HUP9903492A2 - Quinoline derivatives as type iv phosphodiesterase inhibitors, process for their preparation, pharmaceutical compositions containing the same and their use - Google Patents
Quinoline derivatives as type iv phosphodiesterase inhibitors, process for their preparation, pharmaceutical compositions containing the same and their useInfo
- Publication number
- HUP9903492A2 HUP9903492A2 HU9903492A HUP9903492A HUP9903492A2 HU P9903492 A2 HUP9903492 A2 HU P9903492A2 HU 9903492 A HU9903492 A HU 9903492A HU P9903492 A HUP9903492 A HU P9903492A HU P9903492 A2 HUP9903492 A2 HU P9903492A2
- Authority
- HU
- Hungary
- Prior art keywords
- preparation
- pharmaceutical compositions
- type
- same
- compositions containing
- Prior art date
Links
- 229940027991 antiseptic and disinfectant quinoline derivative Drugs 0.000 title 1
- 229940082638 cardiac stimulant phosphodiesterase inhibitors Drugs 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 239000002571 phosphodiesterase inhibitor Substances 0.000 title 1
- 125000002943 quinolinyl group Chemical class N1=C(C=CC2=CC=CC=C12)* 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Immunology (AREA)
- Rheumatology (AREA)
- Hospice & Palliative Care (AREA)
- Psychology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9523267.4A GB9523267D0 (en) | 1995-11-14 | 1995-11-14 | Organic compounds |
Publications (2)
Publication Number | Publication Date |
---|---|
HUP9903492A2 true HUP9903492A2 (en) | 2000-07-28 |
HUP9903492A3 HUP9903492A3 (en) | 2000-08-28 |
Family
ID=10783856
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU9903492A HUP9903492A3 (en) | 1995-11-14 | 1996-11-13 | Quinoline derivatives as type iv phosphodiesterase inhibitors, process for their preparation, pharmaceutical compositions containing the same and their use |
Country Status (17)
Country | Link |
---|---|
EP (1) | EP0873338A1 (en) |
JP (1) | JPH11515000A (en) |
KR (1) | KR19990067574A (en) |
CN (1) | CN1202170A (en) |
AU (1) | AU7570996A (en) |
BR (1) | BR9611504A (en) |
CA (1) | CA2235126A1 (en) |
CO (1) | CO4770973A1 (en) |
CZ (1) | CZ149498A3 (en) |
GB (1) | GB9523267D0 (en) |
HU (1) | HUP9903492A3 (en) |
MX (1) | MX9803839A (en) |
PE (1) | PE17598A1 (en) |
PL (1) | PL326636A1 (en) |
SK (1) | SK63998A3 (en) |
TR (1) | TR199800851T2 (en) |
WO (1) | WO1997018208A1 (en) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MXPA02001830A (en) | 1999-08-21 | 2002-08-12 | Byk Gulden Lomberg Chem Fab | Synergistic combination of pde inhibitors and beta 2 adrenoceptor agonist. |
CA2447619A1 (en) | 2001-05-23 | 2002-11-28 | Tanabe Seiyaku Co., Ltd. | A composition for accelerating bone fracture healing |
MXPA03010672A (en) | 2001-05-23 | 2004-03-02 | Tanabe Seiyaku Co | Therapeutic compositions for repairing chondropathy. |
TW200536851A (en) * | 2004-01-23 | 2005-11-16 | Amgen Inc | Compounds and methods of use |
JP2006347936A (en) | 2005-06-15 | 2006-12-28 | Bayer Cropscience Ag | Insecticidal benzanilides |
US8367829B2 (en) | 2010-05-10 | 2013-02-05 | Gilead Sciences, Inc. | Bi-functional pyrazolopyridine compounds |
UY33372A (en) | 2010-05-10 | 2011-12-30 | Gilead Sciences Inc | ? QUINOLINA BI? FUNCTIONAL ANALOGS, ITS USE IN THE MANUFACTURE OF MEDICINES, COMPOSITIONS THAT UNDERSTAND AND PREPARATION PROCESSES ?. |
BR112015008515A2 (en) | 2012-10-16 | 2017-07-04 | Janssen Pharmaceutica Nv | heteroaryl-linked quinolinyl ror t modulators |
