LV12375A - 1-(3-aminoindazol-5-il)-fenilmetil)-cikliskas urinvielas piemerotas ka HIV proteazes inhibitori - Google Patents
1-(3-aminoindazol-5-il)-fenilmetil)-cikliskas urinvielas piemerotas ka HIV proteazes inhibitoriInfo
- Publication number
- LV12375A LV12375A LV990076A LV990076A LV12375A LV 12375 A LV12375 A LV 12375A LV 990076 A LV990076 A LV 990076A LV 990076 A LV990076 A LV 990076A LV 12375 A LV12375 A LV 12375A
- Authority
- LV
- Latvia
- Prior art keywords
- hiv protease
- aminoindazol
- phenylmethyl
- protease inhibitors
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US2974596P | 1996-11-08 | 1996-11-08 | |
US74710496A | 1996-11-08 | 1996-11-08 | |
PCT/US1997/020035 WO1998020008A1 (en) | 1996-11-08 | 1997-11-04 | 1-(3-aminoindazol-5-yl)-3-phenylmethyl-cyclic ureas useful as hiv protease inhibitors |
Publications (2)
Publication Number | Publication Date |
---|---|
LV12375A true LV12375A (lv) | 1999-11-20 |
LV12375B LV12375B (lv) | 2000-04-20 |
Family
ID=26705293
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
LVP-99-76A LV12375B (lv) | 1996-11-08 | 1999-04-29 | 1-(3-aminoindazol-5-il)-fenilmetil)-cikliskas urīnvielas piemērotas kā hiv proteāzes inhibitori |
Country Status (21)
Country | Link |
---|---|
EP (1) | EP0937067B1 (lv) |
JP (1) | JP2001503428A (lv) |
KR (1) | KR20000053122A (lv) |
CN (1) | CN1235602A (lv) |
AT (1) | ATE244714T1 (lv) |
AU (1) | AU5165198A (lv) |
BR (1) | BR9712910A (lv) |
CA (1) | CA2270966A1 (lv) |
CZ (1) | CZ157599A3 (lv) |
DE (1) | DE69723456T2 (lv) |
EA (1) | EA199900452A1 (lv) |
EE (1) | EE9900188A (lv) |
ES (1) | ES2202645T3 (lv) |
HU (1) | HUP9904676A2 (lv) |
IL (1) | IL129727A0 (lv) |
LV (1) | LV12375B (lv) |
NO (1) | NO992228L (lv) |
PL (1) | PL333421A1 (lv) |
SI (1) | SI20074A (lv) |
SK (1) | SK59699A3 (lv) |
WO (1) | WO1998020008A1 (lv) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU6870098A (en) * | 1997-03-31 | 1998-10-22 | Du Pont Merck Pharmaceutical Company, The | Indazoles of cyclic ureas useful as hiv protease inhibitors |
US7135575B2 (en) | 2003-03-03 | 2006-11-14 | Array Biopharma, Inc. | P38 inhibitors and methods of use thereof |
PT1981851E (pt) | 2006-01-31 | 2012-04-13 | Array Biopharma Inc | Inibidores de cinase e processos para a sua utilização |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5610294A (en) * | 1991-10-11 | 1997-03-11 | The Du Pont Merck Pharmaceutical Company | Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors |
US5532357A (en) * | 1995-06-07 | 1996-07-02 | The Dupont Merck Pharmaceutical Company | Method for preparing N-monosubstituted and N,N'-disubstituted unsymmetrical cyclic ureas |
-
1997
- 1997-11-04 WO PCT/US1997/020035 patent/WO1998020008A1/en not_active Application Discontinuation
- 1997-11-04 EA EA199900452A patent/EA199900452A1/ru unknown
- 1997-11-04 SI SI9720072A patent/SI20074A/sl unknown
- 1997-11-04 EP EP97946494A patent/EP0937067B1/en not_active Expired - Lifetime
- 1997-11-04 IL IL12972797A patent/IL129727A0/xx unknown
- 1997-11-04 AU AU51651/98A patent/AU5165198A/en not_active Abandoned
- 1997-11-04 PL PL97333421A patent/PL333421A1/xx unknown
- 1997-11-04 JP JP52168198A patent/JP2001503428A/ja active Pending
- 1997-11-04 AT AT97946494T patent/ATE244714T1/de not_active IP Right Cessation
- 1997-11-04 BR BR9712910A patent/BR9712910A/pt not_active Application Discontinuation
- 1997-11-04 CZ CZ991575A patent/CZ157599A3/cs unknown
- 1997-11-04 DE DE69723456T patent/DE69723456T2/de not_active Expired - Fee Related
- 1997-11-04 KR KR1019990704048A patent/KR20000053122A/ko not_active Application Discontinuation
- 1997-11-04 HU HU9904676A patent/HUP9904676A2/hu unknown
- 1997-11-04 SK SK596-99A patent/SK59699A3/sk unknown
- 1997-11-04 ES ES97946494T patent/ES2202645T3/es not_active Expired - Lifetime
- 1997-11-04 CA CA002270966A patent/CA2270966A1/en not_active Abandoned
- 1997-11-04 CN CN97199419A patent/CN1235602A/zh active Pending
- 1997-11-04 EE EEP199900188A patent/EE9900188A/xx unknown
-
1999
- 1999-04-29 LV LVP-99-76A patent/LV12375B/lv unknown
- 1999-05-07 NO NO992228A patent/NO992228L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
EP0937067A1 (en) | 1999-08-25 |
SK59699A3 (en) | 1999-12-10 |
EE9900188A (et) | 1999-12-15 |
EA199900452A1 (ru) | 2000-02-28 |
NO992228L (no) | 1999-06-07 |
KR20000053122A (ko) | 2000-08-25 |
CA2270966A1 (en) | 1998-05-14 |
EP0937067B1 (en) | 2003-07-09 |
CZ157599A3 (cs) | 1999-11-17 |
PL333421A1 (en) | 1999-12-06 |
CN1235602A (zh) | 1999-11-17 |
WO1998020008A1 (en) | 1998-05-14 |
ES2202645T3 (es) | 2004-04-01 |
HUP9904676A2 (hu) | 2000-06-28 |
BR9712910A (pt) | 2000-03-21 |
AU5165198A (en) | 1998-05-29 |
DE69723456T2 (de) | 2004-05-27 |
IL129727A0 (en) | 2000-02-29 |
SI20074A (sl) | 2000-04-30 |
LV12375B (lv) | 2000-04-20 |
JP2001503428A (ja) | 2001-03-13 |
NO992228D0 (no) | 1999-05-07 |
ATE244714T1 (de) | 2003-07-15 |
DE69723456D1 (de) | 2003-08-14 |
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LV12375A (lv) | 1-(3-aminoindazol-5-il)-fenilmetil)-cikliskas urinvielas piemerotas ka HIV proteazes inhibitori | |
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