IL172592A0 - Pyrazolopyrimidines - Google Patents

Pyrazolopyrimidines

Info

Publication number
IL172592A0
IL172592A0 IL172592A IL17259205A IL172592A0 IL 172592 A0 IL172592 A0 IL 172592A0 IL 172592 A IL172592 A IL 172592A IL 17259205 A IL17259205 A IL 17259205A IL 172592 A0 IL172592 A0 IL 172592A0
Authority
IL
Israel
Prior art keywords
pyrazolopyrimidines
Prior art date
Application number
IL172592A
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10339360A external-priority patent/DE10339360A1/en
Priority claimed from DE2003157570 external-priority patent/DE10357570A1/en
Priority claimed from PCT/EP2004/006609 external-priority patent/WO2005000851A1/en
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of IL172592A0 publication Critical patent/IL172592A0/en

Links

IL172592A 2003-06-27 2005-12-15 Pyrazolopyrimidines IL172592A0 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE10328996 2003-06-27
DE10339360A DE10339360A1 (en) 2003-06-27 2003-08-27 New 7-amino-5-halo-pyrazolo-(1,5-a)-pyrimidine derivatives, useful as microbicides, especially fungicides or bactericides for protecting plants or materials such as wood
DE2003157570 DE10357570A1 (en) 2003-12-10 2003-12-10 New 7-amino-5-halo-pyrazolo-(1,5-a)-pyrimidine derivatives, useful as microbicides, especially fungicides or bactericides for protecting plants or materials such as wood
PCT/EP2004/006609 WO2005000851A1 (en) 2003-06-27 2004-06-18 Pyrazolopyrimidines

Publications (1)

Publication Number Publication Date
IL172592A0 true IL172592A0 (en) 2006-04-10

Family

ID=40506494

Family Applications (1)

Application Number Title Priority Date Filing Date
IL172592A IL172592A0 (en) 2003-06-27 2005-12-15 Pyrazolopyrimidines

Country Status (3)

Country Link
EA (1) EA009517B1 (en)
EC (1) ECSP056252A (en)
IL (1) IL172592A0 (en)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2738026C (en) 2008-09-22 2017-01-24 Array Biopharma Inc. Substituted imidazo[1,2b]pyridazine compounds as trk kinase inhibitors
DK3106463T6 (en) 2008-10-22 2020-02-24 Array Biopharma Inc PYRAZOLO [1,5-] PYRIMIDINE COMPOUND AS TRK-KINase INHIBITORS
AR077468A1 (en) 2009-07-09 2011-08-31 Array Biopharma Inc PIRAZOLO COMPOUNDS (1,5-A) PYRIMIDINE SUBSTITUTED AS TRK-QUINASA INHIBITORS
CN106977462B (en) * 2011-08-17 2020-04-28 阿达玛马克西姆股份有限公司 5-fluoro-4-imino-3- (substituted) -3, 4-dihydropyrimidin-2 (1H) one derivatives
CA2851142A1 (en) * 2011-10-06 2013-04-11 Bayer Intellectual Property Gmbh Heterocyclylpyri (mi) dinylpyrazole as fungicidals
KR20140072177A (en) * 2011-10-06 2014-06-12 바이엘 인텔렉쳐 프로퍼티 게엠베하 Heterocyclylpyri(mi)dinylpyrazole
CN110003118A (en) * 2012-12-28 2019-07-12 阿达玛马克西姆股份有限公司 The method for preparing carboxylic ester derivative
PL2953463T3 (en) * 2012-12-31 2022-01-03 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
DK3699181T3 (en) 2014-11-16 2023-03-20 Array Biopharma Inc CRYSTALLINE FORM OF (S)-N-(5-((R)-2-(2,5-DIFLUORPHENYL)-PYRROLIDIN-1-YL)-PYRAZOLO[1,5-A]PYRIMIDIN-3-YL)-3 -HYDROXYPYRROLIDINE-1-CARBOXAMIDE HYDROGEN SULFATE
TN2018000138A1 (en) 2015-10-26 2019-10-04 Array Biopharma Inc Point mutations in trk inhibitor-resistant cancer and methods relating to the same
US10045991B2 (en) 2016-04-04 2018-08-14 Loxo Oncology, Inc. Methods of treating pediatric cancers
PE20181888A1 (en) 2016-04-04 2018-12-11 Loxo Oncology Inc LIQUID FORMULATIONS OF (S) -N- (5 - ((R) -2- (2,5-DIFLUOROPHENYL) -PYRROLIDIN-1-IL) -PYRAZOLE [1,5-A] PYRIMIDIN-3-IL) -3 -HYDROXYPYRROLIDINE-1-CARBOXAMIDE
US10604525B2 (en) * 2016-04-15 2020-03-31 Bayal Animal Health Gmbh Pyrazolopyrimidine derivatives
EP3800189B1 (en) 2016-05-18 2023-06-28 Loxo Oncology, Inc. Preparation of (s)-n-(5-((r)-2-(2,5-difluorophenyl)pyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidin-3-yl)-3-hydroxypyrrolidine-1-carboxamide
JOP20190092A1 (en) 2016-10-26 2019-04-25 Array Biopharma Inc PROCESS FOR THE PREPARATION OF PYRAZOLO[1,5-a]PYRIMIDINES AND SALTS THEREOF
JOP20190213A1 (en) 2017-03-16 2019-09-16 Array Biopharma Inc Macrocyclic compounds as ros1 kinase inhibitors

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4908056A (en) * 1986-04-25 1990-03-13 E. I. Du Pont De Nemours And Company Heterocyclic acyl sulfonamides

Also Published As

Publication number Publication date
ECSP056252A (en) 2006-04-19
EA200600021A1 (en) 2006-06-30
EA009517B1 (en) 2008-02-28

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