ID29065A - Penghambat-penghambat farnesil protein transferase - Google Patents
Penghambat-penghambat farnesil protein transferaseInfo
- Publication number
- ID29065A ID29065A IDW00200101310A ID20011310A ID29065A ID 29065 A ID29065 A ID 29065A ID W00200101310 A IDW00200101310 A ID W00200101310A ID 20011310 A ID20011310 A ID 20011310A ID 29065 A ID29065 A ID 29065A
- Authority
- ID
- Indonesia
- Prior art keywords
- transferage
- farnesil
- obstacles
- protein
- transferage protein
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US21656098A | 1998-12-18 | 1998-12-18 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ID29065A true ID29065A (id) | 2001-07-26 |
Family
ID=22807539
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IDW00200101310A ID29065A (id) | 1998-12-18 | 1999-12-16 | Penghambat-penghambat farnesil protein transferase |
Country Status (24)
| Country | Link |
|---|---|
| EP (1) | EP1140904B1 (hu) |
| JP (1) | JP2002533335A (hu) |
| KR (1) | KR20010081115A (hu) |
| CN (1) | CN1285588C (hu) |
| AR (1) | AR021716A1 (hu) |
| AT (1) | ATE293622T1 (hu) |
| AU (1) | AU2347900A (hu) |
| BR (1) | BR9916328A (hu) |
| CA (1) | CA2354774C (hu) |
| CO (1) | CO5160344A1 (hu) |
| CZ (1) | CZ20011900A3 (hu) |
| DE (1) | DE69924876T2 (hu) |
| ES (1) | ES2237963T3 (hu) |
| HK (1) | HK1036279A1 (hu) |
| HU (1) | HUP0203054A3 (hu) |
| ID (1) | ID29065A (hu) |
| IL (1) | IL143409A0 (hu) |
| NO (1) | NO20012960L (hu) |
| PE (1) | PE20001516A1 (hu) |
| PL (1) | PL348294A1 (hu) |
| SK (1) | SK7582001A3 (hu) |
| TR (1) | TR200101754T2 (hu) |
| WO (1) | WO2000037458A1 (hu) |
| ZA (1) | ZA200104236B (hu) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7361663B2 (en) | 1999-11-10 | 2008-04-22 | Aventis Pharmaceuticals Inc. | N-acylpyrrolidin-2-ylalkylbenzamidine derivatives as inhibitors of factor Xa |
| IL149544A0 (en) * | 1999-11-10 | 2002-11-10 | Aventis Pharma Gmbh | N-ACYLPYRROLIDIN-2-YLALKYLBENZAMIDINE DERIVATIVES AS INHIBITORS OF FACTOR Xa |
| US6589978B2 (en) | 2000-06-30 | 2003-07-08 | Hoffman-La Roche Inc. | 1-sulfonyl pyrrolidine derivatives |
| AR033680A1 (es) * | 2000-08-30 | 2004-01-07 | Schering Corp | Compuestos triciclicos utiles como inhibidores de la farnesil proteino transferasa y su uso para la manufactura de medicamentos como agentes antitumorales |
| US7342016B2 (en) | 2000-08-30 | 2008-03-11 | Schering Corporation | Farnesyl protein transferase inhibitors as antitumor agents |
| US6809093B2 (en) | 2000-10-17 | 2004-10-26 | H. Lee Moffitt Cancer & Research Institute, Inc. | 2-substituted heterocyclic compounds |
| AU2002236813A1 (en) | 2001-01-22 | 2002-07-30 | Schering Corporation | Treatment of malaria with farnesyl protein transferase inhibitors |
| ATE313534T1 (de) | 2001-02-16 | 2006-01-15 | Aventis Pharma Inc | Heterocyclische substituierte carbonyl derivate und ihre verwendung als dopamin d3 rezeptor liganden |
| WO2002080895A2 (en) * | 2001-04-06 | 2002-10-17 | Schering Corporation | Treatment of malaria with farsenyl protein transferase inhibitors |
| FR2825705B1 (fr) * | 2001-06-08 | 2005-05-20 | Aventis Pharma Sa | Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens |
| GB0115862D0 (en) * | 2001-06-28 | 2001-08-22 | Smithkline Beecham Plc | Compounds |
| US6740757B2 (en) * | 2001-08-29 | 2004-05-25 | Pfizer Inc | Enantiomers of 6-[(4-chloro-phenyl)-hydroxy-(3-methyl-3h-imidazol-4-yl)-methyl]-4-[3-(3-hydroxy-3-methyl-but-1-ynyl)-phenyl]-1-methyl-1h-quinolin-2-one and salts thereof, useful in the treatment of cancer |
| FR2835186B1 (fr) | 2002-01-28 | 2006-10-20 | Aventis Pharma Sa | Nouveaux composes heterocycliques, actifs comme inhibiteurs de beta-lactamases |
| FR2844273B1 (fr) | 2002-09-05 | 2008-04-04 | Aventis Pharma Sa | Nouveaux composes heterocycliques, procede et intermediaires de preparation et utilisation comme medicament, notamment comme inhibiteurs de beta-lactamases et anti-bacteriens. |
| CA2509758A1 (en) * | 2002-12-17 | 2004-07-22 | Schering Corporation | 17 beta-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases |
| JP2008523104A (ja) * | 2004-12-13 | 2008-07-03 | シェーリング コーポレイション | 癌を治療するための新規なファルネシルタンパク質トランスフェラーゼ阻害剤およびその使用 |
| CA2591123A1 (en) * | 2004-12-14 | 2006-06-22 | Schering Corporation | Farnesyl protein transferase inhibitors and methods for treating proliferative diseases |
