HUP0102313A3 - Imidazo pyridine derivatives, process for their preparation pharmaceutical compositions containing the same and intermediates - Google Patents

Imidazo pyridine derivatives, process for their preparation pharmaceutical compositions containing the same and intermediates

Info

Publication number: HUP0102313A3
Authority: HU; Hungary
Prior art keywords: intermediates; pharmaceutical compositions; same; compositions containing; pyridine derivatives
Prior art date: 1998-04-29

Application number

HU0102313A

Other languages

English (en)

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-04-29

Filing date

1999-04-23

Publication date

2002-10-28

1999-04-23 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2001-12-28 Publication of HUP0102313A2 publication Critical patent/HUP0102313A2/hu

2002-10-28 Publication of HUP0102313A3 publication Critical patent/HUP0102313A3/hu

Links

125000004857 imidazopyridinyl group Chemical class N1C(=NC2=C1C=CC=N2)* 0.000 title 1
239000000543 intermediate Substances 0.000 title 1
239000008194 pharmaceutical composition Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Nutrition Science (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

HU0102313A 1998-04-29 1999-04-23 Imidazo pyridine derivatives, process for their preparation pharmaceutical compositions containing the same and intermediates HUP0102313A3 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
SE9801526A SE9801526D0 (sv)	1998-04-29	1998-04-29	New compounds
PCT/SE1999/000662 WO1999055705A1 (en)	1998-04-29	1999-04-23	Imidazo pyridine derivatives which inhibit gastric acid secretion

Publications (2)

Publication Number	Publication Date
HUP0102313A2 HUP0102313A2 (hu)	2001-12-28
HUP0102313A3 true HUP0102313A3 (en)	2002-10-28

Family

ID=20411154

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
HU0102313A HUP0102313A3 (en)	1998-04-29	1999-04-23	Imidazo pyridine derivatives, process for their preparation pharmaceutical compositions containing the same and intermediates
HU0102425A HUP0102425A3 (en)	1998-04-29	1999-04-23	Imidazo pyridine derivatives which inhibit gastric acid secretion, process for producing them and pharmaceutical compositions containing them

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
HU0102425A HUP0102425A3 (en)	1998-04-29	1999-04-23	Imidazo pyridine derivatives which inhibit gastric acid secretion, process for producing them and pharmaceutical compositions containing them

Country Status (34)

Country	Link
US (2)	US6313137B1 (hu)
EP (4)	EP1073657B1 (hu)
JP (2)	JP3692034B2 (hu)
KR (3)	KR100595805B1 (hu)
CN (2)	CN1174980C (hu)
AR (2)	AR015769A1 (hu)
AT (4)	ATE307130T1 (hu)
AU (2)	AU769108B2 (hu)
BR (2)	BR9909995B1 (hu)
CA (2)	CA2329921A1 (hu)
CZ (2)	CZ293977B6 (hu)
DE (4)	DE69928792T2 (hu)
DK (2)	DK1073657T3 (hu)
EE (2)	EE04916B1 (hu)
ES (2)	ES2252975T3 (hu)
HK (5)	HK1033457A1 (hu)
HU (2)	HUP0102313A3 (hu)
ID (2)	ID27530A (hu)
IL (4)	IL139200A0 (hu)
IS (2)	IS5684A (hu)
MY (2)	MY121379A (hu)
NO (2)	NO317262B1 (hu)
NZ (2)	NZ507639A (hu)
PL (2)	PL195000B1 (hu)
RU (2)	RU2238271C2 (hu)
SA (2)	SA99200065B1 (hu)
SE (1)	SE9801526D0 (hu)
SI (1)	SI1073656T1 (hu)
SK (2)	SK285768B6 (hu)
TR (4)	TR200102728T2 (hu)
TW (2)	TWI250159B (hu)
UA (2)	UA66846C2 (hu)
WO (2)	WO1999055705A1 (hu)
ZA (2)	ZA200005797B (hu)

Families Citing this family (58)

