IT201900003839A1 - Sintesi di apalutamide amorfa stabile - Google Patents
Sintesi di apalutamide amorfa stabileInfo
- Publication number
- IT201900003839A1 IT201900003839A1 IT102019000003839A IT201900003839A IT201900003839A1 IT 201900003839 A1 IT201900003839 A1 IT 201900003839A1 IT 102019000003839 A IT102019000003839 A IT 102019000003839A IT 201900003839 A IT201900003839 A IT 201900003839A IT 201900003839 A1 IT201900003839 A1 IT 201900003839A1
- Authority
- IT
- Italy
- Prior art keywords
- apalutamide
- synthesis
- stable amorphous
- amorphous
- stable
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT102019000003839A IT201900003839A1 (it) | 2019-03-15 | 2019-03-15 | Sintesi di apalutamide amorfa stabile |
PCT/IB2020/052011 WO2020188399A1 (en) | 2019-03-15 | 2020-03-09 | Synthesis of stable amorphous apalutamide |
EP20714281.1A EP3938361A1 (en) | 2019-03-15 | 2020-03-09 | Synthesis of stable amorphous apalutamide |
US17/438,948 US20220153718A1 (en) | 2019-03-15 | 2020-03-09 | Synthesis of stable amorphous apalutamide |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT102019000003839A IT201900003839A1 (it) | 2019-03-15 | 2019-03-15 | Sintesi di apalutamide amorfa stabile |
Publications (1)
Publication Number | Publication Date |
---|---|
IT201900003839A1 true IT201900003839A1 (it) | 2020-09-15 |
Family
ID=67002159
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IT102019000003839A IT201900003839A1 (it) | 2019-03-15 | 2019-03-15 | Sintesi di apalutamide amorfa stabile |
Country Status (4)
Country | Link |
---|---|
US (1) | US20220153718A1 (it) |
EP (1) | EP3938361A1 (it) |
IT (1) | IT201900003839A1 (it) |
WO (1) | WO2020188399A1 (it) |
Citations (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8445507B2 (en) | 2006-03-27 | 2013-05-21 | The Regents Of The University Of California | Androgen receptor modulator for the treatment of prostate cancer and androgen receptor-associated diseases |
WO2013184681A1 (en) | 2012-06-07 | 2013-12-12 | Aragon Pharmaceuticals, Inc. | Crystalline forms of an androgen receptor modulator |
WO2016124149A1 (zh) | 2015-02-06 | 2016-08-11 | 苏州晶云药物科技有限公司 | 一种治疗***癌的抗雄激素类药物的新晶型及其制备方法 |
WO2018112001A1 (en) | 2016-12-13 | 2018-06-21 | Watson Laboratories Inc. | Solid state forms of apalutamide |
WO2019016747A1 (en) | 2017-07-20 | 2019-01-24 | Dr. Reddy's Laboratories Limited | AMORPHOUS SOLID DISPERSIONS OF APALUTAMIDE AND PROCESS FOR THEIR PREPARATION |
-
2019
- 2019-03-15 IT IT102019000003839A patent/IT201900003839A1/it unknown
-
2020
- 2020-03-09 US US17/438,948 patent/US20220153718A1/en active Pending
- 2020-03-09 WO PCT/IB2020/052011 patent/WO2020188399A1/en active Application Filing
- 2020-03-09 EP EP20714281.1A patent/EP3938361A1/en not_active Withdrawn
Patent Citations (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8445507B2 (en) | 2006-03-27 | 2013-05-21 | The Regents Of The University Of California | Androgen receptor modulator for the treatment of prostate cancer and androgen receptor-associated diseases |
WO2013184681A1 (en) | 2012-06-07 | 2013-12-12 | Aragon Pharmaceuticals, Inc. | Crystalline forms of an androgen receptor modulator |
WO2016124149A1 (zh) | 2015-02-06 | 2016-08-11 | 苏州晶云药物科技有限公司 | 一种治疗***癌的抗雄激素类药物的新晶型及其制备方法 |
WO2018112001A1 (en) | 2016-12-13 | 2018-06-21 | Watson Laboratories Inc. | Solid state forms of apalutamide |
WO2019016747A1 (en) | 2017-07-20 | 2019-01-24 | Dr. Reddy's Laboratories Limited | AMORPHOUS SOLID DISPERSIONS OF APALUTAMIDE AND PROCESS FOR THEIR PREPARATION |
Also Published As
Publication number | Publication date |
---|---|
WO2020188399A1 (en) | 2020-09-24 |
EP3938361A1 (en) | 2022-01-19 |
US20220153718A1 (en) | 2022-05-19 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
JP1712167S (ja) | サウンドバー | |
MA54542A (fr) | Compositions de sparsentan amorphe | |
IT201900003839A1 (it) | Sintesi di apalutamide amorfa stabile | |
DK3752507T3 (da) | Triazoloquinazolinon-syntese | |
DK4011201T3 (da) | Stald | |
JP1737418S (ja) | 腕時計 | |
JP1738407S (ja) | 腕時計 | |
JP1725134S (ja) | 腕時計 | |
JP1713400S (ja) | 腕時計 | |
JP1722034S (ja) | 腕時計 | |
JP1707650S (ja) | 腕時計 | |
JP1720149S (ja) | モジュール式コンパクト | |
JP1712579S (ja) | 下敷き | |
JP1718207S (ja) | ついたて | |
JP1717962S (ja) | ついたて | |
JP1717963S (ja) | ついたて | |
JP1710278S (ja) | 上履き | |
JP1718912S (ja) | まないた | |
JP1718202S (ja) | ついたて | |
ES1275522Y (es) | Columbario | |
JP1714341S (ja) | マドラー | |
CA204629S (fr) | Étuve | |
JP1709649S (ja) | ついたて | |
JP1709647S (ja) | ついたて | |
JP1709646S (ja) | ついたて |