JPS5495592A - Cephalosporin derivative and manufacture - Google Patents
Cephalosporin derivative and manufactureInfo
- Publication number
- JPS5495592A JPS5495592A JP15817278A JP15817278A JPS5495592A JP S5495592 A JPS5495592 A JP S5495592A JP 15817278 A JP15817278 A JP 15817278A JP 15817278 A JP15817278 A JP 15817278A JP S5495592 A JPS5495592 A JP S5495592A
- Authority
- JP
- Japan
- Prior art keywords
- manufacture
- cephalosporin derivative
- cephalosporin
- derivative
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19772758001 DE2758001A1 (de) | 1977-12-24 | 1977-12-24 | Cephalosporinderivate und verfahren zu ihrer herstellung |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5495592A true JPS5495592A (en) | 1979-07-28 |
JPH0132226B2 JPH0132226B2 (ja) | 1989-06-29 |
Family
ID=6027279
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP15817278A Granted JPS5495592A (en) | 1977-12-24 | 1978-12-23 | Cephalosporin derivative and manufacture |
Country Status (20)
Country | Link |
---|---|
US (1) | US4293550A (ja) |
EP (1) | EP0002765B1 (ja) |
JP (1) | JPS5495592A (ja) |
AT (1) | AT365599B (ja) |
AU (1) | AU534258B2 (ja) |
CA (1) | CA1109461A (ja) |
DE (2) | DE2758001A1 (ja) |
DK (1) | DK578978A (ja) |
EG (1) | EG13762A (ja) |
ES (1) | ES476109A1 (ja) |
FI (1) | FI66007C (ja) |
GR (1) | GR65234B (ja) |
HU (1) | HU184140B (ja) |
IE (1) | IE48147B1 (ja) |
IL (1) | IL56284A (ja) |
NO (1) | NO784366L (ja) |
NZ (1) | NZ189266A (ja) |
PH (1) | PH15925A (ja) |
PT (1) | PT68964A (ja) |
ZA (1) | ZA787209B (ja) |
Cited By (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5547688A (en) * | 1978-09-08 | 1980-04-04 | Fujisawa Pharmaceut Co Ltd | Novel cephem compound and its preparation |
JPS5657790A (en) * | 1979-10-02 | 1981-05-20 | Glaxo Group Ltd | Cephalosporin antibiotic |
JPS56142289A (en) * | 1980-02-23 | 1981-11-06 | Hoechst Ag | Cephalosporin derivative and manufacture |
JPS57131794A (en) * | 1980-12-31 | 1982-08-14 | Fujisawa Pharmaceut Co Ltd | Novel cephem compound or salt thereof, preparation of the same and preventing agent and remedy for microbism containing the same as active constituent |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4409214A (en) * | 1979-11-19 | 1983-10-11 | Fujisawa Pharmaceutical, Co., Ltd. | 7-Acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof |
US4427677A (en) * | 1980-12-31 | 1984-01-24 | Fujisawa Pharmaceutical Co., Ltd. | Cephem compounds |
EP0055465B1 (en) * | 1980-12-31 | 1989-08-23 | Fujisawa Pharmaceutical Co., Ltd. | 7-acylaminocephalosporanic acid derivatives and processes for the preparation thereof |
US4618606A (en) * | 1982-11-17 | 1986-10-21 | Toyama Chemical Co., Ltd. | Antibiotic 7-(thiazolyl)-3-(pyrazinylmethyl) or (pyridazinylmethyl) cephalosporins |
EP1059293A1 (en) * | 1995-10-12 | 2000-12-13 | Microcide Pharmaceuticals, Inc. | Novel amino chlorothiazole compounds |
IT1295935B1 (it) * | 1997-10-30 | 1999-05-28 | Acs Dobfar Spa | Derivati aminotiazolici utili nella preparazione di antibiotici b -lattamici |
TWI335332B (en) * | 2001-10-12 | 2011-01-01 | Theravance Inc | Cross-linked vancomycin-cephalosporin antibiotics |
JP5491421B2 (ja) | 2008-03-04 | 2014-05-14 | アリーナ ファーマシューティカルズ, インコーポレイテッド | 5−ht2cアゴニストである(r)−8−クロロ−1−メチル−2,3,4,5−テトラヒドロ−1h−3−ベンゾアゼピンに関連する中間体の調製のためのプロセス |
WO2011153206A1 (en) | 2010-06-02 | 2011-12-08 | Arena Pharmaceuticals, Inc. | Processes for the preparation of 5-ht2c receptor agonists |
SG188361A1 (en) | 2010-09-01 | 2013-04-30 | Arena Pharm Inc | Non-hygroscopic salts of 5-ht2c agonists |
ES2704455T3 (es) | 2010-09-01 | 2019-03-18 | Arena Pharm Inc | Formas farmacéuticas de liberación modificada de agonistas de 5-HT2C útiles para la gestión del peso |
NZ608266A (en) | 2010-09-01 | 2015-09-25 | Arena Pharm Inc | Administration of lorcaserin to individuals with renal impairment |
KR20130138770A (ko) | 2010-09-01 | 2013-12-19 | 아레나 파마슈티칼스, 인크. | 광학적으로 활성 산을 갖는 로르카세린의 염 |