* Cited by examiner, † Cited by third party
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US5840737A (en)	1996-01-04	1998-11-24	The Curators Of The University Of Missouri	Omeprazole solution and method for using same
US6489346B1 (en)	1996-01-04	2002-12-03	The Curators Of The University Of Missouri	Substituted benzimidazole dosage forms and method of using same
SE9802794D0 (sv) *	1998-08-21	1998-08-21	Astra Ab	New compounds
SE0003186D0 (sv) *	2000-09-07	2000-09-07	Astrazeneca Ab	New process
US6900324B2 (en)	2000-09-07	2005-05-31	Astrazeneca Ab	Process for preparing a substituted imidazopyridine compound
UA80393C2 (uk)	2000-12-07	2007-09-25	Алтана Фарма Аг	Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
SE0100295D0 (sv) *	2001-02-01	2001-02-01	Astrazeneca Ab	New compounds
SE0100297D0 (sv) *	2001-02-01	2001-02-01	Astrazeneca Ab	New compounds
SE0100296D0 (sv) *	2001-02-01	2001-02-01	Astrazeneca Ab	New compounds
KR20040058103A (ko) *	2001-02-13	2004-07-03	아스트라제네카 아베	신규 개질 방출 제제
IL157461A0 (en) *	2001-03-08	2004-03-28	Astrazeneca Ab Astrazeneca Ab	Use of carboxamido imidazo [1,2] pyridine deivatives in the preparation of medicaments for treating or preventing gastric ulcer
SE0102808D0 (sv) *	2001-08-22	2001-08-22	Astrazeneca Ab	New compounds
MY140561A (en) *	2002-02-20	2009-12-31	Nycomed Gmbh	Dosage form containing pde 4 inhibitor as active ingredient
SE0201939D0 (sv) *	2002-06-20	2002-06-20	Astrazeneca Ab	New combination
SE0201940D0 (sv) *	2002-06-20	2002-06-20	Astrazeneca Ab	New combination II
US6992080B2 (en)	2002-09-19	2006-01-31	Schering Corporation	Imidazopyridines as cyclin dependent kinase inhibitors
CN100384842C (zh)	2002-11-19	2008-04-30	奥坦纳医药公司	8-取代的咪唑并吡啶类化合物
AR043002A1 (es) *	2003-02-18	2005-07-13	Altana Pharma Ag	Imidazopirazinas 6-substituidos
CA2517256C (en) *	2003-02-26	2013-04-30	Sugen, Inc.	Aminoheteroaryl compounds as protein kinase inhibitors
EP1606261B1 (en)	2003-03-10	2009-11-04	Nycomed GmbH	Novel process for the preparation of roflumilast
SE525349C2 (sv) *	2003-06-23	2005-02-08	Volvo Penta Ab	Utombordsdrev för båtar
SE0301903D0 (sv) *	2003-06-26	2003-06-26	Astrazeneca Ab	Novel imidazopyridine compound III with therapeutic effect
SE0301905D0 (sv) *	2003-06-26	2003-06-26	Astrazeneca Ab	Novel imidazopyridine compound I with therapeutic effect
SE0301904D0 (sv) *	2003-06-26	2003-06-26	Astrazeneca Ab	Novel imidazopyridine compound II with therapeutic effect
US8993599B2 (en)	2003-07-18	2015-03-31	Santarus, Inc.	Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
CN1874772A (zh) *	2003-11-03	2006-12-06	阿斯利康(瑞典)有限公司	治疗隐匿性胃食管反流的咪唑并[1,2－a]吡啶衍生物
SE0303451D0 (sv) *	2003-12-18	2003-12-18	Astrazeneca Ab	New compounds
WO2005070927A2 (en) *	2004-01-26	2005-08-04	Altana Pharma Ag	1,2,4-triazolo[1,5-a] pyridines as gastric acid secretion inhibitors
US8906940B2 (en)	2004-05-25	2014-12-09	Santarus, Inc.	Pharmaceutical formulations useful for inhibiting acid secretion and methods for making and using them
EA011512B1 (ru) *	2004-12-17	2009-04-28	Ракуалиа Фарма Инк.	Производные хромана, полезные в качестве антагонистов кислотной помпы
EP1861074B1 (en)	2005-03-16	2013-04-24	Takeda GmbH	Taste masked dosage form containing roflumilast
US7666880B2 (en)	2005-03-21	2010-02-23	S*Bio Pte Ltd.	Imidazo[1,2-A]pyridine derivatives: preparation and pharmaceutical applications
CN101218238B (zh) *	2005-03-21	2011-10-26	S*Bio私人有限公司	咪唑并[1,2-a]吡啶衍生物：制备及药学应用
