MA45141A - Procédé de préparation de n-(5-(3-(7-(3-fluorophényl))-3 h-imidazo[4,5-c]pyridin-2-yl)-1h-indazol-5-yl)pyridin-3-yl)-3-méthylbutanamide - Google Patents

Procédé de préparation de n-(5-(3-(7-(3-fluorophényl))-3 h-imidazo[4,5-c]pyridin-2-yl)-1h-indazol-5-yl)pyridin-3-yl)-3-méthylbutanamide

Info

Publication number
MA45141A
MA45141A MA045141A MA45141A MA45141A MA 45141 A MA45141 A MA 45141A MA 045141 A MA045141 A MA 045141A MA 45141 A MA45141 A MA 45141A MA 45141 A MA45141 A MA 45141A
Authority
MA
Morocco
Prior art keywords
pyridin
methylbutanamide
indazol
imidazo
fluorophenyl
Prior art date
Application number
MA045141A
Other languages
English (en)
Other versions
MA45141B1 (fr
Inventor
Sunil Kumar Kc
Original Assignee
Samumed Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Samumed Llc filed Critical Samumed Llc
Priority claimed from PCT/US2017/035411 external-priority patent/WO2017210407A1/fr
Publication of MA45141A publication Critical patent/MA45141A/fr
Publication of MA45141B1 publication Critical patent/MA45141B1/fr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13Crystalline forms, e.g. polymorphs

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
MA45141A 2016-06-01 2017-06-01 Procédé de préparation de n-(5-(3-(7-(3-fluorophényl))-3 h-imidazo[4,5-c]pyridin-2-yl)-1h-indazol-5-yl)pyridin-3-yl)-3-méthylbutanamide MA45141B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662344170P 2016-06-01 2016-06-01
PCT/US2017/035411 WO2017210407A1 (fr) 2016-06-01 2017-06-01 Procédé de préparation de n-(5-(3-(7-(3-fluorophényl))-3 h-imidazo[4,5-c]pyridin-2-yl)-1h-indazol-5-yl)pyridin-3-yl)-3-méthylbutanamide

Publications (2)

Publication Number Publication Date
MA45141A true MA45141A (fr) 2019-04-10
MA45141B1 MA45141B1 (fr) 2022-12-30

Family

ID=84783663

Family Applications (1)

Application Number Title Priority Date Filing Date
MA45141A MA45141B1 (fr) 2016-06-01 2017-06-01 Procédé de préparation de n-(5-(3-(7-(3-fluorophényl))-3 h-imidazo[4,5-c]pyridin-2-yl)-1h-indazol-5-yl)pyridin-3-yl)-3-méthylbutanamide

Country Status (1)

Country Link
MA (1) MA45141B1 (fr)

Also Published As

Publication number Publication date
MA45141B1 (fr) 2022-12-30

Similar Documents

Publication Publication Date Title
IL263362B (en) Process for preparing n-(5-(3-(7-(3-fluorophenyl)-h3-imidazo[5,4-c]pyridin-2-yl)-h1-indazol-5-yl)pyridin-3-yl) -3-methylbutanamide
IL286912A (en) Process for the preparation of 4-phenyl-5-alkoxycarbonyl-2-thiazol-2-yl-1,4-dihydropyrimidin-6-yl]methyl]-3-oxo-5,6,8,8a-tetrahydro-1h-imidazo[1,5-a]pyrazin-2-yl]-carboxylic acid
SI3555097T1 (sl) Imidazo(4,5-d)pirolo(2,3-b)piridinske spojine kot zaviralci janus kinaz
IL270134B (en) A process for the preparation of compounds 3,2-dihydrothiazolo[2,3-a]pyrimidine-4-threat optical activity
PT3805233T (pt) Enantiómeros (r) e (s) de n-(5-(3-hidroxipirrolidin-1-il)-2 morfolinooxazolo[4,5-b]piridin-6-il)-2-(2-metilpiridin-4-il)oxazole-carboxamida como inibidores de irak4 para o tratamento de cancro
PT3500571T (pt) Compostos de imidazo[1,2-a] piridina, composições que os compreendem, métodos para o uso no tratamento de doenças e seus métodos de preparação
FR22C1058I2 (fr) Formulation de comprimé de 2-fluoro-n-méthyl-4-[7-(quinoline -6-ylméthyl) imidazo[1,2-b][1,2,4]triazine -2-yl]benzamide
IL269214B (en) Novel imidazo[5,4-c]quinoline derivatives as lrrk2 inhibitors
EP3362205A4 (fr) Procédés pour améliorer le traitement thermique de pièces coulées
IL276483B1 (en) A continuous process for the preparation of trazodone
IL269215A (en) Disubstituted imidazole[4,5-C]quinoline derivatives
PL3228619T3 (pl) Sposób wytwarzania apiksabanu
MA45141A (fr) Procédé de préparation de n-(5-(3-(7-(3-fluorophényl))-3 h-imidazo[4,5-c]pyridin-2-yl)-1h-indazol-5-yl)pyridin-3-yl)-3-méthylbutanamide
PL3478684T3 (pl) Nowe sposoby otrzymywania wemurafenibu
HUE047822T2 (hu) Immun- vagy gyulladásos betegségek és rák kezelésére alkalmas 7-(morfolin-4-il)pirazol[1,5-a]pirimidin-származékok
IL265985A (en) Process for the preparation of (3s,4s)-tetrahydrofuran-3-yl 4-isopropyl-6,7-dihydro-3h-imidazo[4,5-c]pyridine-5(4h)-carboxylate
MA52183A (fr) Procédé de préparation de 2,2-diméthylpipérazine