HU194248B - Process for producing 2-azacycloalkyl-peneme derivatives and pharmaceutical compositions containing them - Google Patents
Process for producing 2-azacycloalkyl-peneme derivatives and pharmaceutical compositions containing them Download PDFInfo
- Publication number
- HU194248B HU194248B HU843830A HU383084A HU194248B HU 194248 B HU194248 B HU 194248B HU 843830 A HU843830 A HU 843830A HU 383084 A HU383084 A HU 383084A HU 194248 B HU194248 B HU 194248B
- Authority
- HU
- Hungary
- Prior art keywords
- methyl
- formula
- group
- compound
- oxazolidin
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Bestimmte 2-Azacycloalkylthio-2-penem-3-carbonsaeure-Verbindungen sind als antibakterielle Mittel zur Behandlung von Saeugern brauchbar und haben die Formeloder ein pharmazeutisch annehmbares Salz hiervon, worin RA Alkylen mit 2 bis 4 Kohlenstoffatomen, Alkylen mit 2 bis 4 Kohlenstoffatomen, worin ein Kohlenstoffatom einen Oxo-Substituenten hat, oder Alkylen mit 2 bis 4 Kohlenstoffatomen, worin eine Methylengruppe ersetzt ist durch Sauerstoff, S(O)m oder N-R3;B Carbonyl, Thiocarbonyl, Methylen oder Imin ist;R1 Wasserstoff ist oder eine Estergruppe bildet, die in vivo hydrolysiert wird;R2 Wasserstoff, Formyl, Alkylcarbonyl, N-Alkyl-aminocarbonyl, N-Alkylaminosulfonyl, Aminosulfonyl, Aminocarbonyl, Alkoxycarbonyl mit 2 bis 5 Kohlenstoffatomen, Alkylsulfonyl, Alkyl oder Alkyl substituiert durch Aminocarbonyl, Alkyl-S(O)m-, Hydroxyl, Amino, Alkylcarbonylamino, Formamido oder Alkylsulfonylamino, worin jedes Alkyl 1 bis 4 Kohlenstoffatome hat, ist;R3 Wasserstoff, Methyl, Formyl, Methylcarbonyl oder Methylsulfonyl ist;alk Alkylen mit 1 bis 4 Kohlenstoffatomen ist;n Null oder eins undm Null, eins oder zwei ist.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US54231083A | 1983-10-14 | 1983-10-14 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| HUT35264A HUT35264A (en) | 1985-06-28 |
| HU194248B true HU194248B (en) | 1988-01-28 |
Family
ID=24163252
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU843830A HU194248B (en) | 1983-10-14 | 1984-10-12 | Process for producing 2-azacycloalkyl-peneme derivatives and pharmaceutical compositions containing them |
Country Status (14)
| Country | Link |
|---|---|
| JP (1) | JPS60120881A (de) |
| KR (1) | KR870000525B1 (de) |
| DD (1) | DD223453A5 (de) |
| EG (1) | EG16589A (de) |
| ES (1) | ES536687A0 (de) |
| FI (1) | FI82250C (de) |
| HU (1) | HU194248B (de) |
| NO (1) | NO167573C (de) |
| PH (1) | PH20520A (de) |
| PL (1) | PL150059B1 (de) |
| PT (1) | PT79346B (de) |
| SU (1) | SU1340590A3 (de) |
| YU (1) | YU44241B (de) |
| ZA (1) | ZA847982B (de) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2660243B2 (ja) * | 1985-08-08 | 1997-10-08 | 株式会社半導体エネルギー研究所 | 半導体装置作製方法 |
| JPS6247116A (ja) * | 1985-08-26 | 1987-02-28 | Semiconductor Energy Lab Co Ltd | 半導体装置製造装置 |