AR055321A1 (es) *	2005-03-24	2007-08-15	Glaxo Group Ltd	Compuestos de imidazopiridina uso para a fabricacion de un medicamento para el tratamiento o profilaxis de enfermedades o trastornos en los que se requiere un antagonista de una bomba de acido y composicion farmaceutica que lo comprende
GB0513423D0 (en) *	2005-06-30	2005-08-03	Glaxo Group Ltd	Novel compounds
WO2007066185A2 (en) *	2005-12-05	2007-06-14	Pfizer Products Inc.	Polymorphs of a c-met/hgfr inhibitor
PL1959955T3 (pl) *	2005-12-05	2011-04-29	Pfizer Prod Inc	Sposób traktowania nieprawidłowego wzrostu komórek
CA2645007A1 (en) *	2006-03-17	2007-09-27	Raqualia Pharma Inc.	Chromane derivatives
JP5571380B2 (ja)	2006-07-24	2014-08-13	ルミナスバイオサイエンシズ，インコーポレイテッド	オストワルド熟成を減少させた水不溶性の医薬品物質の固体ナノ粒子処方物
WO2008059373A1 (en) *	2006-11-17	2008-05-22	Raqualia Pharma Inc.	Imidazo [1, 2-a] pyrazine derivatives and their use as acid pump antagonists
EP1974729A1 (en) *	2007-03-28	2008-10-01	Santhera Pharmaceuticals (Schweiz) AG	Substituted imidazopyridine derivates as melanocortin- 4 receptor antagonists
US8513226B2 (en) *	2008-03-31	2013-08-20	Council Of Scientific And Industrial Research	Simultaneous method for the preparation of a mixture of 3-acetoxy-17-acetamido-16-formyl-androst-5,17-diene and 3-acetoxy-2'-chloro-5-androsteno[17,16-b]pyridine
AU2014201644B2 (en) *	2008-12-03	2015-05-21	Cinclus Pharma Holding AB (publ)	Imidazopyridine derivatives which inhibit the secretion of gastric acid
FI20086158A0 (fi) *	2008-12-03	2008-12-03	Mikael Dahlstroem	Imidatsopyridiinijohdannaiset
JP5802898B2 (ja) *	2009-07-09	2015-11-04	ラクオリア創薬株式会社	消化管運動異常が関与する疾患を治療するためのアシッドポンプ拮抗剤
EP3013345B1 (en) *	2013-06-25	2017-11-22	F. Hoffmann-La Roche AG	Compounds for treating spinal muscular atrophy
CA2933811C (en)	2013-12-16	2021-02-09	Asana Biosciences, Llc	P2x3 and/or p2x2/3 compounds and methods
KR20160135234A (ko) *	2014-03-24	2016-11-25	아르퀼 인코포레이티드	3-(3-(4-(1-아미노시클로부틸)페닐)-5-페닐-3h-이미다조[4,5-ｂ]피리딘-2-일)피리딘-2-아민의 제조 방법
CN106279151A (zh) *	2015-06-26	2017-01-04	江苏太瑞生诺生物医药科技有限公司	5-(2-(8-((2,6-二甲基苄基)氨基)-2,3-二甲基咪唑并[1,2-a]吡啶-6-甲酰胺基)乙氧基)-5-氧代戊酸的固体形式及其制备方法
KR101777971B1 (ko) *	2016-07-05	2017-09-12	제일약품주식회사	이미다조[1,2-a]피리딘 유도체, 이의 제조방법 및 이의 용도
KR20190057569A (ko) *	2017-11-20	2019-05-29	제일약품주식회사	7-아미노-1h-인돌-5-카르복사미드 유도체 및 이의 용도
WO2019152977A2 (en)	2018-02-05	2019-08-08	Bio-Rad Laboratories, Inc.	Chromatography resin having an anionic exchange-hydrophobic mixed mode ligand
EP3774719A1 (de) *	2018-04-10	2021-02-17	Bayer Aktiengesellschaft	Verfahren zur herstellung von 2,6-dialkylphenyl-essigsäuren
RU2732297C2 (ru) *	2018-11-14	2020-09-15	Общество с ограниченной ответственностью "Гурус БиоФарм"	Производные нестероидных противовоспалительных средств
MX2022005305A (es)	2019-11-04	2022-08-16	Cinclus Pharma Holding AB	Formulacion oral de x842.
AU2022381536A1 (en)	2021-11-05	2024-05-02	Cinclus Pharma Holding AB (publ)	Polymorphs of the hydrochloride salt of linaprazan glurate
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ZA81219B (en) *	1980-01-23	1982-01-27	Schering Corp	Imidazo (1,2-a) pyridines ,process for their preparation and pharmaceutical compositions containing them
EP0068378B1 (en)	1981-06-26	1986-03-05	Schering Corporation	Novel imidazo(1,2-a)pyridines and pyrazines, processes for their preparation and pharmaceutical compositions containing them
US4725601A (en)	1985-06-04	1988-02-16	Fujisawa Pharmaceutical Co., Ltd.	Certain imidazo[1,2-a]pyridines useful in the treatment of ulcers
EP0228006A1 (en) *	1985-12-16	1987-07-08	Fujisawa Pharmaceutical Co., Ltd.	Imidazopyridine compounds and processes for preparation thereof
GB8722488D0 (en) *	1987-09-24	1987-10-28	Fujisawa Pharmaceutical Co	Imidazopyridine compound

