IL295626A - A triple drug combination that includes dabrafenib, an erk inhibitor and a raf inhibitor - Google Patents

A triple drug combination that includes dabrafenib, an erk inhibitor and a raf inhibitor

Info

Publication number: IL295626A
Authority: IL; Israel
Prior art keywords: braf; dabrafenib; compound; seq; pharmaceutic
Prior art date: 2020-02-28

Application number

IL295626A

Other languages

English (en)

Hebrew (he)

Original Assignee

Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2020-02-28

Filing date

2021-02-26

Publication date

2022-10-01

2021-02-26 Application filed by Novartis Ag filed Critical Novartis Ag

2022-10-01 Publication of IL295626A publication Critical patent/IL295626A/en

Links

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- A61K31/00—Medicinal preparations containing organic active ingredients
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

IL295626A 2020-02-28 2021-02-26 A triple drug combination that includes dabrafenib, an erk inhibitor and a raf inhibitor IL295626A (en)

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US202062983020P	2020-02-28	2020-02-28
PCT/IB2021/051641 WO2021171260A2 (fr)	2020-02-28	2021-02-26	Combinaison pharmaceutique triple comprenant dabrafenib, un inhibiteur d'erk et un inhibiteur de raf ou un inhibiteur de pd-1

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EP (1)	EP4110341A2 (fr)
JP (1)	JP2023516155A (fr)
KR (1)	KR20220148846A (fr)
CN (1)	CN115279374A (fr)
AU (1)	AU2021225491A1 (fr)
CA (1)	CA3173356A1 (fr)
IL (1)	IL295626A (fr)
TW (1)	TW202146024A (fr)
WO (1)	WO2021171260A2 (fr)

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2021
- 2021-02-26 WO PCT/IB2021/051641 patent/WO2021171260A2/fr unknown
- 2021-02-26 EP EP21739775.1A patent/EP4110341A2/fr active Pending
- 2021-02-26 AU AU2021225491A patent/AU2021225491A1/en active Pending
- 2021-02-26 KR KR1020227032733A patent/KR20220148846A/ko unknown
- 2021-02-26 CN CN202180017128.7A patent/CN115279374A/zh active Pending
- 2021-02-26 IL IL295626A patent/IL295626A/en unknown
- 2021-02-26 CA CA3173356A patent/CA3173356A1/fr active Pending
- 2021-02-26 TW TW110107183A patent/TW202146024A/zh unknown
- 2021-02-26 JP JP2022551299A patent/JP2023516155A/ja active Pending

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Publication number	Publication date
EP4110341A2 (fr)	2023-01-04
CN115279374A (zh)	2022-11-01
WO2021171260A2 (fr)	2021-09-02
CA3173356A1 (fr)	2021-09-02
JP2023516155A (ja)	2023-04-18
TW202146024A (zh)	2021-12-16
AU2021225491A1 (en)	2022-10-20
WO2021171260A3 (fr)	2021-10-07
KR20220148846A (ko)	2022-11-07

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