EP2909192B1 (en) | 2012-10-16 | 2017-05-17 | Janssen Pharmaceutica NV | Methylene linked quinolinyl modulators of ror-gamma-t |
SG11201502935VA (en) | 2012-10-16 | 2015-09-29 | Janssen Pharmaceutica Nv | Phenyl linked quinolinyl modulators of ror-gamma-t |
CN105848483A (en) | 2013-10-15 | 2016-08-10 | 詹森药业有限公司 | Quinolinyl modulators of roryt |
US9221804B2 (en) | 2013-10-15 | 2015-12-29 | Janssen Pharmaceutica Nv | Secondary alcohol quinolinyl modulators of RORγt |
US10555941B2 (en) | 2013-10-15 | 2020-02-11 | Janssen Pharmaceutica Nv | Alkyl linked quinolinyl modulators of RORγt |
ES2770727T3 (en) | 2013-10-15 | 2020-07-02 | Janssen Pharmaceutica Nv | Alkyl-Linked Quinylonyl Modulators of ROR (gamma) t |
US9403816B2 (en) | 2013-10-15 | 2016-08-02 | Janssen Pharmaceutica Nv | Phenyl linked quinolinyl modulators of RORγt |
US9284308B2 (en) | 2013-10-15 | 2016-03-15 | Janssen Pharmaceutica Nv | Methylene linked quinolinyl modulators of RORγt |
US9328095B2 (en) | 2013-10-15 | 2016-05-03 | Janssen Pharmaceutica Nv | Heteroaryl linked quinolinyl modulators of RORgammat |
WO2020005830A1 (en) * | 2018-06-24 | 2020-01-02 | Adama Agan Ltd. | Process for the preparation of quinmerac |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9027055D0 (en) * | 1990-12-13 | 1991-02-06 | Sandoz Ltd | Organic compounds |
US5455252A (en) * | 1993-03-31 | 1995-10-03 | Syntex (U.S.A.) Inc. | Optionally substituted 6,8-quinolines |
-
1995
- 1995-11-14 GB GBGB9523267.4A patent/GB9523267D0/en active Pending
-
1996
- 1996-11-12 PE PE1996000810A patent/PE17598A1/en not_active Application Discontinuation
- 1996-11-13 PL PL96326636A patent/PL326636A1/en unknown
- 1996-11-13 SK SK639-98A patent/SK63998A3/en unknown
- 1996-11-13 EP EP96938196A patent/EP0873338A1/en not_active Withdrawn
- 1996-11-13 WO PCT/EP1996/004978 patent/WO1997018208A1/en not_active Application Discontinuation
- 1996-11-13 HU HU9903492A patent/HUP9903492A3/en unknown
- 1996-11-13 CZ CZ981494A patent/CZ149498A3/en unknown
- 1996-11-13 CO CO96059775A patent/CO4770973A1/en unknown
- 1996-11-13 AU AU75709/96A patent/AU7570996A/en not_active Abandoned
- 1996-11-13 KR KR1019980703597A patent/KR19990067574A/en not_active Application Discontinuation
- 1996-11-13 BR BR9611504A patent/BR9611504A/en not_active Application Discontinuation
- 1996-11-13 CA CA002235126A patent/CA2235126A1/en not_active Abandoned
- 1996-11-13 JP JP9515313A patent/JPH11515000A/en not_active Withdrawn
- 1996-11-13 TR TR1998/00851T patent/TR199800851T2/en unknown
- 1996-11-13 CN CN96198305A patent/CN1202170A/en active Pending
-
1998
- 1998-05-14 MX MX9803839A patent/MX9803839A/en unknown
Also Published As
Publication number | Publication date |
---|---|
MX9803839A (en) | 1998-09-30 |
SK63998A3 (en) | 1998-10-07 |
EP0873338A1 (en) | 1998-10-28 |
CZ149498A3 (en) | 1998-08-12 |
WO1997018208A1 (en) | 1997-05-22 |
PL326636A1 (en) | 1998-10-12 |
HUP9903492A3 (en) | 2000-08-28 |
CO4770973A1 (en) | 1999-04-30 |
CA2235126A1 (en) | 1997-05-22 |
BR9611504A (en) | 1999-03-02 |
PE17598A1 (en) | 1998-04-06 |
CN1202170A (en) | 1998-12-16 |
TR199800851T2 (en) | 1998-08-21 |
AU7570996A (en) | 1997-06-05 |
KR19990067574A (en) | 1999-08-25 |
JPH11515000A (en) | 1999-12-21 |
GB9523267D0 (en) | 1996-01-17 |
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