1998
- 1998-04-29 SE SE9801526A patent/SE9801526D0/xx unknown
1999
- 1999-04-16 TW TW088106128A patent/TWI250159B/zh not_active IP Right Cessation
- 1999-04-16 AR ARP990101777A patent/AR015769A1/es active IP Right Grant
- 1999-04-16 TW TW088106129A patent/TW490466B/zh not_active IP Right Cessation
- 1999-04-16 AR ARP990101776A patent/AR015768A1/es active IP Right Grant
- 1999-04-23 US US09/319,973 patent/US6313137B1/en not_active Expired - Fee Related
- 1999-04-23 CN CNB998077992A patent/CN1174980C/zh not_active Expired - Fee Related
- 1999-04-23 UA UA2000106034A patent/UA66846C2/uk unknown
- 1999-04-23 KR KR1020057022787A patent/KR100595805B1/ko not_active IP Right Cessation
- 1999-04-23 ES ES99947038T patent/ES2252975T3/es not_active Expired - Lifetime
- 1999-04-23 PL PL343801A patent/PL195000B1/pl not_active IP Right Cessation
- 1999-04-23 CZ CZ20003981A patent/CZ293977B6/cs not_active IP Right Cessation
- 1999-04-23 CZ CZ20003982A patent/CZ292567B6/cs not_active IP Right Cessation
- 1999-04-23 NZ NZ507639A patent/NZ507639A/en unknown
- 1999-04-23 RU RU2000127019/04A patent/RU2238271C2/ru active
- 1999-04-23 DE DE69928792T patent/DE69928792T2/de not_active Expired - Lifetime
- 1999-04-23 EE EEP200000664A patent/EE04916B1/xx not_active IP Right Cessation
- 1999-04-23 IL IL13920099A patent/IL139200A0/xx unknown
- 1999-04-23 TR TR2001/02728T patent/TR200102728T2/xx unknown
- 1999-04-23 WO PCT/SE1999/000662 patent/WO1999055705A1/en not_active Application Discontinuation
- 1999-04-23 BR BRPI9909995-0A patent/BR9909995B1/pt not_active IP Right Cessation
- 1999-04-23 SK SK1492-2000A patent/SK285768B6/sk not_active IP Right Cessation
- 1999-04-23 US US09/319,890 patent/US6313136B1/en not_active Expired - Fee Related
- 1999-04-23 CA CA002329921A patent/CA2329921A1/en not_active Abandoned
- 1999-04-23 UA UA2000106033A patent/UA67769C2/uk unknown
- 1999-04-23 IL IL13929799A patent/IL139297A0/xx active IP Right Grant
- 1999-04-23 AT AT99947037T patent/ATE307130T1/de not_active IP Right Cessation
- 1999-04-23 AU AU43006/99A patent/AU769108B2/en not_active Ceased
- 1999-04-23 DE DE69927803T patent/DE69927803T2/de not_active Expired - Lifetime
- 1999-04-23 EE EEP200000626A patent/EE04676B1/xx not_active IP Right Cessation
- 1999-04-23 HU HU0102313A patent/HUP0102313A3/hu unknown
- 1999-04-23 EP EP99947038A patent/EP1073657B1/en not_active Expired - Lifetime
- 1999-04-23 CA CA002329922A patent/CA2329922C/en not_active Expired - Fee Related
- 1999-04-23 TR TR2001/02612T patent/TR200102612T2/xx unknown
- 1999-04-23 BR BRPI9909996-9A patent/BR9909996B1/pt not_active IP Right Cessation
- 1999-04-23 ID IDW20002205A patent/ID27530A/id unknown
- 1999-04-23 AT AT99947038T patent/ATE312101T1/de not_active IP Right Cessation
- 1999-04-23 JP JP2000545865A patent/JP3692034B2/ja not_active Expired - Fee Related
- 1999-04-23 KR KR1020007012027A patent/KR100595806B1/ko not_active IP Right Cessation
