JPWO2019236567A5 - - Google Patents

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Publication number
JPWO2019236567A5
JPWO2019236567A5 JP2020567774A JP2020567774A JPWO2019236567A5 JP WO2019236567 A5 JPWO2019236567 A5 JP WO2019236567A5 JP 2020567774 A JP2020567774 A JP 2020567774A JP 2020567774 A JP2020567774 A JP 2020567774A JP WO2019236567 A5 JPWO2019236567 A5 JP WO2019236567A5
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JP
Japan
Prior art keywords
moiety
peptidase
drug conjugate
binder
drug
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2020567774A
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English (en)
Japanese (ja)
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JP2021527042A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/035374 external-priority patent/WO2019236567A2/fr
Publication of JP2021527042A publication Critical patent/JP2021527042A/ja
Publication of JPWO2019236567A5 publication Critical patent/JPWO2019236567A5/ja
Pending legal-status Critical Current

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JP2020567774A 2018-06-04 2019-06-04 腫瘍微小環境活性化薬物・結合剤コンジュゲート、及びそれに関連する使用 Pending JP2021527042A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862680300P 2018-06-04 2018-06-04
US62/680,300 2018-06-04
PCT/US2019/035374 WO2019236567A2 (fr) 2018-06-04 2019-06-04 Conjugué médicament-liant activé par un micro-environnement tumoral et utilisations associées

Publications (2)

Publication Number Publication Date
JP2021527042A JP2021527042A (ja) 2021-10-11
JPWO2019236567A5 true JPWO2019236567A5 (fr) 2022-06-01

Family

ID=68769932

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020567774A Pending JP2021527042A (ja) 2018-06-04 2019-06-04 腫瘍微小環境活性化薬物・結合剤コンジュゲート、及びそれに関連する使用

Country Status (11)

Country Link
US (1) US20210353652A1 (fr)
EP (1) EP3801634A4 (fr)
JP (1) JP2021527042A (fr)
KR (1) KR20210016372A (fr)
CN (1) CN112601554A (fr)
AU (1) AU2019282150A1 (fr)
CA (1) CA3101640A1 (fr)
IL (2) IL279133B1 (fr)
SG (1) SG11202010890PA (fr)
TW (1) TWI834673B (fr)
WO (1) WO2019236567A2 (fr)

Families Citing this family (17)

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Publication number Priority date Publication date Assignee Title
KR20230149857A (ko) 2016-07-07 2023-10-27 더 보드 어브 트러스티스 어브 더 리랜드 스탠포드 주니어 유니버시티 항체-애쥬번트 접합체
US11583516B2 (en) 2016-09-07 2023-02-21 Trustees Of Tufts College Dash inhibitors, and uses related thereto
EP3937984A1 (fr) 2019-03-15 2022-01-19 Bolt Biotherapeutics, Inc. Immunoconjugués ciblant le her2
TW202110482A (zh) * 2019-05-24 2021-03-16 日商糖鎖工學研究所股份有限公司 新穎的人工蛋白質觸媒
TW202120500A (zh) 2019-08-02 2021-06-01 美商梅爾莎納醫療公司 干擾素基因刺激蛋白(sting)激動劑化合物及用途
TW202221030A (zh) * 2020-07-30 2022-06-01 英商阿法克塔生命科學有限公司 血清白蛋白結合多肽
TW202221031A (zh) * 2020-07-30 2022-06-01 英商阿法克塔生命科學有限公司 血清半衰期延長之pd-l1抑制多肽
US20230390409A1 (en) 2020-10-30 2023-12-07 Avacta Life Sciences Limited Fap-activated serum extended half-life therapeutic conjugates
EP4237011A1 (fr) * 2020-10-30 2023-09-06 Avacta Life Sciences Limited Conjugués thérapeutiques à demi-vie sérique étendue activés par enzyme
WO2022133288A1 (fr) 2020-12-17 2022-06-23 Trustees Of Tufts College Radiothéranostiques activés par fap et utilisations associées
WO2022234003A1 (fr) 2021-05-07 2022-11-10 Avacta Life Sciences Limited Polypeptides se liant à cd33 avec protéine stefin a
CN113648429B (zh) * 2021-07-06 2023-11-10 中山大学 靶向肿瘤周围细胞激活免疫的聚合物及其制备方法与应用
WO2023057946A1 (fr) 2021-10-07 2023-04-13 Avacta Life Sciences Limited Polypeptides sériques de liaison pd-l1 prolongés à demi-vie
TW202334196A (zh) 2021-10-07 2023-09-01 英商阿法克塔生命科學有限公司 Pd-l1結合多肽
CN114404429B (zh) * 2021-11-30 2023-06-30 重庆医科大学附属第二医院 一种纳米银修饰的单宁酸-铁网络的载药纳米复合物及其制备方法和逆转肿瘤耐药应用
KR20230121575A (ko) * 2022-02-10 2023-08-18 주식회사 아피셀테라퓨틱스 Cd40l에 특이적으로 결합하는 스테핀 a 단백질 변이체 및 이의 용도
WO2023218243A1 (fr) 2022-05-12 2023-11-16 Avacta Life Sciences Limited Protéines de fusion de liaison lag-3/pd-l1

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0807065D0 (en) * 2008-04-18 2008-05-21 Univ Leeds Novel scaffolds
DK3024851T3 (en) * 2013-07-25 2018-08-06 Cytomx Therapeutics Inc MULTI-SPECIFIC ANTIBODIES, MULTI-SPECIFICALLY ACTIVABLE ANTIBODIES, AND METHODS FOR USING IT
WO2015114166A2 (fr) * 2014-02-03 2015-08-06 Philochem Ag Conjugués médicamenteux ciblés
SI3154594T1 (sl) * 2014-06-13 2023-10-30 Bach Biosciences, Llc FAP-aktivirana terapevtska sredstva in z njimi povezane uporabe
CN112587672A (zh) * 2014-09-01 2021-04-02 博笛生物科技有限公司 用于***的抗-pd-l1结合物
TWI716362B (zh) * 2014-10-14 2021-01-21 瑞士商諾華公司 針對pd-l1之抗體分子及其用途
JP2018518506A (ja) * 2015-06-23 2018-07-12 ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company 大環状ベンゾジアゼピン二量体、その結合体の製造および使用
US20170158772A1 (en) * 2015-12-07 2017-06-08 Opi Vi - Ip Holdco Llc Compositions of antibody construct - agonist conjugates and methods of use thereof
MX2018015352A (es) * 2016-06-10 2019-03-28 Io Therapeutics Inc Subtipos de receptores y compuestos retinoides y rexinoides de funcion selectiva combinados con moduladores inmunitarios para inmunoterapia contra el cancer.
US11649285B2 (en) * 2016-08-03 2023-05-16 Bio-Techne Corporation Identification of VSIG3/VISTA as a novel immune checkpoint and use thereof for immunotherapy
US11583516B2 (en) * 2016-09-07 2023-02-21 Trustees Of Tufts College Dash inhibitors, and uses related thereto
WO2018053552A2 (fr) * 2016-09-19 2018-03-22 Cellerant Therapeutics, Inc. Isoquinolidinobenzodiazépines
GB201805963D0 (en) * 2018-04-11 2018-05-23 Avacta Life Sciences Ltd PD-L1 Binding Affirmers and Uses Related Thereto
US20220025061A1 (en) * 2018-12-10 2022-01-27 Bioxcel Therapeutics, Inc. Combination therapies for treating disease using an innate immunity modifier and an ox40 agonist

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