ITTO920606A1 - Derivati di decaidro-8h-isochino/2, 1-g/1, 6/naftiridina e decaidrobenzo /a/pirrolo/2, 3-e/chinolizina. - Google Patents

Derivati di decaidro-8h-isochino/2, 1-g/1, 6/naftiridina e decaidrobenzo /a/pirrolo/2, 3-e/chinolizina.

Info

Publication number
ITTO920606A1
ITTO920606A1 IT000606A ITTO920606A ITTO920606A1 IT TO920606 A1 ITTO920606 A1 IT TO920606A1 IT 000606 A IT000606 A IT 000606A IT TO920606 A ITTO920606 A IT TO920606A IT TO920606 A1 ITTO920606 A1 IT TO920606A1
Authority
IT
Italy
Prior art keywords
quinolizina
naftiridina
decaidrobenzo
decaidro
isochino
Prior art date
Application number
IT000606A
Other languages
English (en)
Inventor
Robin D Clark
Redfern William Salisbury
Michael Spedding
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of ITTO920606A0 publication Critical patent/ITTO920606A0/it
Publication of ITTO920606A1 publication Critical patent/ITTO920606A1/it
Application granted granted Critical
Publication of IT1256880B publication Critical patent/IT1256880B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
ITTO920606A 1991-07-17 1992-07-16 Derivati di decaidro-8h-isochino/2,1-g/1,6/naftiridina e decaidrobenzo/a/pirrolo/2,3-e/chinolizina IT1256880B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US73169191A 1991-07-17 1991-07-17

Publications (3)

Publication Number Publication Date
ITTO920606A0 ITTO920606A0 (it) 1992-07-16
ITTO920606A1 true ITTO920606A1 (it) 1994-01-16
IT1256880B IT1256880B (it) 1995-12-27

Family

ID=24940584

Family Applications (1)

Application Number Title Priority Date Filing Date
ITTO920606A IT1256880B (it) 1991-07-17 1992-07-16 Derivati di decaidro-8h-isochino/2,1-g/1,6/naftiridina e decaidrobenzo/a/pirrolo/2,3-e/chinolizina

Country Status (14)

Country Link
EP (1) EP0524004A1 (it)
JP (1) JPH0665242A (it)
KR (1) KR930002346A (it)
AU (1) AU655998B2 (it)
CA (1) CA2074038A1 (it)
FI (1) FI923267A (it)
HU (2) HUT61550A (it)
IE (1) IE922314A1 (it)
IL (1) IL102521A (it)
IT (1) IT1256880B (it)
NO (1) NO922812L (it)
NZ (1) NZ243586A (it)
TW (1) TW209219B (it)
ZA (1) ZA925324B (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ543863A (en) 2003-06-20 2009-05-31 Hoffmann La Roche Hexahydropyridoisoquinolines as DPP-IV inhibitors
CN103387583B (zh) * 2012-05-09 2018-04-13 中国科学院上海药物研究所 二芳基并[a,g]喹嗪类化合物、其制备方法、药物组合物及其应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4791108A (en) * 1987-04-13 1988-12-13 Syntex (U.S.A.) Inc. Sulfonyl-decahydro-8H-isoquino[2,1-G][1,6]-naphthyridines and related compounds useful as α2 -blockers

Also Published As

Publication number Publication date
HU9202333D0 (en) 1992-10-28
KR930002346A (ko) 1993-02-23
AU655998B2 (en) 1995-01-19
FI923267A (fi) 1993-01-18
ZA925324B (en) 1994-07-17
IT1256880B (it) 1995-12-27
AU2031392A (en) 1993-01-21
IE922314A1 (en) 1993-01-27
HU210711A9 (en) 1995-06-28
NO922812D0 (no) 1992-07-16
TW209219B (it) 1993-07-11
EP0524004A1 (en) 1993-01-20
CA2074038A1 (en) 1993-01-18
NZ243586A (en) 1995-03-28
HUT61550A (en) 1993-01-28
JPH0665242A (ja) 1994-03-08
NO922812L (no) 1993-01-18
ITTO920606A0 (it) 1992-07-16
FI923267A0 (fi) 1992-07-16
IL102521A (en) 1996-05-14

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Legal Events

Date Code Title Description
0001 Granted
TA Fee payment date (situation as of event date), data collected since 19931001

Effective date: 19950731