IN2011CH01927A - - Google Patents
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- Publication number
- IN2011CH01927A IN2011CH01927A IN1927CH2011A IN2011CH01927A IN 2011CH01927 A IN2011CH01927 A IN 2011CH01927A IN 1927CH2011 A IN1927CH2011 A IN 1927CH2011A IN 2011CH01927 A IN2011CH01927 A IN 2011CH01927A
- Authority
- IN
- India
- Prior art keywords
- provides
- present
- novel process
- palladium content
- fosaprepitant dimeglumine
- Prior art date
Links
- KDLHZDBZIXYQEI-UHFFFAOYSA-N Palladium Chemical compound [Pd] KDLHZDBZIXYQEI-UHFFFAOYSA-N 0.000 abstract 2
- 229940044880 fosaprepitant dimeglumine Drugs 0.000 abstract 1
- VRQHBYGYXDWZDL-OOZCZQCLSA-N fosaprepitant dimeglumine Chemical compound CNC[C@H](O)[C@@H](O)[C@H](O)[C@H](O)CO.CNC[C@H](O)[C@@H](O)[C@H](O)[C@H](O)CO.O([C@@H]([C@@H]1C=2C=CC(F)=CC=2)O[C@H](C)C=2C=C(C=C(C=2)C(F)(F)F)C(F)(F)F)CCN1CC1=NN(P(O)(O)=O)C(=O)N1 VRQHBYGYXDWZDL-OOZCZQCLSA-N 0.000 abstract 1
- 229910052763 palladium Inorganic materials 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
- C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Catalysts (AREA)
Priority Applications (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP12793409.9A EP2714701B1 (en) | 2011-06-03 | 2012-05-21 | Process for fosaprepitant |
| ES12793409.9T ES2594828T3 (es) | 2011-06-03 | 2012-05-21 | Procedimiento para fosaprepitant |
| PCT/IN2012/000360 WO2012164576A2 (en) | 2011-06-03 | 2012-05-21 | Process for fosaprepitant |
| US14/123,290 US9540406B2 (en) | 2011-06-03 | 2012-05-21 | Process for fosaprepitant |
| IN1927CH2011 IN2011CH01927A (uk) | 2011-06-03 | 2012-05-21 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN1927CH2011 IN2011CH01927A (uk) | 2011-06-03 | 2012-05-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2011CH01927A true IN2011CH01927A (uk) | 2015-10-02 |
Family
ID=47260000
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN1927CH2011 IN2011CH01927A (uk) | 2011-06-03 | 2012-05-21 |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US9540406B2 (uk) |
| EP (1) | EP2714701B1 (uk) |
| ES (1) | ES2594828T3 (uk) |
| IN (1) | IN2011CH01927A (uk) |
| WO (1) | WO2012164576A2 (uk) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ITMI20130744A1 (it) * | 2013-05-08 | 2014-11-09 | Olon Spa | Procedimento per la preparazione di fosaprepitant dimeglumina |
| CN105254668B (zh) * | 2013-05-14 | 2017-10-10 | 北京百川汇德医药技术开发有限公司 | 一种福沙匹坦及其可药用盐的制备新方法 |
| CN104650141A (zh) * | 2013-11-22 | 2015-05-27 | 上海汇伦生命科技有限公司 | 一种福沙匹坦二甲葡胺的精制方法 |
| CN104650142B (zh) * | 2013-11-25 | 2018-06-22 | 山东新时代药业有限公司 | 一种福沙匹坦二甲葡胺的制备方法 |
| WO2015083033A1 (en) * | 2013-12-02 | 2015-06-11 | Piramal Enterprises Limited | An improved process for the preparation of fosaprepitant having improved purity |
| TWI659039B (zh) * | 2014-05-21 | 2019-05-11 | 台灣神隆股份有限公司 | 製備福沙吡坦二甲葡胺之方法 |
| CN105294547A (zh) * | 2014-07-30 | 2016-02-03 | 连云港宏创药业有限公司 | 吡仑帕奈粗品的除钯方法 |
| US9850267B2 (en) | 2015-06-03 | 2017-12-26 | Navinta, Llc | Crystalline fosaprepitant dicyclohexylamine salt and its preparation |
| US9913853B2 (en) * | 2015-11-03 | 2018-03-13 | Cipla Limited | Stabilized liquid fosaprepitant formulations |
| WO2017093899A1 (en) | 2015-12-01 | 2017-06-08 | Piramal Enterprises Limited | A process for preparation of fosaprepitant dimeglumine and an intermediate thereof |
| CN107176964B (zh) * | 2016-03-09 | 2019-09-20 | 杭州九源基因工程有限公司 | 一种福沙匹坦的精制除钯工艺 |
| CN106588989A (zh) * | 2016-11-08 | 2017-04-26 | 山东裕欣药业有限公司 | 一种福沙匹坦双葡甲胺化合物的新晶型及其制备方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8623844B2 (en) * | 2008-07-17 | 2014-01-07 | Navin Ganesh Bhatt | Fosaprepitant dimeglumine intermediate, neutral fosaprepitant, and amorphous fosaprepitant dimeglumine and processes for their preparations |
| AU2009294875C1 (en) | 2008-09-22 | 2015-05-14 | Aileron Therapeutics, Inc. | Methods for preparing purified polypeptide compositions |
| WO2011045817A2 (en) | 2009-10-15 | 2011-04-21 | Sandoz Private Limited | Process for the preparation of fosaprepitant, intermediate and pharmaceutical acceptable salt thereof |
-
2012
- 2012-05-21 US US14/123,290 patent/US9540406B2/en active Active
- 2012-05-21 IN IN1927CH2011 patent/IN2011CH01927A/en unknown
- 2012-05-21 EP EP12793409.9A patent/EP2714701B1/en active Active
- 2012-05-21 ES ES12793409.9T patent/ES2594828T3/es active Active
- 2012-05-21 WO PCT/IN2012/000360 patent/WO2012164576A2/en active Application Filing
Also Published As
| Publication number | Publication date |
|---|---|
| EP2714701B1 (en) | 2016-07-13 |
| EP2714701A2 (en) | 2014-04-09 |
| ES2594828T3 (es) | 2016-12-22 |
| US9540406B2 (en) | 2017-01-10 |
| WO2012164576A3 (en) | 2013-03-28 |
| EP2714701A4 (en) | 2014-12-24 |
| US20140107337A1 (en) | 2014-04-17 |
| WO2012164576A2 (en) | 2012-12-06 |
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