HUP9902404A2 - 5-(2-(4-(1,2-Benzizotiazol-3-il)-1-piperazinil)-etil)-6-klór-1,3-dihidro-2-(2H)-indol-2-on (ziprazidon) mezilát-dihidrát sói, a vegyületek előállitása és dopamin D2 antagonistaként történő alkalmazása - Google Patents

5-(2-(4-(1,2-Benzizotiazol-3-il)-1-piperazinil)-etil)-6-klór-1,3-dihidro-2-(2H)-indol-2-on (ziprazidon) mezilát-dihidrát sói, a vegyületek előállitása és dopamin D2 antagonistaként történő alkalmazása

Info

Publication number
HUP9902404A2
HUP9902404A2 HU9902404A HUP9902404A HUP9902404A2 HU P9902404 A2 HUP9902404 A2 HU P9902404A2 HU 9902404 A HU9902404 A HU 9902404A HU P9902404 A HUP9902404 A HU P9902404A HU P9902404 A2 HUP9902404 A2 HU P9902404A2
Authority
HU
Hungary
Prior art keywords
benzisothiazol
indol
piperazinyl
dihydro
ethyl
Prior art date
Application number
HU9902404A
Other languages
English (en)
Inventor
Frank Robert Busch
Carol Anne Rose
Russell James Shine
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Priority to HU9902404A priority Critical patent/HUP9902404A3/hu
Publication of HUP9902404A2 publication Critical patent/HUP9902404A2/hu
Publication of HUP9902404A3 publication Critical patent/HUP9902404A3/hu

Links

Abstract

A találmány tárgya 5-(2-(4-(1,2-benzizőtiazől-3-il)-1-piperazinil)-etil)-6-klór-1,3-dihidrő-2H-indől-2-őn-mezilátdihidrát sói, a mezilát-dihidrát sókat tartalmazó gyógyászati készítmények és eljárás avegyületek alkalmazására pszichőtikűs rendellenességek kezelésénél. ŕ
HU9902404A 1997-04-10 1997-04-10 Mesylate dihydrate salts of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)-ethyl)-6-choloro-1,3-dihydro-2(2h)-indol-2-one (-ziprasidone), its preparation and its use as dopamine d2 antagonist HUP9902404A3 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
HU9902404A HUP9902404A3 (en) 1997-04-10 1997-04-10 Mesylate dihydrate salts of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)-ethyl)-6-choloro-1,3-dihydro-2(2h)-indol-2-one (-ziprasidone), its preparation and its use as dopamine d2 antagonist

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU9902404A HUP9902404A3 (en) 1997-04-10 1997-04-10 Mesylate dihydrate salts of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)-ethyl)-6-choloro-1,3-dihydro-2(2h)-indol-2-one (-ziprasidone), its preparation and its use as dopamine d2 antagonist

Publications (2)

Publication Number Publication Date
HUP9902404A2 true HUP9902404A2 (hu) 2000-02-28
HUP9902404A3 HUP9902404A3 (en) 2000-03-28

Family

ID=89998782

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9902404A HUP9902404A3 (en) 1997-04-10 1997-04-10 Mesylate dihydrate salts of 5-(2-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)-ethyl)-6-choloro-1,3-dihydro-2(2h)-indol-2-one (-ziprasidone), its preparation and its use as dopamine d2 antagonist

Country Status (1)

Country Link
HU (1) HUP9902404A3 (hu)

Also Published As

Publication number Publication date
HUP9902404A3 (en) 2000-03-28

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Legal Events

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FD9A Lapse of provisional protection due to non-payment of fees