IT1105064B - Alchil(inferiore)2-tri-alchil(inferiore)sililacetilen-n-carbossiglicinati e procedimento per il loro impiego per la preparazione di prodotti farmaceutici - Google Patents

Alchil(inferiore)2-tri-alchil(inferiore)sililacetilen-n-carbossiglicinati e procedimento per il loro impiego per la preparazione di prodotti farmaceutici

Info

Publication number
IT1105064B
IT1105064B IT50013/78A IT5001378A IT1105064B IT 1105064 B IT1105064 B IT 1105064B IT 50013/78 A IT50013/78 A IT 50013/78A IT 5001378 A IT5001378 A IT 5001378A IT 1105064 B IT1105064 B IT 1105064B
Authority
IT
Italy
Prior art keywords
alchil
sililacetylen
carboxylicinates
tri
procedure
Prior art date
Application number
IT50013/78A
Other languages
English (en)
Other versions
IT7850013A0 (it
Original Assignee
Merrell Toraude & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Toraude & Co filed Critical Merrell Toraude & Co
Publication of IT7850013A0 publication Critical patent/IT7850013A0/it
Application granted granted Critical
Publication of IT1105064B publication Critical patent/IT1105064B/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/0803Compounds with Si-C or Si-Si linkages
    • C07F7/081Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IT50013/78A 1977-07-01 1978-06-23 Alchil(inferiore)2-tri-alchil(inferiore)sililacetilen-n-carbossiglicinati e procedimento per il loro impiego per la preparazione di prodotti farmaceutici IT1105064B (it)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/812,065 US4088667A (en) 1977-07-01 1977-07-01 Lower alkyl 2-tri-(lower)alkylsilylacetylene-N-carbethoxyglycinates and process for using same

Publications (2)

Publication Number Publication Date
IT7850013A0 IT7850013A0 (it) 1978-06-23
IT1105064B true IT1105064B (it) 1985-10-28

Family

ID=25208385

Family Applications (1)

Application Number Title Priority Date Filing Date
IT50013/78A IT1105064B (it) 1977-07-01 1978-06-23 Alchil(inferiore)2-tri-alchil(inferiore)sililacetilen-n-carbossiglicinati e procedimento per il loro impiego per la preparazione di prodotti farmaceutici

Country Status (12)

Country Link
US (1) US4088667A (it)
JP (1) JPS5414927A (it)
AU (1) AU514961B2 (it)
BE (1) BE868587A (it)
CA (1) CA1104141A (it)
DE (1) DE2828579A1 (it)
ES (1) ES471267A1 (it)
FR (1) FR2396014A1 (it)
GB (1) GB2001087B (it)
IT (1) IT1105064B (it)
NL (1) NL7807088A (it)
ZA (1) ZA783357B (it)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4103089A (en) * 1977-07-01 1978-07-25 Merrell Toraude Et Compagnie α-Acetylene and α-vinyl derivatives of amino acids
US4088667A (en) * 1977-07-01 1978-05-09 Merrell Toraude Et Compagnie Lower alkyl 2-tri-(lower)alkylsilylacetylene-N-carbethoxyglycinates and process for using same
US4100349A (en) * 1977-07-01 1978-07-11 Brian Walter Metcalf α-Acetylenic derivatives of histamine and related compounds
US4323704A (en) * 1979-06-25 1982-04-06 Merrell Toraude Et Compagnie αAcetylene and α-vinyl derivatives of amino acids
NZ197394A (en) * 1980-06-16 1984-09-28 Merrell Dow Pharma Inhibition of protozoal growth in animals with certain-substituted-amines or amino acids

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3959356A (en) * 1975-03-18 1976-05-25 Richardson-Merrell Inc. Acetylene derivatives of amino acids
US3946060A (en) * 1975-03-18 1976-03-23 Richardson-Merrell Inc. Acetylene derivatives
US4088667A (en) * 1977-07-01 1978-05-09 Merrell Toraude Et Compagnie Lower alkyl 2-tri-(lower)alkylsilylacetylene-N-carbethoxyglycinates and process for using same

Also Published As

Publication number Publication date
ES471267A1 (es) 1979-10-01
BE868587A (fr) 1978-10-16
AU514961B2 (en) 1981-03-05
ZA783357B (en) 1979-06-27
NL7807088A (nl) 1979-01-03
JPS5414927A (en) 1979-02-03
FR2396014A1 (fr) 1979-01-26
AU3732278A (en) 1980-01-03
US4088667A (en) 1978-05-09
CA1104141A (en) 1981-06-30
DE2828579A1 (de) 1979-01-11
IT7850013A0 (it) 1978-06-23
GB2001087A (en) 1979-01-24
GB2001087B (en) 1982-01-13

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