ITMI20062208A1 - PROCESS FOR THE PREPARATION OF IMATINIB AND ITS INTERMEDIATES - Google Patents
PROCESS FOR THE PREPARATION OF IMATINIB AND ITS INTERMEDIATESInfo
- Publication number
- ITMI20062208A1 ITMI20062208A1 ITMI20062208A ITMI20062208A1 IT MI20062208 A1 ITMI20062208 A1 IT MI20062208A1 IT MI20062208 A ITMI20062208 A IT MI20062208A IT MI20062208 A1 ITMI20062208 A1 IT MI20062208A1
- Authority
- IT
- Italy
- Prior art keywords
- imatinib
- intermediates
- preparation
- Prior art date
Links
Priority Applications (12)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ITMI20062208 ITMI20062208A1 (en) | 2006-11-16 | 2006-11-16 | PROCESS FOR THE PREPARATION OF IMATINIB AND ITS INTERMEDIATES |
US12/515,105 US8168787B2 (en) | 2006-11-16 | 2007-11-15 | Process for the preparation of imatinib and intermediates thereof |
CN2007800392449A CN101528700B (en) | 2006-11-16 | 2007-11-15 | Process for the preparation of imatinib and intermediates thereof |
ES07849757.5T ES2496592T3 (en) | 2006-11-16 | 2007-11-15 | Process for the preparation of Imatinib and intermediate compounds thereof |
JP2009536868A JP5265562B2 (en) | 2006-11-16 | 2007-11-15 | Process for the preparation of imatinib and its intermediates |
RU2009122692/04A RU2480461C2 (en) | 2006-11-16 | 2007-11-15 | Method of producing imatinib and intermediate compounds thereof |
EP07849757.5A EP2074095B1 (en) | 2006-11-16 | 2007-11-15 | Process for the preparation of imatinib and intermediates thereof |
KR1020097011914A KR101420892B1 (en) | 2006-11-16 | 2007-11-15 | Process for the preparation of Imatinib and intermediates thereof |
BRPI0718812-9A2A BRPI0718812A2 (en) | 2006-11-16 | 2007-11-15 | PROCESS FOR PREPARATION OF IMATINIB AND INTERMEDIARIES OF THIS |
PCT/IT2007/000804 WO2008059551A2 (en) | 2006-11-16 | 2007-11-15 | Process for the preparation of imatinib and intermediates thereof |
IL197954A IL197954A (en) | 2006-11-16 | 2009-04-05 | Process for the preparation of imatinib, intermediates thereof and process for preparing said intermediates |
US12/784,366 US8334381B2 (en) | 2006-11-16 | 2010-05-20 | Process for the preparation of intermediates useful in the synthesis of imatinib |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ITMI20062208 ITMI20062208A1 (en) | 2006-11-16 | 2006-11-16 | PROCESS FOR THE PREPARATION OF IMATINIB AND ITS INTERMEDIATES |
Publications (1)
Publication Number | Publication Date |
---|---|
ITMI20062208A1 true ITMI20062208A1 (en) | 2008-05-17 |
Family
ID=40277989
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ITMI20062208 ITMI20062208A1 (en) | 2006-11-16 | 2006-11-16 | PROCESS FOR THE PREPARATION OF IMATINIB AND ITS INTERMEDIATES |
Country Status (2)
Country | Link |
---|---|
CN (1) | CN101528700B (en) |
IT (1) | ITMI20062208A1 (en) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN102372690B (en) * | 2010-08-20 | 2014-05-28 | 成都地奥制药集团有限公司 | Intermediate for synthesizing imatinib and application of intermediate in imatinib synthesis |
CN103539639B (en) * | 2010-11-09 | 2015-05-20 | 常州制药厂有限公司 | Method for preparing key intermediate of medicament |
CN102001920B (en) * | 2010-11-09 | 2013-05-15 | 常州制药厂有限公司 | Preparation method of medicine intermediate |
CN102382100B (en) * | 2011-03-09 | 2014-04-16 | 上海昕盛医药科技有限公司 | Preparation method of imatinib |
CN102617475A (en) * | 2012-03-07 | 2012-08-01 | 南开大学 | Method for decarboxylation of N-methyl-3-alkyl-4 -nitropyrazole formate |
CN102796074B (en) * | 2012-06-21 | 2015-04-08 | 苏州立新制药有限公司 | Method for preparing imatinib mesylate intermediate |
CN103694145B (en) * | 2013-11-28 | 2016-02-10 | 山东鑫泉医药有限公司 | The synthetic method of (2-methyl-5-nitrophenyl) guanidine sulfate |
CN108148003B (en) * | 2018-01-16 | 2021-03-26 | 棓诺(苏州)新材料有限公司 | Method for synthesizing benzoylpyrimidine compound serving as intermediate of OLED (organic light emitting diode) material |
CN109682914A (en) * | 2019-01-16 | 2019-04-26 | 徐州立兴佳正医药科技有限公司 | A kind of method that LC-MS measures Imatinib concentration in blood plasma |
-
2006
- 2006-11-16 IT ITMI20062208 patent/ITMI20062208A1/en unknown
-
2007
- 2007-11-15 CN CN2007800392449A patent/CN101528700B/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
CN101528700A (en) | 2009-09-09 |
CN101528700B (en) | 2012-05-30 |
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