KR890002011A - 5-할로 게노-6-아미노-니코틴산 할라이드. 이의 제조방법 및 용도 - Google Patents

5-할로 게노-6-아미노-니코틴산 할라이드. 이의 제조방법 및 용도 Download PDF

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Publication number
KR890002011A
KR890002011A KR1019880008248A KR880008248A KR890002011A KR 890002011 A KR890002011 A KR 890002011A KR 1019880008248 A KR1019880008248 A KR 1019880008248A KR 880008248 A KR880008248 A KR 880008248A KR 890002011 A KR890002011 A KR 890002011A
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KR
South Korea
Prior art keywords
alkyl
amino
nicotinic acid
hydrogen
halogeno
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KR1019880008248A
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English (en)
Inventor
린델 한스
할렌바흐 베르너
Original Assignee
요아힘 그렘.루디 마이어
바이엘 아크티엔게젤샤프트
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Application filed by 요아힘 그렘.루디 마이어, 바이엘 아크티엔게젤샤프트 filed Critical 요아힘 그렘.루디 마이어
Publication of KR890002011A publication Critical patent/KR890002011A/ko

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/26—Radicals substituted by halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/73—Unsubstituted amino or imino radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

내용 없음

Description

5-할로 게노-6-아미노-니코틴산 할라이드. 이의 제조방법 및 용도
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (3)

  1. 일반식(Ⅰ)의 5-할로게노-6-아미노-니코틴산 할라이드.
    상기식에서, R1은 소수, 또는 알킬이며, R1은 수소 알킬 또는 아실이거나,R 및 R1은 이들이 결합된 질소원자와 함께 임의 치환된 헤테로사이클릭 래디칼을 형성하며,R2및 Hal은 할로겐이다.
  2. 일반식(Ⅱ)의 5-할로계노=6-아미노-니코틴산을 할로겐화시킴을 특징으로 하는, 일반적(Ⅰ)의 5-할로계노 -6-아미노-니코틴산 할라이드의 제조방법.
    상기식에서, R은 수소 또는 알킬이며, R1은 수소, 알킬 또는 아실이거나 R 및 R1은 이들이 결합된 질소원자와 함께 임의 치환된 헤테로사이클릭 래디칼을 헝성하며, R2및 Hal은 할로겐이다.
  3. 일반식(Ⅰ)의 5-할로게노-6-아미노-니코틴산-할라이드를 일반식(Ⅳ)의 화합물과 반응시킨 후 생성물을 가수분해하고 탈카복실화함을 특징으로 하는, 일반식(Ⅲ)외 5-아세틸피리딘의 제조를 위한 일반식(Ⅰ)의 5-할로계노-6-아미노-니코틴상 할라이드의 용도.
    상기식에서, R은 수소 또른 알킬이며, R1은 수소 알킬 또는 아실 이거나, R 및 R1은 이들이 결합된 질소원자와 함께 임의 치환된 헤테로사이클릭 라이칼을 형성하며, R2및 Hal온 할로겐이며, R3는 C1내지C3알킬이며, R4는 수소 또는 C1-C2-알킬이다.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019880008248A 1987-07-11 1988-07-04 5-할로 게노-6-아미노-니코틴산 할라이드. 이의 제조방법 및 용도 KR890002011A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19873723069 DE3723069A1 (de) 1987-07-11 1987-07-11 5-halogen-6-amino-nikotinsaeurehalogenide, ihre herstellung und ihre verwendung
DEP3723069.7 1987-07-11

Publications (1)

Publication Number Publication Date
KR890002011A true KR890002011A (ko) 1989-04-07

Family

ID=6331447

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019880008248A KR890002011A (ko) 1987-07-11 1988-07-04 5-할로 게노-6-아미노-니코틴산 할라이드. 이의 제조방법 및 용도

Country Status (12)

Country Link
US (1) US4895950A (ko)
EP (1) EP0302227B1 (ko)
JP (1) JPS6431768A (ko)
KR (1) KR890002011A (ko)
AT (1) ATE84524T1 (ko)
DD (1) DD274213A5 (ko)
DE (2) DE3723069A1 (ko)
DK (1) DK384188A (ko)
ES (1) ES2053626T3 (ko)
HU (1) HU199420B (ko)
IL (1) IL87043A (ko)
ZA (1) ZA884914B (ko)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100386086B1 (ko) * 2000-10-27 2003-06-02 김병수 해조류의 추출물을 이용한 건강식품 및 그의제조방법

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4006794A1 (de) * 1990-03-03 1991-09-05 Bayer Ag Verfahren zur herstellung von aminoethanolderivaten
WO2008093392A1 (ja) * 2007-01-29 2008-08-07 Fujifilm Finechemicals Co., Ltd. ２，３'－ビピリジル－６'－オンの製造方法
BR112016014906B1 (pt) * 2013-12-27 2019-08-06 Agro-Kanesho Co., Ltd. Método para produzir um derivado de éster benzílico de ácido 2-aminonicotínico

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4129734A (en) * 1976-12-03 1978-12-12 The Dow Chemical Company Substituted pyridine carbonyl halides and derivatives
US4596883A (en) * 1984-07-05 1986-06-24 Ppg Industries, Inc. Herbicidally active substituted diphenyl ethers
JPS6172753A (ja) * 1984-09-18 1986-04-14 Dainippon Pharmaceut Co Ltd ピリジルケトン誘導体
DE3615293A1 (de) * 1986-05-06 1987-11-12 Bayer Ag Verwendung von heteroarylethylaminen zur leistungsfoerderung bei tieren, heteroarylethylamine und verfahren zu ihrer herstellung

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100386086B1 (ko) * 2000-10-27 2003-06-02 김병수 해조류의 추출물을 이용한 건강식품 및 그의제조방법

Also Published As

Publication number Publication date
ES2053626T3 (es) 1994-08-01
DE3723069A1 (de) 1989-01-19
HUT48595A (en) 1989-06-28
EP0302227A3 (en) 1989-03-15
HU199420B (en) 1990-02-28
EP0302227A2 (de) 1989-02-08
JPS6431768A (en) 1989-02-02
DE3877455D1 (de) 1993-02-25
ATE84524T1 (de) 1993-01-15
US4895950A (en) 1990-01-23
IL87043A (en) 1992-03-29
DD274213A5 (de) 1989-12-13
ZA884914B (en) 1989-03-29
DK384188A (da) 1989-01-12
DK384188D0 (da) 1988-07-08
EP0302227B1 (de) 1993-01-13
IL87043A0 (en) 1988-12-30

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