HK1215436A1 - 取代的 -甲基氨基甲酰基- -氟苯基氨基 四氫呋喃- -甲酸 變體 和其酯,其製備方法和用途 - Google Patents
取代的 -甲基氨基甲酰基- -氟苯基氨基 四氫呋喃- -甲酸 變體 和其酯,其製備方法和用途Info
- Publication number
- HK1215436A1 HK1215436A1 HK16103440.2A HK16103440A HK1215436A1 HK 1215436 A1 HK1215436 A1 HK 1215436A1 HK 16103440 A HK16103440 A HK 16103440A HK 1215436 A1 HK1215436 A1 HK 1215436A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- fluorophenylam
- methylcarbamoyl
- variants
- ester
- substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/04—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D307/18—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D307/24—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/10—Spiro-condensed systems
- C07D491/107—Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic System
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/0803—Compounds with Si-C or Si-Si linkages
- C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
- C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
RU2013108672/04A RU2520134C1 (ru) | 2013-02-27 | 2013-02-27 | Замещенные (r)-3-(4-метилкарбамоил-3-фторфениламино)-тетрагидро-фуран-3-енкарбоновые кислоты и их эфиры, способ их получения и применения |
PCT/RU2014/000122 WO2014133416A2 (ru) | 2013-02-27 | 2014-02-26 | Замещенная (r)-3-(4-метилкарбамоил-3-фторфениламино)тетрагидрофуран-3-енкарбоновая кислота (варианты) и ее эфир, способ получения и применения |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1215436A1 true HK1215436A1 (zh) | 2016-08-26 |
Family
ID=51216931
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK16103440.2A HK1215436A1 (zh) | 2013-02-27 | 2016-03-23 | 取代的 -甲基氨基甲酰基- -氟苯基氨基 四氫呋喃- -甲酸 變體 和其酯,其製備方法和用途 |
Country Status (11)
Country | Link |
---|---|
US (1) | US20160016925A1 (zh) |
EP (1) | EP2963026B1 (zh) |
JP (1) | JP6341939B2 (zh) |
KR (1) | KR102204267B1 (zh) |
CN (2) | CN105008340A (zh) |
AU (1) | AU2014221468B2 (zh) |
CA (1) | CA2901107C (zh) |
EA (1) | EA027369B1 (zh) |
HK (1) | HK1215436A1 (zh) |
RU (1) | RU2520134C1 (zh) |
WO (1) | WO2014133416A2 (zh) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
RU2557235C1 (ru) * | 2014-07-08 | 2015-07-20 | Александр Васильевич Иващенко | Замещенные 2-тиоксо-имидазолидин-4-оны и их спироаналоги, противораковый активный компонент, фармацевтическая композиция, лекарственный препарат, способ лечения рака простаты |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR101431407B1 (ko) * | 2005-05-13 | 2014-08-18 | 더 리전트 오브 더 유니버시티 오브 캘리포니아 | 디아릴히단토인 화합물 |
AU2007245022A1 (en) * | 2006-03-29 | 2007-11-08 | The Regents Of The University Of California | Diarylthiohydantoin compounds |
PE20081834A1 (es) * | 2006-12-31 | 2009-01-16 | Boehringer Ingelheim Int | Proceso para la sintesis de derivados de acido 3-amino-tetrahidrofuran-3-carboxilico y uso de los mismos como medicamentos |
WO2008119015A2 (en) * | 2007-03-27 | 2008-10-02 | Sloan-Kettering Institute For Cancer Research | Synthesis of thiohydantoins |
EP2416657A4 (en) * | 2009-04-09 | 2012-09-05 | Medivation Prostate Therapeutics Inc | COMPOUNDS COMPRISING SUBSTITUTED DI-ARYLHYDANTOIDS AND DI-ARYLTHIOHYDANTOINES AND METHODS OF USE THEREOF |
ES2671343T3 (es) | 2010-02-24 | 2018-06-06 | Medivation Prostate Therapeutics Llc | Procesos para la síntesis de compuestos de diariltiohidantoína y diarilhidantoína |
RU2434851C1 (ru) * | 2010-07-22 | 2011-11-27 | Александр Васильевич Иващенко | Циклические n, n'-диарилтиомочевины или n, n'-диарилмочевины - антагонисты андрогенных рецепторов, противораковое средство, способ получения и применения |
-
2013
- 2013-02-27 RU RU2013108672/04A patent/RU2520134C1/ru active IP Right Revival
-
2014
- 2014-02-26 AU AU2014221468A patent/AU2014221468B2/en active Active
- 2014-02-26 CA CA2901107A patent/CA2901107C/en active Active
- 2014-02-26 CN CN201480010767.0A patent/CN105008340A/zh active Pending
- 2014-02-26 WO PCT/RU2014/000122 patent/WO2014133416A2/ru active Application Filing
- 2014-02-26 EA EA201500754A patent/EA027369B1/ru unknown
- 2014-02-26 KR KR1020157026287A patent/KR102204267B1/ko active IP Right Grant
- 2014-02-26 US US14/828,540 patent/US20160016925A1/en not_active Abandoned
- 2014-02-26 EP EP14756865.3A patent/EP2963026B1/en active Active
- 2014-02-26 JP JP2015560137A patent/JP6341939B2/ja active Active
- 2014-02-26 CN CN201910962530.7A patent/CN110669027B/zh active Active
-
2016
- 2016-03-23 HK HK16103440.2A patent/HK1215436A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
CN105008340A (zh) | 2015-10-28 |
WO2014133416A3 (ru) | 2014-12-18 |
JP2016510025A (ja) | 2016-04-04 |
CA2901107A1 (en) | 2014-09-04 |
EP2963026A4 (en) | 2016-08-03 |
KR20150130327A (ko) | 2015-11-23 |
EP2963026B1 (en) | 2020-04-29 |
WO2014133416A2 (ru) | 2014-09-04 |
RU2520134C1 (ru) | 2014-06-20 |
WO2014133416A8 (ru) | 2015-09-11 |
KR102204267B1 (ko) | 2021-01-18 |
EA201500754A1 (ru) | 2016-01-29 |
CN110669027A (zh) | 2020-01-10 |
US20160016925A1 (en) | 2016-01-21 |
EP2963026A2 (en) | 2016-01-06 |
JP6341939B2 (ja) | 2018-06-13 |
CA2901107C (en) | 2020-10-27 |
AU2014221468A1 (en) | 2015-09-24 |
EA027369B1 (ru) | 2017-07-31 |
AU2014221468B2 (en) | 2018-05-17 |
CN110669027B (zh) | 2021-07-06 |
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