- 1999-04-23 JP JP2000545864A patent/JP3883383B2/ja not_active Expired - Fee Related
- 1999-04-23 DK DK99947038T patent/DK1073657T3/da active
- 1999-04-23 EP EP04023091A patent/EP1491543B1/en not_active Expired - Lifetime
- 1999-04-23 AT AT04023091T patent/ATE372340T1/de not_active IP Right Cessation
- 1999-04-23 DE DE69937076T patent/DE69937076T2/de not_active Expired - Lifetime
- 1999-04-23 ES ES99947037T patent/ES2249913T3/es not_active Expired - Lifetime
- 1999-04-23 AU AU43007/99A patent/AU769190B2/en not_active Ceased
- 1999-04-23 WO PCT/SE1999/000663 patent/WO1999055706A1/en not_active Application Discontinuation
- 1999-04-23 ID IDW20002206A patent/ID26819A/id unknown
- 1999-04-23 HU HU0102425A patent/HUP0102425A3/hu unknown
- 1999-04-23 EP EP99947037A patent/EP1073656B1/en not_active Expired - Lifetime
- 1999-04-23 EP EP04023090A patent/EP1491542B1/en not_active Expired - Lifetime
- 1999-04-23 KR KR1020007012028A patent/KR100650472B1/ko not_active IP Right Cessation
- 1999-04-23 SI SI9930850T patent/SI1073656T1/sl unknown
- 1999-04-23 PL PL99343797A patent/PL343797A1/xx unknown
- 1999-04-23 TR TR2000/03176T patent/TR200003176T2/xx unknown
- 1999-04-23 RU RU2000127020/04A patent/RU2235725C2/ru active
- 1999-04-23 NZ NZ507638A patent/NZ507638A/en unknown
- 1999-04-23 SK SK1491-2000A patent/SK14912000A3/sk unknown
- 1999-04-23 AT AT04023090T patent/ATE372339T1/de not_active IP Right Cessation
- 1999-04-23 TR TR2000/03149T patent/TR200003149T2/xx unknown
- 1999-04-23 DE DE69937077T patent/DE69937077T2/de not_active Expired - Lifetime
- 1999-04-23 CN CNB998078026A patent/CN1165535C/zh not_active Expired - Fee Related
- 1999-04-23 DK DK99947037T patent/DK1073656T3/da active
- 1999-04-27 MY MYPI99001650A patent/MY121379A/en unknown
- 1999-04-27 MY MYPI99001649A patent/MY121389A/en unknown
- 1999-05-01 SA SA99200065A patent/SA99200065B1/ar unknown
- 1999-05-01 SA SA99200064A patent/SA99200064B1/ar unknown
2000
- 2000-10-18 ZA ZA200005797A patent/ZA200005797B/en unknown
- 2000-10-18 ZA ZA200005796A patent/ZA200005796B/en unknown
- 2000-10-23 IL IL139200A patent/IL139200A/en not_active IP Right Cessation
- 2000-10-25 IS IS5684A patent/IS5684A/is unknown
- 2000-10-25 IS IS5683A patent/IS5683A/is unknown
- 2000-10-26 IL IL139297A patent/IL139297A/en not_active IP Right Cessation
- 2000-10-27 NO NO20005450A patent/NO317262B1/no not_active IP Right Cessation
- 2000-10-27 NO NO20005451A patent/NO318203B1/no not_active IP Right Cessation
2001
- 2001-06-12 HK HK01104026A patent/HK1033457A1/xx not_active IP Right Cessation
- 2001-06-13 HK HK05103978A patent/HK1071139A1/xx not_active IP Right Cessation
- 2001-06-13 HK HK01104064A patent/HK1033317A1/xx not_active IP Right Cessation
- 2001-11-07 HK HK01107808A patent/HK1036981A1/xx not_active IP Right Cessation
- 2001-11-08 HK HK01107857A patent/HK1036984A1/xx not_active IP Right Cessation

