de pirazoles.
RU2012100111A (ru) Способ получения 2- и 2,3-замещенных хинолинов
UA102091C2 (ru) Способ получения сульфонилпиролов как ингибиторов hdac
EA201300100A3 (ru) Способ ферментативного синтеза(7s)-3,4-диметоксибицикло[4.2.0]окта-1,3,5-триен-7-карбоновой кислоты или ее сложных эфиров, и применение для синтеза ивабрадина и его соли
AR053972A1 (es) Procedimiento para produccion de 2 - cloro-4- nitroimidazol
MD4443C1 (ro) Procedeu de sinteză a 3,4-dimetoxibiciclo[4.2.0]octa-1,3,5-trien-7-carbonitrilului şi aplicarea lui în sinteza ivabradinei şi a sărurilor sale de adiţie cu un acid acceptabil farmaceutic
UA114297C2 (uk) Сполуки анілінового типу
MX2014015622A (es) Procedimiento para preparar derivados de 2,2-difluoroetilamina por alquilacion de 2,2-difluoroetilamina.
RU2013138523A (ru) Способ получения производного ароматического амида карбоновой кислоты
RU2007122003A (ru) Способ получения 1-гидрокси-1,2-дигидро[60]фуллерена