KR100446068B1 - 구굴스테론의 제조방법 - Google Patents
구굴스테론의 제조방법 Download PDFInfo
- Publication number
- KR100446068B1 KR100446068B1 KR10-2001-0065507A KR20010065507A KR100446068B1 KR 100446068 B1 KR100446068 B1 KR 100446068B1 KR 20010065507 A KR20010065507 A KR 20010065507A KR 100446068 B1 KR100446068 B1 KR 100446068B1
- Authority
- KR
- South Korea
- Prior art keywords
- diol
- gugulsterone
- acetate
- transprenadiene
- pregnadiene
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J13/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17
- C07J13/007—Normal steroids containing carbon, hydrogen, halogen or oxygen having a carbon-to-carbon double bond from or to position 17 with double bond in position 17 (20)
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Steroid Compounds (AREA)
Abstract
Description
Claims (1)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR10-2001-0065507A KR100446068B1 (ko) | 2001-10-23 | 2001-10-23 | 구굴스테론의 제조방법 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR10-2001-0065507A KR100446068B1 (ko) | 2001-10-23 | 2001-10-23 | 구굴스테론의 제조방법 |
Publications (2)
Publication Number | Publication Date |
---|---|
KR20030033504A KR20030033504A (ko) | 2003-05-01 |
KR100446068B1 true KR100446068B1 (ko) | 2004-08-30 |
Family
ID=29566045
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
KR10-2001-0065507A KR100446068B1 (ko) | 2001-10-23 | 2001-10-23 | 구굴스테론의 제조방법 |
Country Status (1)
Country | Link |
---|---|
KR (1) | KR100446068B1 (ko) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100543542B1 (ko) * | 2003-04-24 | 2006-01-20 | 강헌중 | 4-안드로스텐-3,17-디온으로부터 구굴스테론의 제조방법및 이를 제조하기 위한 중간체 |
ES2376549T3 (es) * | 2003-04-24 | 2012-03-14 | Seoul National University Industry Foundation | Procedimiento para la preparación de guggulsteronas y guggulsterol. |
KR100543533B1 (ko) * | 2003-04-24 | 2006-01-20 | 강헌중 | 5-안드로스텐-3β-올-17-온으로부터4,17(20)-프로스타디엔-3,16-디온의 제조방법 및 이를제조하기 위한 중간체 |
KR100543544B1 (ko) * | 2003-04-24 | 2006-01-20 | 강헌중 | 테스토스테론으로부터 구굴스테론의 제조방법 및 이를제조하기 위한 중간체 |
KR100639655B1 (ko) * | 2003-04-24 | 2006-10-30 | 강헌중 | 16α,17α-에폭시프레그네놀론으로부터4,17(20)-프로스타디엔-3,16-디온의 제조방법 및 이를제조하기 위한 중간체 |
KR100543547B1 (ko) * | 2003-04-24 | 2006-01-20 | 강헌중 | 프로제스테론으로부터 구굴스테론의 제조방법 및 이를제조하기 위한 중간체 |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0447706A1 (en) * | 1990-03-22 | 1991-09-25 | Cipla Limited | A process for the preparation of pharmacologically active synthetic z and e steroisomeric mixture of guggulsterones |
-
2001
- 2001-10-23 KR KR10-2001-0065507A patent/KR100446068B1/ko active IP Right Grant
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0447706A1 (en) * | 1990-03-22 | 1991-09-25 | Cipla Limited | A process for the preparation of pharmacologically active synthetic z and e steroisomeric mixture of guggulsterones |
Also Published As
Publication number | Publication date |
---|---|
KR20030033504A (ko) | 2003-05-01 |
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FR2510584A1 (ko) |
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