HU194891B - Process for production of 6-/trisubstituated-methil/-penicillane acid and its derivatives - Google Patents

Process for production of 6-/trisubstituated-methil/-penicillane acid and its derivatives Download PDF

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Publication number
HU194891B
HU194891B HU85759A HU75985A HU194891B HU 194891 B HU194891 B HU 194891B HU 85759 A HU85759 A HU 85759A HU 75985 A HU75985 A HU 75985A HU 194891 B HU194891 B HU 194891B
Authority
HU
Hungary
Prior art keywords
formula
hydrogen
compound
acid
ppm
Prior art date
Application number
HU85759A
Other languages
German (de)
English (en)
Hungarian (hu)
Other versions
HUT40443A (en
Inventor
Liang C Yuhpyng
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of HUT40443A publication Critical patent/HUT40443A/hu
Publication of HU194891B publication Critical patent/HU194891B/hu

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HU85759A 1984-01-30 1985-01-29 Process for production of 6-/trisubstituated-methil/-penicillane acid and its derivatives HU194891B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US57535484A 1984-01-30 1984-01-30

Publications (2)

Publication Number Publication Date
HUT40443A HUT40443A (en) 1986-12-28
HU194891B true HU194891B (en) 1988-03-28

Family

ID=24299979

Family Applications (2)

Application Number Title Priority Date Filing Date
HU85322A HU194567B (en) 1984-01-30 1985-01-29 Process for production of derivatives of 6-substituated methilen-penicillane acid
HU85759A HU194891B (en) 1984-01-30 1985-01-29 Process for production of 6-/trisubstituated-methil/-penicillane acid and its derivatives

Family Applications Before (1)

Application Number Title Priority Date Filing Date
HU85322A HU194567B (en) 1984-01-30 1985-01-29 Process for production of derivatives of 6-substituated methilen-penicillane acid

Country Status (15)

Country Link
JP (1) JPS61109791A (ru)
KR (1) KR880001029B1 (ru)
CS (5) CS248749B2 (ru)
DD (3) DD247677A5 (ru)
EG (1) EG16904A (ru)
ES (5) ES8604972A1 (ru)
FI (1) FI85376C (ru)
HU (2) HU194567B (ru)
IL (1) IL74190A (ru)
NO (1) NO165594C (ru)
PL (5) PL147514B1 (ru)
PT (1) PT79893B (ru)
SU (4) SU1395144A3 (ru)
YU (5) YU44770B (ru)
ZA (1) ZA85682B (ru)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY102312A (en) * 1987-01-27 1992-05-28 Pfizer 6-beta (substituted)-c-hydroxymethyl-penicillanic acids and derivatives thereof
ES2178301T3 (es) 1997-12-29 2002-12-16 Res Corp Technologies Inc Derivados del acido penicilanico 2-beta-sustituido-6-alquilideno como inhibidores de la beta-lactama.
US6407091B1 (en) 1999-04-15 2002-06-18 Research Corporation Technologies, Inc. β-lactamase inhibiting compounds
AU2002353768A1 (en) 2001-07-24 2003-03-18 Alamx, L.L.C. 7-alkylidene-3-substituted-3-cephem-4-carboxylates as beta-lactamase inhibitors.
AU2003224874A1 (en) 2002-04-04 2003-10-27 Alamx, L.L.C. INHIBITORS OF SERINE AND METALLO-ss-LACTAMASES
GB0711776D0 (en) * 2007-06-18 2007-07-25 Syngenta Participations Ag Substituted aromatic heterocyclic compounds as fungicides
JP6183053B2 (ja) * 2012-08-22 2017-08-23 宇部興産株式会社 テトラヒドロピラニルピリミジン化合物の製造方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4272439A (en) * 1978-06-02 1981-06-09 Schering Corporation 6-(Substituted-hydroxymethylene penams)
DE2927004A1 (de) * 1979-07-04 1981-05-27 Bayer Ag, 5090 Leverkusen Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel
US4287181A (en) * 1979-10-22 1981-09-01 Pfizer Inc. Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors

Also Published As

Publication number Publication date
YU44770B (en) 1991-02-28
ES539890A0 (es) 1986-02-16
FI85376B (fi) 1991-12-31
ES8700860A1 (es) 1986-11-16
CS248746B2 (en) 1987-02-12
PT79893A (en) 1985-02-01
YU119787A (en) 1988-04-30
ES548429A0 (es) 1987-04-16
PT79893B (en) 1987-02-03
SU1503683A3 (ru) 1989-08-23
KR880001029B1 (ko) 1988-06-15
PL256014A1 (en) 1986-12-02
YU44805B (en) 1991-02-28
CS248748B2 (en) 1987-02-12
ES8705451A1 (es) 1987-05-01
ES8604972A1 (es) 1986-02-16
CS248749B2 (en) 1987-02-12
ES548427A0 (es) 1987-05-01
PL149797B1 (en) 1990-03-31
YU14085A (en) 1987-12-31
HUT40443A (en) 1986-12-28
PL251750A1 (en) 1985-12-17
PL256013A1 (en) 1986-10-21
SU1396969A3 (ru) 1988-05-15
NO165594B (no) 1990-11-26
HU194567B (en) 1988-02-29
FI850375A0 (fi) 1985-01-29
PL145130B1 (en) 1988-08-31
YU44636B (en) 1990-10-31
HUT37799A (en) 1986-02-28
KR850005445A (ko) 1985-08-26
YU119587A (en) 1988-02-29
EG16904A (en) 1992-06-30
PL256015A1 (en) 1986-11-18
PL256016A1 (en) 1986-12-02
YU44635B (en) 1990-10-31
YU44634B (en) 1990-10-31
PL145990B1 (en) 1988-12-31
DD234015A5 (de) 1986-03-19
DD247677A5 (de) 1987-07-15
PL147514B1 (en) 1989-06-30
DD247678A5 (de) 1987-07-15
JPS61109791A (ja) 1986-05-28
YU119487A (en) 1988-02-29
ES548426A0 (es) 1986-11-16
FI850375L (fi) 1985-07-31
SU1395144A3 (ru) 1988-05-07
FI85376C (fi) 1992-04-10
YU119687A (en) 1988-04-30
ES8702916A1 (es) 1987-01-16
PL149242B1 (en) 1990-01-31
CS248747B2 (en) 1987-02-12
NO165594C (no) 1991-03-06
ES548428A0 (es) 1987-01-16
IL74190A0 (en) 1985-04-30
NO850350L (no) 1985-07-31
IL74190A (en) 1989-09-28
ES8704952A1 (es) 1987-04-16
ZA85682B (en) 1986-09-24
CS248733B2 (en) 1987-02-12
SU1508961A3 (ru) 1989-09-15

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Legal Events

Date Code Title Description
HU90 Patent valid on 900628
HMM4 Cancellation of final prot. due to non-payment of fee