| WO2007084498A1 (en) * | 2006-01-19 | 2007-07-26 | Schering Corporation | Piperazine derivatives as farnesyl protein transferase inhibitors |
| AU2009249306B8 (en) * | 2008-05-22 | 2013-07-25 | Merck Canada Inc. | Process for the preparation of an orexin receptor antagonist |
| HU231150B1 (hu) | 2017-03-13 | 2021-03-29 | Richter Gedeon Nyrt | Eljárás racém 3-alkilpiperidin-3-karbonsav-etil-észterek optikai izomerjeinek elválasztására |
| TW202220992A (zh) | 2020-08-05 | 2022-06-01 | 匈牙利商羅特格登公司 | 具藥理活性之經雜環取代的吡唑并〔１，５－ａ〕嘧啶衍生物 |
| CN114349711B (zh) * | 2022-02-28 | 2023-08-15 | 四川依维欣医药科技有限公司 | 一种（R）-1-Boc-3-羟甲基哌嗪的合成方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL111235A (en) * | 1993-10-15 | 2001-03-19 | Schering Plough Corp | Medicinal preparations for inhibiting protein G activity and for the treatment of malignant diseases, containing tricyclic compounds, some such new compounds and a process for the preparation of some of them |
| GB9420172D0 (en) * | 1994-10-06 | 1994-11-23 | Boots Co Plc | Therapeutic agents |
| IL117798A (en) * | 1995-04-07 | 2001-11-25 | Schering Plough Corp | Tricyclic compounds useful for inhibiting the function of protein - G and for the treatment of malignant diseases, and pharmaceutical preparations containing them |
| ATE273299T1 (de) * | 1997-06-17 | 2004-08-15 | Schering Corp | Benzpyrido cycloheptan derivate mit farnesyl protein transferase inhibierender wirkung |
-
1999
- 1999-12-16 BR BR9916328-4A patent/BR9916328A/pt not_active IP Right Cessation
- 1999-12-16 ES ES99967139T patent/ES2237963T3/es not_active Expired - Lifetime
- 1999-12-16 SK SK758-2001A patent/SK7582001A3/sk unknown
- 1999-12-16 KR KR1020017007535A patent/KR20010081115A/ko not_active Application Discontinuation
- 1999-12-16 AR ARP990106459A patent/AR021716A1/es unknown
- 1999-12-16 WO PCT/US1999/027938 patent/WO2000037458A1/en active IP Right Grant
- 1999-12-16 DE DE69924876T patent/DE69924876T2/de not_active Expired - Fee Related
- 1999-12-16 CA CA002354774A patent/CA2354774C/en not_active Expired - Fee Related
- 1999-12-16 CO CO99078838A patent/CO5160344A1/es unknown
- 1999-12-16 JP JP2000589530A patent/JP2002533335A/ja active Pending
- 1999-12-16 AT AT99967139T patent/ATE293622T1/de not_active IP Right Cessation
- 1999-12-16 ID IDW00200101310A patent/ID29065A/id unknown
- 1999-12-16 AU AU23479/00A patent/AU2347900A/en not_active Abandoned
- 1999-12-16 CN CNB998162078A patent/CN1285588C/zh not_active Expired - Fee Related
- 1999-12-16 TR TR2001/01754T patent/TR200101754T2/xx unknown
- 1999-12-16 PL PL99348294A patent/PL348294A1/xx not_active Application Discontinuation
- 1999-12-16 CZ CZ20011900A patent/CZ20011900A3/cs unknown
- 1999-12-16 HU HU0203054A patent/HUP0203054A3/hu unknown
- 1999-12-16 IL IL14340999A patent/IL143409A0/xx unknown
- 1999-12-16 EP EP99967139A patent/EP1140904B1/en not_active Expired - Lifetime
- 1999-12-17 PE PE1999001293A patent/PE20001516A1/es not_active Application Discontinuation
-
2001
- 2001-05-23 ZA ZA200104236A patent/ZA200104236B/en unknown
- 2001-06-15 NO NO20012960A patent/NO20012960L/no not_active Application Discontinuation
- 2001-10-11 HK HK01107119A patent/HK1036279A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| HUP0203054A3 (en) | 2004-01-28 |
| CZ20011900A3 (cs) | 2002-02-13 |
| SK7582001A3 (en) | 2002-03-05 |
| AU2347900A (en) | 2000-07-12 |
| ES2237963T3 (es) | 2005-08-01 |
| NO20012960D0 (no) | 2001-06-15 |
| DE69924876D1 (de) | 2005-05-25 |
| EP1140904A1 (en) | 2001-10-10 |
| PE20001516A1 (es) | 2001-01-06 |
| NO20012960L (no) | 2001-08-15 |
| CN1352642A (zh) | 2002-06-05 |
| KR20010081115A (ko) | 2001-08-27 |
| IL143409A0 (en) | 2002-04-21 |
| BR9916328A (pt) | 2001-10-02 |
| AR021716A1 (es) | 2002-07-31 |
| ATE293622T1 (de) | 2005-05-15 |
| PL348294A1 (en) | 2002-05-20 |
| CA2354774C (en) | 2009-05-26 |
| ZA200104236B (en) | 2002-08-23 |
| EP1140904B1 (en) | 2005-04-20 |
| TR200101754T2 (tr) | 2002-05-21 |
| CN1285588C (zh) | 2006-11-22 |
| DE69924876T2 (de) | 2006-03-02 |
| JP2002533335A (ja) | 2002-10-08 |
| HUP0203054A2 (hu) | 2003-01-28 |
| CO5160344A1 (es) | 2002-05-30 |
| HK1036279A1 (en) | 2001-12-28 |
| WO2000037458A1 (en) | 2000-06-29 |
| CA2354774A1 (en) | 2000-06-29 |
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