JPS6479192A - Moranoline derivative - Google Patents

Moranoline derivative

Info

Publication number
JPS6479192A
JPS6479192A JP62235499A JP23549987A JPS6479192A JP S6479192 A JPS6479192 A JP S6479192A JP 62235499 A JP62235499 A JP 62235499A JP 23549987 A JP23549987 A JP 23549987A JP S6479192 A JPS6479192 A JP S6479192A
Authority
JP
Japan
Prior art keywords
group
alkyl
positions
formula
moranoline
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP62235499A
Other languages
Japanese (ja)
Inventor
Akira Hasegawa
Makoto Kiso
Yoshiaki Yoshikuni
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Nippon Shinyaku Co Ltd
Original Assignee
Nippon Shinyaku Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nippon Shinyaku Co Ltd filed Critical Nippon Shinyaku Co Ltd
Priority to JP62235499A priority Critical patent/JPS6479192A/en
Publication of JPS6479192A publication Critical patent/JPS6479192A/en
Pending legal-status Critical Current

Links

Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

NEW MATERIAL:A derivative expressed by formula I [R<1> is H, alkyl or alkoxycarbonyl; R<2> and R<3> are H or together link to form a cyclic group and represent a group expressed by formula II (A is H, alkyl, or aryl); R<4> is acyl- substituted or unsubstituted amino group]. EXAMPLE:3-Acetamido-1,5-imino-1,3,5-trideoxy-D-glucose. USE:Useful as a medicinal composition having antimicrobial activity. PREPARATION:The N atom, 4- and 6-positions of moranoline are protected and the 2- and 3-positions are epoxidized. Azide group is then introduced using sodium azide, etc. The resultant compound is then reduced with palladium- carbon, etc., or acylated with ammonium formate, etc., and the protecting groups, as necessary, are removed to afford the aimed compound.
JP62235499A 1987-09-18 1987-09-18 Moranoline derivative Pending JPS6479192A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP62235499A JPS6479192A (en) 1987-09-18 1987-09-18 Moranoline derivative

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP62235499A JPS6479192A (en) 1987-09-18 1987-09-18 Moranoline derivative

Publications (1)

Publication Number Publication Date
JPS6479192A true JPS6479192A (en) 1989-03-24

Family

ID=16986933

Family Applications (1)

Application Number Title Priority Date Filing Date
JP62235499A Pending JPS6479192A (en) 1987-09-18 1987-09-18 Moranoline derivative

Country Status (1)

Country Link
JP (1) JPS6479192A (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5206251A (en) * 1992-04-01 1993-04-27 G. D. Searle & Co. 2- and 3- amino and azido derivatives of 1,5-iminosugars
US5216168A (en) * 1992-04-01 1993-06-01 G. D. Searle & Co. 2- and 3- amino and azido derivatives of 1,5-iminosugars

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5206251A (en) * 1992-04-01 1993-04-27 G. D. Searle & Co. 2- and 3- amino and azido derivatives of 1,5-iminosugars
US5216168A (en) * 1992-04-01 1993-06-01 G. D. Searle & Co. 2- and 3- amino and azido derivatives of 1,5-iminosugars
JPH0616631A (en) * 1992-04-01 1994-01-25 G D Searle & Co 2- and 3- amino azido derivatives of 1,5-iminosaccharides

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