| JPS6251210A (ja) * | 1985-08-30 | 1987-03-05 | Semiconductor Energy Lab Co Ltd | 半導体装置作製方法 |
| JPS6252924A (ja) * | 1985-09-01 | 1987-03-07 | Semiconductor Energy Lab Co Ltd | 半導体装置作製方法 |
| JPH0696580B2 (ja) * | 1985-09-17 | 1994-11-30 | 三共株式会社 | ペネム−３−カルボン酸誘導体 |
| JPS6269608A (ja) * | 1985-09-24 | 1987-03-30 | Semiconductor Energy Lab Co Ltd | 半導体装置作製方法 |
| JP2006001841A (ja) * | 2004-06-15 | 2006-01-05 | Sumitomo Chemical Co Ltd | 含窒素へテロ環化合物の製造方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS57176988A (en) * | 1981-04-09 | 1982-10-30 | Sankyo Co Ltd | Penam-3-carboxylic acid derivative and its preparation |
| JPS57200392A (en) * | 1981-06-03 | 1982-12-08 | Sankyo Co Ltd | Penem-3-carboxylic acid derivative and its preparation |
| DE3382761T2 (de) * | 1982-11-29 | 1995-03-09 | Schering Corp | Verfahren zur Herstellung von Penem-Verbindungen. |
| US4614738A (en) * | 1983-03-25 | 1986-09-30 | Schering Corporation | 2-(N-heterocycloaliphaticthio)penems |
-
1984
- 1984-10-10 YU YU1735/84A patent/YU44241B/xx unknown
- 1984-10-11 ES ES536687A patent/ES536687A0/es active Granted
- 1984-10-11 PT PT79346A patent/PT79346B/pt not_active IP Right Cessation
- 1984-10-12 DD DD84268285A patent/DD223453A5/de not_active IP Right Cessation
- 1984-10-12 NO NO844090A patent/NO167573C/no unknown
- 1984-10-12 FI FI844023A patent/FI82250C/fi not_active IP Right Cessation
- 1984-10-12 PH PH31330A patent/PH20520A/en unknown
- 1984-10-12 ZA ZA847982A patent/ZA847982B/xx unknown
- 1984-10-12 SU SU843804830A patent/SU1340590A3/ru active
- 1984-10-12 HU HU843830A patent/HU194248B/hu not_active IP Right Cessation
- 1984-10-13 EG EG628/84A patent/EG16589A/xx active
- 1984-10-13 KR KR1019840006347A patent/KR870000525B1/ko not_active IP Right Cessation
- 1984-10-15 JP JP59216022A patent/JPS60120881A/ja active Pending
- 1984-10-15 PL PL1984250031A patent/PL150059B1/pl unknown
Also Published As
| Publication number | Publication date |
|---|---|
| FI82250C (fi) | 1991-02-11 |
| YU44241B (en) | 1990-04-30 |
| JPS60120881A (ja) | 1985-06-28 |
| YU173584A (en) | 1987-02-28 |
| FI844023A0 (fi) | 1984-10-12 |
| PT79346A (en) | 1984-11-01 |
| PL250031A1 (en) | 1985-07-02 |
| ES8602012A1 (es) | 1985-11-16 |
| DD223453A5 (de) | 1985-06-12 |
| ZA847982B (en) | 1986-05-28 |
| PT79346B (en) | 1986-11-20 |
| SU1340590A3 (ru) | 1987-09-23 |
| EG16589A (en) | 1989-03-30 |
| ES536687A0 (es) | 1985-11-16 |
| FI82250B (fi) | 1990-10-31 |
| HUT35264A (en) | 1985-06-28 |
| NO167573B (no) | 1991-08-12 |
| KR870000525B1 (ko) | 1987-03-14 |
| PH20520A (en) | 1987-01-30 |
| NO844090L (no) | 1985-04-15 |
| KR850002987A (ko) | 1985-05-28 |
| NO167573C (no) | 1991-11-20 |
| FI844023L (fi) | 1985-04-15 |
| PL150059B1 (en) | 1990-04-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| HU90 | Patent valid on 900628 | ||
| HMM4 | Cancellation of final prot. due to non-payment of fee |