JPH07625B2 - セファロスポリン中間体の製造方法 - Google Patents

セファロスポリン中間体の製造方法

Info

Publication number
JPH07625B2
JPH07625B2 JP60501797A JP50179785A JPH07625B2 JP H07625 B2 JPH07625 B2 JP H07625B2 JP 60501797 A JP60501797 A JP 60501797A JP 50179785 A JP50179785 A JP 50179785A JP H07625 B2 JPH07625 B2 JP H07625B2
Authority
JP
Japan
Prior art keywords
formula
amino
group
acid
thiazolyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP60501797A
Other languages
English (en)
Japanese (ja)
Other versions
JPS61501780A (ja
Inventor
アツシヤー、ゲルト
シユツルム、フベルト
ターラー、ハインリツヒ
フアイト、ベルネル
Original Assignee
ビオヘミ−・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ビオヘミ−・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング filed Critical ビオヘミ−・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング
Priority claimed from PCT/EP1985/000156 external-priority patent/WO1985004659A1/de
Publication of JPS61501780A publication Critical patent/JPS61501780A/ja
Publication of JPH07625B2 publication Critical patent/JPH07625B2/ja
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D277/70—Sulfur atoms
    • C07D277/74—Sulfur atoms substituted by carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP60501797A 1984-04-10 1985-04-04 セファロスポリン中間体の製造方法 Expired - Lifetime JPH07625B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
AT119784A AT381496B (de) 1984-04-10 1984-04-10 Verfahren zur herstellung von cephalosporinantibiotika
AT1197/84 1984-04-10
PCT/EP1985/000156 WO1985004659A1 (en) 1984-04-10 1985-04-04 Intermediary products of cephalosporine, preparation process thereof and utilization thereof

Related Child Applications (2)

Application Number Title Priority Date Filing Date
JP5144701A Division JPH0751575B2 (ja) 1984-04-10 1993-06-16 ２−アミノチアゾール化合物およびその製造法
JP6184491A Division JP2529093B2 (ja) 1984-04-10 1994-08-05 セファロスポリン中間体の製造方法

Publications (2)

Publication Number Publication Date
JPS61501780A JPS61501780A (ja) 1986-08-21
JPH07625B2 true JPH07625B2 (ja) 1995-01-11

Family

ID=3508702

Family Applications (2)

Application Number Title Priority Date Filing Date
JP60501797A Expired - Lifetime JPH07625B2 (ja) 1984-04-10 1985-04-04 セファロスポリン中間体の製造方法
JP5144701A Expired - Lifetime JPH0751575B2 (ja) 1984-04-10 1993-06-16 ２−アミノチアゾール化合物およびその製造法

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP5144701A Expired - Lifetime JPH0751575B2 (ja) 1984-04-10 1993-06-16 ２−アミノチアゾール化合物およびその製造法

Country Status (2)

Country Link
JP (2) JPH07625B2 (de)
AT (2) AT382149B (de)

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS53112895A (en) * 1977-03-12 1978-10-02 Hoechst Ag Cephem derivative and process for preparing same
JPS56152488A (en) * 1980-03-28 1981-11-26 Biochemie Gmbh Novel manufacture of cephalosporin type antibiotics and novel intermediate therefor and manufacture of intermediate
JPS5821682A (ja) * 1981-07-31 1983-02-08 Sankyo Co Ltd セファロスポリン誘導体
DE3433147A1 (de) * 1983-09-12 1985-03-28 Biochemie GmbH, Kundl, Tirol Neues verfahren zur herstellung von cephalosporinantibiotika

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU526540B2 (en) * 1976-04-12 1983-01-20 Fujisawa Pharmaceutical Co., Ltd. Oximes of substituted phenyl, thiazolyl - glyoxylic acids
PH17188A (en) * 1977-03-14 1984-06-14 Fujisawa Pharmaceutical Co New cephem and cepham compounds and their pharmaceutical compositions and method of use
SE439312B (sv) * 1977-03-25 1985-06-10 Roussel Uclaf Sett att framstella nya oximderivat av 3-acetoximetyl-7-aminotiazolylacetamido cefalosporansyra

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS53112895A (en) * 1977-03-12 1978-10-02 Hoechst Ag Cephem derivative and process for preparing same
JPS56152488A (en) * 1980-03-28 1981-11-26 Biochemie Gmbh Novel manufacture of cephalosporin type antibiotics and novel intermediate therefor and manufacture of intermediate
JPS5821682A (ja) * 1981-07-31 1983-02-08 Sankyo Co Ltd セファロスポリン誘導体
DE3433147A1 (de) * 1983-09-12 1985-03-28 Biochemie GmbH, Kundl, Tirol Neues verfahren zur herstellung von cephalosporinantibiotika

Also Published As

Publication number Publication date
AT382149B (de) 1987-01-12
JPH0625236A (ja) 1994-02-01
JPS61501780A (ja) 1986-08-21
JPH0751575B2 (ja) 1995-06-05
AT381496B (de) 1986-10-27
ATA108585A (de) 1986-06-15
ATA119784A (de) 1986-03-15

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