HUP0102662A2 - Imidazoylalkyl substituted with a five, six or seven membered heterocyclic ring containing one nitrogen atom - Google Patents

Imidazoylalkyl substituted with a five, six or seven membered heterocyclic ring containing one nitrogen atom

Info

Publication number: HUP0102662A2
Authority: HU; Hungary
Prior art keywords: nitrogen atom; heterocyclic ring; membered heterocyclic; ring containing; imidazoylalkyl
Prior art date: 1997-11-07

Application number

HU0102662A

Other languages

Hungarian (hu)

Inventor

Robert G. Aslanian

John J. Piwinski

Stuart B. Rosenblum

Daniel M. Solomon

Wayne D. Vaccaro

Ronald L. Wolin

Original Assignee

Schering Corp.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-11-07

Filing date

1998-11-05

Publication date

2001-12-28

1998-11-05 Application filed by Schering Corp. filed Critical Schering Corp.

2001-12-28 Publication of HUP0102662A2 publication Critical patent/HUP0102662A2/en

2003-01-28 Publication of HUP0102662A3 publication Critical patent/HUP0102662A3/en

Links

125000000623 heterocyclic group Chemical group 0.000 title 1
229910052757 nitrogen Inorganic materials 0.000 title 1
125000004433 nitrogen atom Chemical group N* 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Epidemiology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Ophthalmology & Optometry (AREA)
Psychiatry (AREA)
Hospice & Palliative Care (AREA)
Pain & Pain Management (AREA)
Child & Adolescent Psychology (AREA)
Diabetes (AREA)
Hematology (AREA)
Obesity (AREA)
Anesthesiology (AREA)
Pulmonology (AREA)
Immunology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

HU0102662A 1997-11-07 1998-11-05 Imidazoylalkyl substituted with a five, six or seven membered heterocyclic ring containing one nitrogen atom HUP0102662A3 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US96575497A	1997-11-07	1997-11-07
PCT/US1998/023224 WO1999024421A1 (en)	1997-11-07	1998-11-05	Imidazoylalkyl substituted with a five, six or seven membered heterocyclic ring containing one nitrogen atom

Publications (2)

Publication Number	Publication Date
HUP0102662A2 true HUP0102662A2 (en)	2001-12-28
HUP0102662A3 HUP0102662A3 (en)	2003-01-28

Family

ID=25510440

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
HU0102662A HUP0102662A3 (en)	1997-11-07	1998-11-05	Imidazoylalkyl substituted with a five, six or seven membered heterocyclic ring containing one nitrogen atom

Country Status (12)

Country	Link
EP (1)	EP1028956A1 (en)
JP (1)	JP2001522845A (en)
KR (1)	KR20010031839A (en)
CN (1)	CN1285828A (en)
AR (1)	AR016671A1 (en)
AU (1)	AU1296799A (en)
CA (1)	CA2309609A1 (en)
HU (1)	HUP0102662A3 (en)
IL (1)	IL135727A0 (en)
PE (1)	PE130699A1 (en)
WO (1)	WO1999024421A1 (en)
ZA (1)	ZA9810186B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6140337A (en) *	1997-12-23	2000-10-31	Schering Corporation	Methods for the treatment of mental disorders
FR2827863A1 (en) *	2001-07-27	2003-01-31	Sanofi Synthelabo	New dihydropyrrolyl alkyl imidazole derivatives having histamine receptor antagonist activity for treatment of obesity, diabetes, and central nervous system disorders
US7880017B2 (en)	2003-11-11	2011-02-01	Allergan, Inc.	Process for the synthesis of imidazoles
US7183305B2 (en)	2003-11-11	2007-02-27	Allergan, Inc.	Process for the synthesis of imidazoles
WO2005058823A1 (en) *	2003-12-17	2005-06-30	Takeda Pharmaceutical Company Limited	Urea derivative, process for producing the same, and use
NZ590148A (en) *	2004-12-30	2012-04-27	Janssen Pharmaceutica Nv	Piperazinyl and piperidinyl ureas as modulators of fatty acid amide hydrolase
UA108233C2 (en)	2010-05-03	2015-04-10		Fatty acid amide hydrolysis activity modulators
WO2013151982A1 (en)	2012-04-03	2013-10-10	Arena Pharmaceuticals, Inc.	Methods and compounds useful in treating pruritus, and methods for identifying such compounds
WO2022175384A1 (en) *	2021-02-17	2022-08-25	Fundación Universidad Católica De Valencia San Vicente Mártir	Small-molecule agents with antiviral activity against rna viruses

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
MX9207393A (en) *	1991-12-18	1994-06-30	Schering Corp	IMIDAZOIL OR RENT IMIDAZOIL SUBSTITUTED WITH A HETERO-CYCLE CHAIN OF FOUR OR FIVE MEMBERS CONTAINING NITROGEN.
ATE140223T1 (en) *	1991-12-18	1996-07-15	Schering Corp	IMIDOLYLALKYL DERIVATIVES SUBSTITUTED WITH A NITROGEN CONTAINING 6-MEMBED RING
AU7823894A (en) *	1993-08-27	1995-03-21	Vrije Universiteit	New imidazole derivatives having agonistic or antagonistic activity on the histamine h3 receptor
BR9711149A (en) *	1996-08-16	1999-08-17	Schering Corp	Treatment of allergic responses of the upper respiratory tract with a combination of histamine receptor antagonists

1998
- 1998-11-05 CN CN98812984A patent/CN1285828A/en active Pending
- 1998-11-05 KR KR1020007004911A patent/KR20010031839A/en not_active Application Discontinuation
- 1998-11-05 WO PCT/US1998/023224 patent/WO1999024421A1/en not_active Application Discontinuation
- 1998-11-05 HU HU0102662A patent/HUP0102662A3/en unknown
- 1998-11-05 AU AU12967/99A patent/AU1296799A/en not_active Abandoned
- 1998-11-05 IL IL13572798A patent/IL135727A0/en unknown
- 1998-11-05 EP EP98956443A patent/EP1028956A1/en not_active Withdrawn
- 1998-11-05 JP JP2000520435A patent/JP2001522845A/en not_active Withdrawn
- 1998-11-05 CA CA002309609A patent/CA2309609A1/en not_active Abandoned
- 1998-11-06 ZA ZA9810186A patent/ZA9810186B/en unknown
- 1998-11-06 PE PE1998001072A patent/PE130699A1/en not_active Application Discontinuation
- 1998-11-06 AR ARP980105620A patent/AR016671A1/en unknown

Also Published As

Publication number	Publication date
PE130699A1 (en)	1999-12-16
IL135727A0 (en)	2001-05-20
WO1999024421A1 (en)	1999-05-20
CA2309609A1 (en)	1999-05-20
WO1999024421A8 (en)	1999-08-26
ZA9810186B (en)	1999-05-06
KR20010031839A (en)	2001-04-16
HUP0102662A3 (en)	2003-01-28
AR016671A1 (en)	2001-07-25
AU1296799A (en)	1999-05-31
EP1028956A1 (en)	2000-08-23
JP2001522845A (en)	2001-11-20
CN1285828A (en)	2001-02-28

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