US20150297610A1 (en) | 2012-10-09 | 2015-10-22 | Arena Pharmaceuticals, Inc. | Method of weight management |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS51149296A (en) * | 1975-06-09 | 1976-12-22 | Takeda Chem Ind Ltd | Cephems or penams and their preparation |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5168589A (ja) * | 1974-12-06 | 1976-06-14 | Shionogi Seiyaku Kk | |
DK154939C (da) | 1974-12-19 | 1989-06-12 | Takeda Chemical Industries Ltd | Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf |
DE2760123C2 (de) * | 1976-01-23 | 1986-04-30 | Roussel-Uclaf, Paris | 7-Aminothiazolyl-syn-oxyiminoacetamidocephalosporansäuren, ihre Herstellung und sie enthaltende pharmazeutische Zusammensetzungen |
-
1977
- 1977-12-24 DE DE19772758001 patent/DE2758001A1/de not_active Withdrawn
-
1978
- 1978-12-16 DE DE7878101738T patent/DE2861043D1/de not_active Expired
- 1978-12-16 EP EP78101738A patent/EP0002765B1/de not_active Expired
- 1978-12-19 ES ES476109A patent/ES476109A1/es not_active Expired
- 1978-12-20 EG EG721/78A patent/EG13762A/xx active
- 1978-12-20 US US05/971,558 patent/US4293550A/en not_active Expired - Lifetime
- 1978-12-21 FI FI783960A patent/FI66007C/fi not_active IP Right Cessation
- 1978-12-21 ZA ZA00787209A patent/ZA787209B/xx unknown
- 1978-12-21 IE IE2546/78A patent/IE48147B1/en unknown
- 1978-12-21 PT PT68964A patent/PT68964A/pt unknown
- 1978-12-21 NZ NZ189266A patent/NZ189266A/xx unknown
- 1978-12-22 AT AT0924178A patent/AT365599B/de not_active IP Right Cessation
- 1978-12-22 AU AU42848/78A patent/AU534258B2/en not_active Expired
- 1978-12-22 IL IL56284A patent/IL56284A/xx unknown
- 1978-12-22 DK DK578978A patent/DK578978A/da not_active Application Discontinuation
- 1978-12-22 HU HU78HO2127A patent/HU184140B/hu unknown
- 1978-12-22 CA CA318,496A patent/CA1109461A/en not_active Expired
- 1978-12-22 NO NO784366A patent/NO784366L/no unknown
- 1978-12-22 GR GR57978A patent/GR65234B/el unknown
- 1978-12-22 PH PH21988A patent/PH15925A/en unknown
- 1978-12-23 JP JP15817278A patent/JPS5495592A/ja active Granted
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS51149296A (en) * | 1975-06-09 | 1976-12-22 | Takeda Chem Ind Ltd | Cephems or penams and their preparation |
Cited By (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5547688A (en) * | 1978-09-08 | 1980-04-04 | Fujisawa Pharmaceut Co Ltd | Novel cephem compound and its preparation |
JPH0121154B2 (ja) * | 1978-09-08 | 1989-04-19 | Fujisawa Pharmaceutical Co | |
JPS5657790A (en) * | 1979-10-02 | 1981-05-20 | Glaxo Group Ltd | Cephalosporin antibiotic |
JPS56142289A (en) * | 1980-02-23 | 1981-11-06 | Hoechst Ag | Cephalosporin derivative and manufacture |
JPS57131794A (en) * | 1980-12-31 | 1982-08-14 | Fujisawa Pharmaceut Co Ltd | Novel cephem compound or salt thereof, preparation of the same and preventing agent and remedy for microbism containing the same as active constituent |
Also Published As
Publication number | Publication date |
---|---|
FI66007B (fi) | 1984-04-30 |
IL56284A (en) | 1983-03-31 |
DE2861043D1 (en) | 1981-11-26 |
ES476109A1 (es) | 1979-10-16 |
HU184140B (en) | 1984-07-30 |
DK578978A (da) | 1979-06-25 |
DE2758001A1 (de) | 1979-07-12 |
FI66007C (fi) | 1984-08-10 |
GR65234B (en) | 1980-07-30 |
NO784366L (no) | 1979-06-26 |
ZA787209B (en) | 1979-12-27 |
NZ189266A (en) | 1981-12-15 |
AT365599B (de) | 1982-01-25 |
ATA924178A (de) | 1981-06-15 |
EP0002765A1 (de) | 1979-07-11 |
IL56284A0 (en) | 1979-03-12 |
AU4284878A (en) | 1979-06-28 |
US4293550A (en) | 1981-10-06 |
JPH0132226B2 (ja) | 1989-06-29 |
CA1109461A (en) | 1981-09-22 |
IE48147B1 (en) | 1984-10-17 |
EP0002765B1 (de) | 1981-09-02 |
IE782546L (en) | 1979-06-24 |
PT68964A (de) | 1979-01-01 |
PH15925A (en) | 1983-04-26 |
AU534258B2 (en) | 1984-01-12 |
FI783960A (fi) | 1979-06-25 |
EG13762A (en) | 1982-09-30 |
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