Also Published As

Publication number	Publication date
DE69937076T2 (de)	2008-05-29
ATE372340T1 (de)	2007-09-15
NZ507638A (en)	2003-10-31
ZA200005796B (en)	2002-01-18
KR20010043133A (ko)	2001-05-25
HK1033317A1 (en)	2001-08-24
IL139297A (en)	2007-06-03
SA99200065B1 (ar)	2006-11-07
ID26819A (id)	2001-02-15
EP1073656A1 (en)	2001-02-07
CA2329922C (en)	2006-04-11
NO20005451L (no)	2000-12-27
BR9909996A (pt)	2000-12-26
IL139297A0 (en)	2001-11-25
KR20050121760A (ko)	2005-12-27
TR200102612T2 (tr)	2002-06-21
IS5684A (is)	2000-10-25
EE04916B1 (et)	2007-10-15
DE69937077D1 (de)	2007-10-18
HK1036984A1 (en)	2002-01-25
EP1073656B1 (en)	2005-10-19
HUP0102425A3 (en)	2002-12-28
NO20005450L (no)	2000-12-22
NO20005451D0 (no)	2000-10-27
AU4300699A (en)	1999-11-16
EP1491542A3 (en)	2005-01-05
SA99200064B1 (ar)	2006-10-11
HUP0102313A2 (hu)	2001-12-28
WO1999055705A1 (en)	1999-11-04
EP1491543B1 (en)	2007-09-05
CZ292567B6 (cs)	2003-10-15
TR200003176T2 (tr)	2001-03-21
ES2252975T3 (es)	2006-05-16
KR100595806B1 (ko)	2006-07-03
DK1073657T3 (da)	2006-03-13
PL343801A1 (en)	2001-09-10
SE9801526D0 (sv)	1998-04-29
TWI250159B (en)	2006-03-01
HUP0102425A2 (hu)	2001-11-28
ES2249913T3 (es)	2006-04-01
CA2329921A1 (en)	1999-11-04
IS5683A (is)	2000-10-25
DE69937076D1 (de)	2007-10-18
ID27530A (id)	2001-04-12
CZ20003982A3 (cs)	2001-02-14
DE69928792T2 (de)	2006-07-20
CN1306533A (zh)	2001-08-01
BR9909995A (pt)	2000-12-26
CZ20003981A3 (cs)	2001-03-14
AU4300799A (en)	1999-11-16
EE04676B1 (et)	2006-08-15
CN1307577A (zh)	2001-08-08
ATE307130T1 (de)	2005-11-15
HK1033457A1 (en)	2001-08-31
AR015768A1 (es)	2001-05-16
SK14912000A3 (sk)	2001-06-11
BR9909995B1 (pt)	2010-07-13
PL195000B1 (pl)	2007-07-31
EP1491542A2 (en)	2004-12-29
AU769190B2 (en)	2004-01-22
UA66846C2 (uk)	2004-06-15
SA99200065A (ar)	2005-12-03
EP1073657A1 (en)	2001-02-07
TW490466B (en)	2002-06-11
MY121379A (en)	2006-01-28
RU2238271C2 (ru)	2004-10-20
TR200003149T2 (tr)	2001-03-21
RU2235725C2 (ru)	2004-09-10
JP2002513024A (ja)	2002-05-08
UA67769C2 (uk)	2004-07-15
CN1165535C (zh)	2004-09-08
NO317262B1 (no)	2004-09-27
DK1073656T3 (da)	2006-01-16
HK1071139A1 (en)	2005-07-08
HK1036981A1 (en)	2002-01-25
DE69927803T2 (de)	2006-07-06
SI1073656T1 (sl)	2006-02-28
WO1999055706A1 (en)	1999-11-04
TR200102728T2 (tr)	2002-06-21
ATE312101T1 (de)	2005-12-15
US6313136B1 (en)	2001-11-06
PL343797A1 (en)	2001-09-10
CN1174980C (zh)	2004-11-10
EP1073657B1 (en)	2005-12-07
WO1999055706A9 (en)	2000-03-16
IL139200A (en)	2010-04-29
JP3692034B2 (ja)	2005-09-07
ATE372339T1 (de)	2007-09-15
KR20010043134A (ko)	2001-05-25
NZ507639A (en)	2004-01-30
CZ293977B6 (cs)	2004-09-15
EP1491543A1 (en)	2004-12-29
NO20005450D0 (no)	2000-10-27
DE69927803D1 (de)	2006-03-02
NO318203B1 (no)	2005-02-14
CA2329922A1 (en)	1999-11-04
DE69937077T2 (de)	2008-05-29
SK14922000A3 (sk)	2001-06-11
ZA200005797B (en)	2002-01-18
EE200000626A (et)	2002-04-15
AR015769A1 (es)	2001-05-16
BR9909996B1 (pt)	2010-08-24
KR100650472B1 (ko)	2006-11-28
DE69928792D1 (de)	2006-01-12
JP3883383B2 (ja)	2007-02-21
JP2002513025A (ja)	2002-05-08
US6313137B1 (en)	2001-11-06
KR100595805B1 (ko)	2006-07-03
EE200000664A (et)	2002-04-15
EP1491542B1 (en)	2007-09-05
AU769108B2 (en)	2004-01-15
IL139200A0 (en)	2001-11-25
SK285768B6 (sk)	2007-07-06
MY121389A (en)	2006-01-28

