ITMI991740A0 - Derivati di 1h-pirido 3,4-b indol-1-one - Google Patents

Derivati di 1h-pirido 3,4-b indol-1-one

Info

Publication number
ITMI991740A0
ITMI991740A0 IT99MI001740A ITMI991740A ITMI991740A0 IT MI991740 A0 ITMI991740 A0 IT MI991740A0 IT 99MI001740 A IT99MI001740 A IT 99MI001740A IT MI991740 A ITMI991740 A IT MI991740A IT MI991740 A0 ITMI991740 A0 IT MI991740A0
Authority
IT
Italy
Prior art keywords
pyrido
indol
derivatives
Prior art date
Application number
IT99MI001740A
Other languages
English (en)
Inventor
Nicoletta Pescalli
Ernesto Menta
Silvano Spinelli
Original Assignee
Novuspharma Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novuspharma Spa filed Critical Novuspharma Spa
Priority to IT1999MI001740A priority Critical patent/IT1313592B1/it
Publication of ITMI991740A0 publication Critical patent/ITMI991740A0/it
Priority to PCT/EP2000/007279 priority patent/WO2001009129A2/en
Priority to AU68315/00A priority patent/AU6831500A/en
Publication of ITMI991740A1 publication Critical patent/ITMI991740A1/it
Application granted granted Critical
Publication of IT1313592B1 publication Critical patent/IT1313592B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
IT1999MI001740A 1999-08-03 1999-08-03 Derivati di 1h-pirido 3,4-b indol-1-one. IT1313592B1 (it)

Priority Applications (3)

Application Number Priority Date Filing Date Title
IT1999MI001740A IT1313592B1 (it) 1999-08-03 1999-08-03 Derivati di 1h-pirido 3,4-b indol-1-one.
PCT/EP2000/007279 WO2001009129A2 (en) 1999-08-03 2000-07-28 1h-pirido[3, 4-b]indol-1-one derivatives
AU68315/00A AU6831500A (en) 1999-08-03 2000-07-28 1h-pirido[3, 4-b]indol-1-one derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
IT1999MI001740A IT1313592B1 (it) 1999-08-03 1999-08-03 Derivati di 1h-pirido 3,4-b indol-1-one.

Publications (3)

Publication Number Publication Date
ITMI991740A0 true ITMI991740A0 (it) 1999-08-03
ITMI991740A1 ITMI991740A1 (it) 2001-02-03
IT1313592B1 IT1313592B1 (it) 2002-09-09

Family

ID=11383490

Family Applications (1)

Application Number Title Priority Date Filing Date
IT1999MI001740A IT1313592B1 (it) 1999-08-03 1999-08-03 Derivati di 1h-pirido 3,4-b indol-1-one.

Country Status (3)

Country Link
AU (1) AU6831500A (it)
IT (1) IT1313592B1 (it)
WO (1) WO2001009129A2 (it)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2823975B1 (fr) 2001-04-27 2003-05-30 Sanofi Synthelabo Nouvelle utilisation de pyridoindolone
FR2846329B1 (fr) * 2002-10-23 2004-12-03 Sanofi Synthelabo Derives de pyridoindolone substitues en -3 par un phenyle, leur preparation et leur application en therapeutique
US7456193B2 (en) 2002-10-23 2008-11-25 Sanofi-Aventis Pyridoindolone derivatives substituted in the 3-position by a heterocyclic group, their preparation and their application in therapeutics
FR2869316B1 (fr) 2004-04-21 2006-06-02 Sanofi Synthelabo Derives de pyridoindolone substitues en -6, leur preparation et leur application en therapeutique.
FR2892416B1 (fr) 2005-10-20 2008-06-27 Sanofi Aventis Sa Derives de 6-heteroarylpyridoindolone, leur preparation et leur application en therapeutique
CA3041868C (en) * 2008-10-09 2023-03-07 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Bis sulfonamide piperazinyl and piperidinyl activators of human pyruvatekinase
CN102127074A (zh) * 2010-12-17 2011-07-20 中国药科大学 6-氨磺酰基取代-β-咔啉-1-酮类细胞周期蛋白依赖性激酶2抑制剂及其用途
WO2012157744A1 (ja) * 2011-05-19 2012-11-22 国立大学法人 富山大学 1-チオキソ-1,2,3,4-テトラヒドロ-β-カルボリン誘導体およびそれらを含有する抗がん剤
FR3034095A1 (fr) * 2015-03-26 2016-09-30 Agronomique Inst Nat Rech Prevention et/ou traitement des parasitoses induites par des parasites appartenant au phylum des apicomplexes

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4897391A (en) * 1988-06-17 1990-01-30 Schering Corporation Tricyclic anti-allergy, antiinflammatory and anti-hyperproliferative compounds

Also Published As

Publication number Publication date
AU6831500A (en) 2001-02-19
ITMI991740A1 (it) 2001-02-03
WO2001009129A2 (en) 2001-02-08
IT1313592B1 (it) 2002-09-09
WO2001009129A3 (en) 2001-04-26

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