Legal Events

Date	Code	Title	Description
2011-02-28	FD9A	Lapse of provisional protection due to non-payment of fees

Publication	Publication Date	Title
HUP0102313A3 (en)	2002-10-28	Imidazo pyridine derivatives, process for their preparation pharmaceutical compositions containing the same and intermediates
HUP0104199A3 (en)	2002-12-28	Substituted pyrimido pyrimidinone derivatives, pharmaceutical compositions containing the same, process for the preparation thereof and intermediates
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HUP9700358A3 (en)	1999-08-30	New oxazolidinon derivatives, process for their preparation and pharmaceutical compositions containing them
HUP0203316A3 (en)	2004-07-28	Amino-triazolopyridine derivatives, process for their preparation and pharmaceutical compositions containing them
HUP9700328A3 (en)	1998-09-28	Heteroaryl-oxazolidinones, process for their preparation, pharmaceutical compositions containing the same, their use and intermediates
HUP0203052A3 (en)	2004-06-28	Bicyclic imidazo-3-yl-amine derivatives, process for their preparation, pharmaceutical compositions containing them and their use
HUP9601240A1 (en)	1997-09-29	Pyridin and pyrimidin derivatives, suitable as beta-adrenerg agonists, pharmaceutical compositions containing the same and their intermediates
HUP0001555A3 (en)	2001-01-29	Tetrahydro-imidazo-naphthyridine derivatives, pharmaceutical compositions thereof and process for their preparation
HUP0201516A2 (en)	2002-08-28	13-methyl-erythromycin derivatives, process for their preparation and pharmaceutical compositions containing them
HUP0000851A3 (en)	2002-04-29	Novel pyrimidine derivatives, processes for the preparation thereof and pharmaceutical compositions containing them
HUP0003748A3 (en)	2002-02-28	Halogen substituted tetracyclic tetrahydrofuran derivatives, process for their preparation their use and pharmaceutical compositions containing the same
HUP0203140A3 (en)	2004-06-28	Bicyclic imidazo-5-yl-amine derivatives, process for their preparation and pharmaceutical compositions containing them
HUP0201753A2 (en)	2002-09-28	Pyridopyranoazepine derivatives, process for their preparation and pharmaceutical compositions containing them
HUP0202075A3 (en)	2003-03-28	Substituted 2-dialkylaminoalkylbiphenyl derivatives, process for their preparation, pharmaceutical compositions containing them and their use
HUP0102215A3 (en)	2002-05-28	Benzoylpyridazines, pharmaceutical compositions containing the same and process for their preparation
HUP0203184A3 (en)	2004-12-28	Isoxazolecarboxamide derivatives, process for their preparation and pharmaceutical compositions containing them
HUP0003413A3 (en)	2003-11-28	New fused pyridine derivatives, process for their preparation and pharmaceutical compositions containing them